EE200100611A - New pharmaceutical combinations of NOS inhibitors - Google Patents

New pharmaceutical combinations of NOS inhibitors

Info

Publication number
EE200100611A
EE200100611A EEP200100611A EEP200100611A EE200100611A EE 200100611 A EE200100611 A EE 200100611A EE P200100611 A EEP200100611 A EE P200100611A EE P200100611 A EEP200100611 A EE P200100611A EE 200100611 A EE200100611 A EE 200100611A
Authority
EE
Estonia
Prior art keywords
pharmaceutical combinations
new pharmaceutical
nos inhibitors
inhibitors
nos
Prior art date
Application number
EEP200100611A
Other languages
Estonian (et)
Inventor
David Saltarelli Mario
Adams Lowe John Iii
Original Assignee
Pfizer Products Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Products Inc. filed Critical Pfizer Products Inc.
Publication of EE200100611A publication Critical patent/EE200100611A/en

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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • AHUMAN NECESSITIES
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    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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    • AHUMAN NECESSITIES
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    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/135Amines having aromatic rings, e.g. ketamine, nortriptyline
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    • A61K31/13Amines
    • A61K31/135Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/138Aryloxyalkylamines, e.g. propranolol, tamoxifen, phenoxybenzamine
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    • A61K31/13Amines
    • A61K31/15Oximes (>C=N—O—); Hydrazines (>N—N<); Hydrazones (>N—N=) ; Imines (C—N=C)
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    • A61K31/34Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide
    • A61K31/343Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide condensed with a carbocyclic ring, e.g. coumaran, bufuralol, befunolol, clobenfurol, amiodarone
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    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
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  • Emergency Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
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EEP200100611A 1999-05-21 2000-03-16 New pharmaceutical combinations of NOS inhibitors EE200100611A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US13552099P 1999-05-21 1999-05-21
PCT/IB2000/000295 WO2000071107A2 (en) 1999-05-21 2000-03-16 New pharmaceutical combinations for nos inhibitors

Publications (1)

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DE10001785A1 (en) * 2000-01-18 2001-07-19 Boehringer Ingelheim Pharma Use of NK-1 receptor antagonists for treatment of restless legs syndrome
GB0019006D0 (en) * 2000-08-04 2000-09-20 Astrazeneca Ab Novel compounds
US20030045449A1 (en) * 2001-08-15 2003-03-06 Pfizer, Inc. Pharmaceutical combinations for the treatment of neurodegenerative diseases
DOP2002000467A (en) * 2001-10-10 2003-04-15 Pfizer Prod Inc 2-AMINO-6 (PHENYL REPLACED IN POSITIONS 2,4,5) -PIRIDINES
US6803470B2 (en) * 2001-10-10 2004-10-12 Pfizer Inc 2-amino-6-(2,4,5-substituted-phenyl)-pyridines
US7407970B2 (en) * 2003-06-24 2008-08-05 Neurosearch A/S 8-aza-bicyclo[3.2.1]octane derivatives and their use as monoamine neurotransmitter re-uptake inhibitors
EP1634598A1 (en) * 2004-09-07 2006-03-15 Laboratorios Del Dr. Esteve, S.A. Use of piperazine derivatives and analogues for the manufacture of a medicament for the prophylaxis and/or treatment of disorders of food ingestion
CA2687912C (en) 2007-06-08 2015-11-03 Janssen Pharmaceutica N.V. Piperidine/piperazine derivatives
CA2687754C (en) 2007-06-08 2015-12-08 Janssen Pharmaceutica N.V. Piperidine, piperazine derivatives for use as dgat inhibitors
US8633197B2 (en) 2007-06-08 2014-01-21 Janssen Pharmaceutica N.V. Piperidine/piperazine derivatives
JO2972B1 (en) 2007-06-08 2016-03-15 جانسين فارماسوتيكا ان. في Piperidine/Piperazine derivatives
UY31863A (en) 2008-06-05 2010-01-05 Janssen Pharmaceutica Nv DRUG COMBINATIONS UNDERSTANDING A DGAT INHIBITOR AND A PPAR AGONIST
WO2010101246A1 (en) * 2009-03-05 2010-09-10 塩野義製薬株式会社 Piperidine and pyrrolidine derivatives having npy y5 receptor antagonism
WO2014078568A1 (en) 2012-11-14 2014-05-22 The Johns Hopkins University Methods and compositions for treating schizophrenia
AU2020291468A1 (en) * 2019-06-14 2022-01-06 Srx Cardio, Llc Compounds for the modulation of proprotein convertase subtilisin/kexin type 9 (PCSK9)

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TNSN00106A1 (en) 2005-11-10
GT200000071A (en) 2001-11-08
CA2374668A1 (en) 2000-11-30
PL358538A1 (en) 2004-08-09
CN1617743A (en) 2005-05-18
OA11943A (en) 2006-04-12
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BR0010820A (en) 2002-03-05
IL145955A0 (en) 2002-07-25
TR200103351T2 (en) 2002-06-21
CO5160295A1 (en) 2002-05-30
EA200101110A1 (en) 2002-08-29
NO20015651D0 (en) 2001-11-20
UY26148A1 (en) 2000-12-29
PA8494601A1 (en) 2002-08-29
AP2001002326A0 (en) 2001-12-31
IS6126A (en) 2001-10-26
MXPA01011978A (en) 2002-05-06
HUP0301287A3 (en) 2005-03-29
AU2935300A (en) 2000-12-12
NO20015651L (en) 2002-01-18
AR022640A1 (en) 2002-09-04
MA26732A1 (en) 2004-12-20
HRP20010862A2 (en) 2003-06-30
BG106208A (en) 2002-09-30
PE20010157A1 (en) 2001-02-16
JP2003523941A (en) 2003-08-12
KR20020010916A (en) 2002-02-06
SK16602001A3 (en) 2003-03-04
ZA200109555B (en) 2004-04-07
EP1178784A1 (en) 2002-02-13
WO2000071107A8 (en) 2002-01-24
WO2000071107A2 (en) 2000-11-30
DZ3041A1 (en) 2004-03-27

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