EP3024446A1 - Formulation comprenant un agent hypolipidémiant - Google Patents

Formulation comprenant un agent hypolipidémiant

Info

Publication number
EP3024446A1
EP3024446A1 EP14787059.6A EP14787059A EP3024446A1 EP 3024446 A1 EP3024446 A1 EP 3024446A1 EP 14787059 A EP14787059 A EP 14787059A EP 3024446 A1 EP3024446 A1 EP 3024446A1
Authority
EP
European Patent Office
Prior art keywords
pharmaceutical composition
sodium
formula
formulation
calcium
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
EP14787059.6A
Other languages
German (de)
English (en)
Inventor
Jitendre D. PATEL
Prakash DAVADRA
Snehal Patel
Shafiq Sheikh
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Zydus Lifesciences Ltd
Original Assignee
Cadila Healthcare Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Cadila Healthcare Ltd filed Critical Cadila Healthcare Ltd
Publication of EP3024446A1 publication Critical patent/EP3024446A1/fr
Withdrawn legal-status Critical Current

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2009—Inorganic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics

Abstract

La présente invention concerne une composition pharmaceutique stable d'un agent hypolipidémiant approprié. De préférence, la présente invention décrit de nouvelles formulations du composé de formule (I), ou des sels pharmaceutiquement acceptables de composés de formule (1). Plus particulièrement, la présente invention concerne la composition pharmaceutique stable de composés de formule (I), comprenant des composés de formule (I) ou ses sels pharmaceutiquement acceptables, le pH de la formulation étant maintenu au-dessus de 7. Formule (I)
EP14787059.6A 2013-07-25 2014-07-24 Formulation comprenant un agent hypolipidémiant Withdrawn EP3024446A1 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IN2470MU2013 IN2013MU02470A (fr) 2013-07-25 2013-07-25
PCT/IN2014/000489 WO2015011730A1 (fr) 2013-07-25 2014-07-24 Formulation comprenant un agent hypolipidémiant

Publications (1)

Publication Number Publication Date
EP3024446A1 true EP3024446A1 (fr) 2016-06-01

Family

ID=51787141

Family Applications (1)

Application Number Title Priority Date Filing Date
EP14787059.6A Withdrawn EP3024446A1 (fr) 2013-07-25 2014-07-24 Formulation comprenant un agent hypolipidémiant

Country Status (21)

Country Link
US (2) US9610277B2 (fr)
EP (1) EP3024446A1 (fr)
JP (1) JP2016523895A (fr)
KR (1) KR101786843B1 (fr)
CN (1) CN105407873A (fr)
AP (1) AP2015008876A0 (fr)
AR (1) AR097067A1 (fr)
AU (1) AU2014294548B2 (fr)
BR (1) BR112015031878A2 (fr)
CA (1) CA2917923A1 (fr)
EA (1) EA201690072A1 (fr)
HK (1) HK1219222A1 (fr)
IN (1) IN2013MU02470A (fr)
MA (1) MA38865A1 (fr)
MX (1) MX2015016971A (fr)
NZ (1) NZ714558A (fr)
PH (1) PH12015502802A1 (fr)
SG (1) SG11201509798PA (fr)
TW (1) TW201545773A (fr)
WO (1) WO2015011730A1 (fr)
ZA (1) ZA201508682B (fr)

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CN101427486B (zh) 2006-05-23 2013-06-19 英特尔公司 具有定向天线和一个或多个毫米波反射器的毫米波通信系统
UA110813C2 (uk) 2011-01-31 2016-02-25 Каділа Хелткере Лімітед Лікування ліподистрофії
EP2988736A1 (fr) 2013-04-22 2016-03-02 Cadila Healthcare Limited Nouvelle composition pour la stéatose hépatique non alcoolique (nafld)
EP3004053B1 (fr) 2013-05-30 2021-03-24 Cadila Healthcare Limited Procédé de préparation de pyrroles présentant des activités hypocholestérolémiques hypolipidémiques
TW201636015A (zh) 2013-07-05 2016-10-16 卡地拉保健有限公司 協同性組成物
IN2013MU02470A (fr) 2013-07-25 2015-06-26 Cadila Healthcare Ltd
WO2015033357A2 (fr) 2013-09-06 2015-03-12 Cadila Healthcare Limited Procédé amélioré de préparation de dérivés de pyrrole
US10385017B2 (en) 2015-10-14 2019-08-20 Cadila Healthcare Limited Pyrrole compound, compositions and process for preparation thereof
KR101913830B1 (ko) * 2016-12-05 2018-10-31 주식회사 코쿤디자인 기능성 led 어셈블리를 이용한 디스플레이 장치
US20180243263A1 (en) 2016-12-09 2018-08-30 Cadila Healthcare Ltd. Treatment for primary biliary cholangitis
US20220175721A1 (en) * 2019-02-13 2022-06-09 Cadila Healthcare Limited Treatment for polycystic ovarian syndrome (pcos)
US20220169603A1 (en) * 2019-03-11 2022-06-02 Cadila Healthcare Ltd. Novel salts, crystalline forms and premix of hypolipidemic agent

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UA110813C2 (uk) * 2011-01-31 2016-02-25 Каділа Хелткере Лімітед Лікування ліподистрофії
EP2988736A1 (fr) 2013-04-22 2016-03-02 Cadila Healthcare Limited Nouvelle composition pour la stéatose hépatique non alcoolique (nafld)
EP3004053B1 (fr) 2013-05-30 2021-03-24 Cadila Healthcare Limited Procédé de préparation de pyrroles présentant des activités hypocholestérolémiques hypolipidémiques
TW201636015A (zh) 2013-07-05 2016-10-16 卡地拉保健有限公司 協同性組成物
IN2013MU02470A (fr) 2013-07-25 2015-06-26 Cadila Healthcare Ltd
WO2015029066A1 (fr) 2013-08-29 2015-03-05 Cadila Healthcare Limited Forme polymorphe de dérivé du pyrrole et intermédiaire
WO2015033357A2 (fr) 2013-09-06 2015-03-12 Cadila Healthcare Limited Procédé amélioré de préparation de dérivés de pyrrole

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Also Published As

Publication number Publication date
WO2015011730A1 (fr) 2015-01-29
BR112015031878A2 (pt) 2017-07-25
AU2014294548A1 (en) 2015-12-17
AU2014294548B2 (en) 2017-08-10
MX2015016971A (es) 2016-04-25
US10098868B2 (en) 2018-10-16
TW201545773A (zh) 2015-12-16
US20160136131A1 (en) 2016-05-19
IN2013MU02470A (fr) 2015-06-26
US20170266158A1 (en) 2017-09-21
AR097067A1 (es) 2016-02-17
CA2917923A1 (fr) 2015-01-29
PH12015502802A1 (en) 2016-03-14
CN105407873A (zh) 2016-03-16
NZ714558A (en) 2017-02-24
EA201690072A1 (ru) 2016-06-30
MA38865A1 (fr) 2017-12-29
US9610277B2 (en) 2017-04-04
KR101786843B1 (ko) 2017-10-18
AP2015008876A0 (en) 2015-11-30
JP2016523895A (ja) 2016-08-12
SG11201509798PA (en) 2016-02-26
HK1219222A1 (zh) 2017-03-31
ZA201508682B (en) 2017-03-29
KR20160013150A (ko) 2016-02-03

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