ES2001682A6 - Nuevo procedimiento para la preparacion de derivados 1,4-perhidrotiazepina - Google Patents

Nuevo procedimiento para la preparacion de derivados 1,4-perhidrotiazepina

Info

Publication number
ES2001682A6
ES2001682A6 ES8601893A ES8601893A ES2001682A6 ES 2001682 A6 ES2001682 A6 ES 2001682A6 ES 8601893 A ES8601893 A ES 8601893A ES 8601893 A ES8601893 A ES 8601893A ES 2001682 A6 ES2001682 A6 ES 2001682A6
Authority
ES
Spain
Prior art keywords
compound
formula
carboxyl
protecting group
perhydro
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES8601893A
Other languages
English (en)
Inventor
Hiroaki Yanagisawa
Sadao Ishihara
Akiko Ando
Takuro Kanazaki
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Sankyo Co Ltd
Original Assignee
Sankyo Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sankyo Co Ltd filed Critical Sankyo Co Ltd
Publication of ES2001682A6 publication Critical patent/ES2001682A6/es
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D281/00—Heterocyclic compounds containing rings of more than six members having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D281/02—Seven-membered rings
    • C07D281/04—Seven-membered rings having the hetero atoms in positions 1 and 4
    • C07D281/06—Seven-membered rings having the hetero atoms in positions 1 and 4 not condensed with other rings
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

NUEVO PROCEDIMIENTO PARA LA PREPARACION DE DERIVADOS DE 1,4-PERHIDROTIAZEPINA. LOS COMPUESTOS (I) EN LOS QUE R1, R2, R3, R4 Y R5 REPRESENTAN VARIOS RADICALES ORGANICOS SE OBTIENEN POR REACCION DE (II) CON (III) PARA DAR UN COMPUESTO (IV) QUE SE HACE REACCIONAR CON (V) PARA DAR (VI), SEGUIDO OPCIONALMENTE DE SEPARACION DE GRUPOS PROTECTORES, SOLIDIFICACION Y/O ESTERIFICACION. LOS COMPUESTOS (I) TIENEN UNA VALIOSA ACTIVIDAD INHIBIDORA DE ECA, SIENDO UTILES COMO AGENTES ANTIHIPERTENSIVOS.
ES8601893A 1985-09-12 1986-09-12 Nuevo procedimiento para la preparacion de derivados 1,4-perhidrotiazepina Expired ES2001682A6 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP20216485 1985-09-12

Publications (1)

Publication Number Publication Date
ES2001682A6 true ES2001682A6 (es) 1988-06-01

Family

ID=16453016

Family Applications (1)

Application Number Title Priority Date Filing Date
ES8601893A Expired ES2001682A6 (es) 1985-09-12 1986-09-12 Nuevo procedimiento para la preparacion de derivados 1,4-perhidrotiazepina

Country Status (4)

Country Link
JP (1) JPH07113020B2 (es)
KR (1) KR910005688B1 (es)
CA (1) CA1332943C (es)
ES (1) ES2001682A6 (es)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN1585744A (zh) * 2001-03-27 2005-02-23 兰贝克赛实验室有限公司 贝那普利的制备方法
GB2423085C (en) * 2005-02-11 2011-11-09 Cambridge Entpr Ltd Ligands for G-protein coupled receptors
JP5450927B2 (ja) * 2007-02-26 2014-03-26 ダイト株式会社 塩酸テモカプリルのｉ型結晶の製造方法

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4460579A (en) * 1983-02-28 1984-07-17 E. R. Squibb & Sons, Inc. Thiazine and thiazepine containing compounds

Also Published As

Publication number Publication date
KR870003079A (ko) 1987-04-15
JPS62161775A (ja) 1987-07-17
CA1332943C (en) 1994-11-08
KR910005688B1 (ko) 1991-08-02
JPH07113020B2 (ja) 1995-12-06

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Legal Events

Date Code Title Description
SA6 Expiration date (snapshot 920101)

Free format text: 2006-09-12

FD1A Patent lapsed

Effective date: 20060913