EP2089366A2 - Derives du 3-pyrazolone et/ou 3-pyridazinone en tant qu'inhibiteurs de lysyl oxidase - Google Patents

Derives du 3-pyrazolone et/ou 3-pyridazinone en tant qu'inhibiteurs de lysyl oxidase

Info

Publication number
EP2089366A2
EP2089366A2 EP05818002A EP05818002A EP2089366A2 EP 2089366 A2 EP2089366 A2 EP 2089366A2 EP 05818002 A EP05818002 A EP 05818002A EP 05818002 A EP05818002 A EP 05818002A EP 2089366 A2 EP2089366 A2 EP 2089366A2
Authority
EP
European Patent Office
Prior art keywords
turbocharger
passage
insert
housing according
main body
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
EP05818002A
Other languages
German (de)
English (en)
Inventor
Erfindernennung liegt noch nicht vor Die
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Individual
Original Assignee
Individual
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Individual filed Critical Individual
Publication of EP2089366A2 publication Critical patent/EP2089366A2/fr
Withdrawn legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Supercharger (AREA)

Abstract

La présente invention se rapporte à un logement de turbocompresseur, qui comprend un corps principal (1) destiné à supporter un arbre (2) portant une roue de turbine et une roue de compresseur (3), et une partie joint (4) permettant d'assurer l'étanchéité de l'espace existant entre l'arbre (2) et le logement de turbocompresseur. L'on forme la partie joint (4) en montant une garniture (5) sur le corps principal (1), ladite garniture (5) étant dotée d'un passage (6, 7) destiné à fournir un fluide à ladite partie joint (4).
EP05818002A 2004-11-22 2005-11-20 Derives du 3-pyrazolone et/ou 3-pyridazinone en tant qu'inhibiteurs de lysyl oxidase Withdrawn EP2089366A2 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE102004056226A DE102004056226A1 (de) 2004-11-22 2004-11-22 Neuartige Inhibitoren der Lysyloxidase
PCT/DE2005/002086 WO2006053555A2 (fr) 2004-11-22 2005-11-20 Nouveaux inhibiteurs de la lysyloxydase

Publications (1)

Publication Number Publication Date
EP2089366A2 true EP2089366A2 (fr) 2009-08-19

Family

ID=36177758

Family Applications (1)

Application Number Title Priority Date Filing Date
EP05818002A Withdrawn EP2089366A2 (fr) 2004-11-22 2005-11-20 Derives du 3-pyrazolone et/ou 3-pyridazinone en tant qu'inhibiteurs de lysyl oxidase

Country Status (3)

Country Link
EP (1) EP2089366A2 (fr)
DE (2) DE102004056226A1 (fr)
WO (1) WO2006053555A2 (fr)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP3265456B1 (fr) * 2015-03-06 2020-11-18 Pharmakea, Inc. Inhibiteurs fluorés de la lysyl oxydase-like 2 et utilisations desdits inhibiteurs
EP3265445B1 (fr) 2015-03-06 2021-05-05 Pharmakea, Inc. Inhibiteurs de la lysyl oxydase-like 2 et utilisations desdits inhibiteurs
WO2017003862A1 (fr) * 2015-07-01 2017-01-05 Pharmakea, Inc. Inhibiteurs de lysyl oxydase-like 2 et utilisations desdits inhibiteurs
CA3013917A1 (fr) 2016-02-09 2017-08-17 Pharmakea, Inc. Inhibiteurs quinolinone de la lysyl oxydase-like 2 et utilisations desdits inhibiteurs
GB201602934D0 (en) 2016-02-19 2016-04-06 Cancer Res Inst Royal Compounds
MX2019002612A (es) 2016-09-07 2019-08-21 Pharmakea Inc Usos de un inhibidor de lisil-oxidasa tipo 2.
CA3036064A1 (fr) 2016-09-07 2018-03-15 Pharmakea, Inc. Formes cristallines d'un inhibiteur de lysyl oxydase de type 2 et leurs procedes de fabrication
GB201809295D0 (en) 2018-06-06 2018-07-25 Institute Of Cancer Res Royal Cancer Hospital Lox inhibitors
CA3105599A1 (fr) 2018-08-03 2020-02-06 Pharmaxis Ltd. Inhibiteurs de lysyl oxydases derives d'halogenoallylamine sulfone et utilisations associees
GB201818750D0 (en) 2018-11-16 2019-01-02 Institute Of Cancer Res Royal Cancer Hospital Lox inhibitors
US12018015B2 (en) 2021-06-18 2024-06-25 Aligos Therapeutics, Inc. Methods and compositions for targeting PD-L1

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5328913A (en) * 1992-12-11 1994-07-12 Duke University Minoxidil analogs as inhibitors of cell proliferation and lysyl hydroxylase
KR100657189B1 (ko) * 1998-08-14 2006-12-14 니혼노야쿠가부시키가이샤 피리다지논 유도체 및 이를 함유하는 의약 조성물
DE10216144A1 (de) * 2002-04-12 2003-11-06 Bayer Ag Substituierte 2-Phenyl-3(2H)-Pyridazinone

Also Published As

Publication number Publication date
WO2006053555A3 (fr) 2006-07-27
DE102004056226A1 (de) 2006-05-24
DE112005003431A5 (de) 2007-10-31
WO2006053555A2 (fr) 2006-05-26

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Inventor name: BURCHARDT, ELMAR REINHOLD, DR. DR.

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