ES2018709B3 - Metodo para la preparacion de 1-oxoacetato de azetidinona por oxidacion del 2-hidroxiacetato correspondiente. - Google Patents
Metodo para la preparacion de 1-oxoacetato de azetidinona por oxidacion del 2-hidroxiacetato correspondiente.Info
- Publication number
- ES2018709B3 ES2018709B3 ES88302271T ES88302271T ES2018709B3 ES 2018709 B3 ES2018709 B3 ES 2018709B3 ES 88302271 T ES88302271 T ES 88302271T ES 88302271 T ES88302271 T ES 88302271T ES 2018709 B3 ES2018709 B3 ES 2018709B3
- Authority
- ES
- Spain
- Prior art keywords
- oxoacetate
- azetidinone
- chem
- preparation
- hydroxyacetate
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
Links
- 238000000034 method Methods 0.000 title abstract 2
- AEMRFAOFKBGASW-UHFFFAOYSA-M Glycolate Chemical compound OCC([O-])=O AEMRFAOFKBGASW-UHFFFAOYSA-M 0.000 title 1
- MNFORVFSTILPAW-UHFFFAOYSA-N azetidin-2-one Chemical compound O=C1CCN1 MNFORVFSTILPAW-UHFFFAOYSA-N 0.000 title 1
- 230000003647 oxidation Effects 0.000 title 1
- 238000007254 oxidation reaction Methods 0.000 title 1
- NUJOXMJBOLGQSY-UHFFFAOYSA-N manganese dioxide Chemical compound O=[Mn]=O NUJOXMJBOLGQSY-UHFFFAOYSA-N 0.000 abstract 2
- 125000004169 (C1-C6) alkyl group Chemical group 0.000 abstract 1
- -1 2-oxo-1-azetidinyl Chemical group 0.000 abstract 1
- 239000003242 anti bacterial agent Substances 0.000 abstract 1
- 125000003178 carboxy group Chemical group [H]OC(*)=O 0.000 abstract 1
- 125000002887 hydroxy group Chemical group [H]O* 0.000 abstract 1
- 238000004519 manufacturing process Methods 0.000 abstract 1
- 239000003960 organic solvent Substances 0.000 abstract 1
- 125000006239 protecting group Chemical group 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
- C07F7/02—Silicon compounds
- C07F7/08—Compounds having one or more C—Si linkages
- C07F7/18—Compounds having one or more C—Si linkages as well as one or more C—O—Si linkages
- C07F7/1804—Compounds having Si-O-C linkages
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Cephalosporin Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US07/028,380 US4751297A (en) | 1987-03-20 | 1987-03-20 | Method for preparation of azetidinone-1-oxoacetate by oxidation of the corresponding 2-hydroxyacetate |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES2018709B3 true ES2018709B3 (es) | 1991-05-01 |
Family
ID=21843131
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES88302271T Expired - Lifetime ES2018709B3 (es) | 1987-03-20 | 1988-03-16 | Metodo para la preparacion de 1-oxoacetato de azetidinona por oxidacion del 2-hidroxiacetato correspondiente. |
Country Status (9)
| Country | Link |
|---|---|
| US (1) | US4751297A (es) |
| EP (1) | EP0283253B1 (es) |
| JP (1) | JPS63258455A (es) |
| AT (1) | ATE58376T1 (es) |
| DE (1) | DE3861034D1 (es) |
| DK (1) | DK148188A (es) |
| ES (1) | ES2018709B3 (es) |
| GR (1) | GR3002531T3 (es) |
| PT (1) | PT87000B (es) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5191077A (en) * | 1987-05-11 | 1993-03-02 | Pfizer Inc. | Diastereomeric 5R,6S-6-(1R-hydroxyethyl)-2-(cis-1-oxo-3-thiolanylthio)-2-penem-3-carboxylic acids |
| US4895940A (en) * | 1988-10-19 | 1990-01-23 | Pfizer Inc. | Process for the preparation of penems |
| US5191075A (en) * | 1988-10-19 | 1993-03-02 | Pfizer Inc | Process for the preparation of penems |
| US4992543A (en) * | 1988-10-19 | 1991-02-12 | Pfizer Inc. | Penem derivatives |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE2624822A1 (de) * | 1976-05-31 | 1977-12-15 | Schering Ag | Benzodioxolderivate, verfahren zur herstellung dieser verbindungen sowie diese enthaltende herbizide mittel |
| EP0042026B1 (de) * | 1978-02-02 | 1986-01-08 | Ciba-Geigy Ag | 3,4-Disubstituierte Azetidin-2-onverbindungen und Verfahren zu ihrer Herstellung |
| HU196412B (en) * | 1981-03-23 | 1988-11-28 | Pfizer | Process for production of penicillin-acid-penicillakiroloximethil-esthers |
| JPS58198486A (ja) * | 1982-05-14 | 1983-11-18 | Sankyo Co Ltd | ペネムまたはカルバペネム−３−カルボン酸誘導体およびその製法 |
| US4619924A (en) * | 1984-05-18 | 1986-10-28 | Pfizer Inc. | 2-alkylthiopenem derivatives |
| US4695626A (en) * | 1986-07-29 | 1987-09-22 | Pfizer Inc. | 1-aza-4,5-dithiabicyclo [4.2.0] oct-2-en-8-one-2 carboxylate esters |
-
1987
- 1987-03-20 US US07/028,380 patent/US4751297A/en not_active Expired - Lifetime
-
1988
- 1988-03-16 AT AT88302271T patent/ATE58376T1/de active
- 1988-03-16 DE DE8888302271T patent/DE3861034D1/de not_active Expired - Lifetime
- 1988-03-16 ES ES88302271T patent/ES2018709B3/es not_active Expired - Lifetime
- 1988-03-16 EP EP88302271A patent/EP0283253B1/en not_active Expired - Lifetime
- 1988-03-17 JP JP63064637A patent/JPS63258455A/ja active Pending
- 1988-03-17 PT PT87000A patent/PT87000B/pt not_active IP Right Cessation
- 1988-03-18 DK DK148188A patent/DK148188A/da not_active Application Discontinuation
-
1990
- 1990-11-15 GR GR90400885T patent/GR3002531T3/el unknown
Also Published As
| Publication number | Publication date |
|---|---|
| PT87000B (pt) | 1992-06-30 |
| PT87000A (pt) | 1988-04-01 |
| US4751297A (en) | 1988-06-14 |
| DK148188D0 (da) | 1988-03-18 |
| EP0283253B1 (en) | 1990-11-14 |
| GR3002531T3 (en) | 1993-01-25 |
| JPS63258455A (ja) | 1988-10-25 |
| EP0283253A1 (en) | 1988-09-21 |
| ATE58376T1 (de) | 1990-11-15 |
| DK148188A (da) | 1988-09-21 |
| DE3861034D1 (de) | 1990-12-20 |
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