ECSP088275A - Asociación de agonistas de los receptores beta3 y de inhibidores de la recaptación de monoaminas, composición farmacéutica que la contiene y su utilización en terapéutica - Google Patents

Asociación de agonistas de los receptores beta3 y de inhibidores de la recaptación de monoaminas, composición farmacéutica que la contiene y su utilización en terapéutica

Info

Publication number
ECSP088275A
ECSP088275A EC2008008275A ECSP088275A ECSP088275A EC SP088275 A ECSP088275 A EC SP088275A EC 2008008275 A EC2008008275 A EC 2008008275A EC SP088275 A ECSP088275 A EC SP088275A EC SP088275 A ECSP088275 A EC SP088275A
Authority
EC
Ecuador
Prior art keywords
association
therapeutics
pharmaceutical composition
agonists
inhibitors
Prior art date
Application number
EC2008008275A
Other languages
English (en)
Inventor
Guy Griebel
Jeanne Stemmelin
Original Assignee
Sanofi Aventis
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Aventis filed Critical Sanofi Aventis
Publication of ECSP088275A publication Critical patent/ECSP088275A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/135Amines having aromatic rings, e.g. ketamine, nortriptyline
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/135Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/136Amines having aromatic rings, e.g. ketamine, nortriptyline having the amino group directly attached to the aromatic ring, e.g. benzeneamine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/135Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/138Aryloxyalkylamines, e.g. propranolol, tamoxifen, phenoxybenzamine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/192Carboxylic acids, e.g. valproic acid having aromatic groups, e.g. sulindac, 2-aryl-propionic acids, ethacrynic acid 
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/195Carboxylic acids, e.g. valproic acid having an amino group
    • A61K31/196Carboxylic acids, e.g. valproic acid having an amino group the amino group being directly attached to a ring, e.g. anthranilic acid, mefenamic acid, diclofenac, chlorambucil
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/21Esters, e.g. nitroglycerine, selenocyanates
    • A61K31/215Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
    • A61K31/22Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acyclic acids, e.g. pravastatin
    • A61K31/222Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acyclic acids, e.g. pravastatin with compounds having aromatic groups, e.g. dipivefrine, ibopamine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/335Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/34Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide
    • A61K31/343Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide condensed with a carbocyclic ring, e.g. coumaran, bufuralol, befunolol, clobenfurol, amiodarone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/22Anxiolytics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Emergency Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

La invención se refiere a la asociación de al menos un agonista de los receptores b3 adrenérgicos (o agonista b3) con un inhibidor de la recaptación de monoaminas (IRMA). La invención también se refiere a una composición farmacéutica que comprende la asociación de la invención y su utilización en terapéutica.
EC2008008275A 2005-09-19 2008-03-14 Asociación de agonistas de los receptores beta3 y de inhibidores de la recaptación de monoaminas, composición farmacéutica que la contiene y su utilización en terapéutica ECSP088275A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR0509528A FR2890862B1 (fr) 2005-09-19 2005-09-19 Association d'agoniste aux recepteurs beta 3 et d'inhibiteur de la recapture de monoamnies, compostion pharmaceutique la contenant et son utilisation en therapeutique.
PCT/FR2006/002125 WO2007034056A1 (fr) 2005-09-19 2006-09-18 ASSOCIATION D'AGONISTE AUX RECEPTEURS ß3 ET D'INHIBITEURS DE LA RECAPTURE DE MONOAMINES, COMPOSITION PHARMACEUTIQUE LA CONTENANT ET SON UTILISATION EN THERAPEUTIQUE

Publications (1)

Publication Number Publication Date
ECSP088275A true ECSP088275A (es) 2008-04-28

Family

ID=36384391

Family Applications (1)

Application Number Title Priority Date Filing Date
EC2008008275A ECSP088275A (es) 2005-09-19 2008-03-14 Asociación de agonistas de los receptores beta3 y de inhibidores de la recaptación de monoaminas, composición farmacéutica que la contiene y su utilización en terapéutica

Country Status (23)

Country Link
US (1) US20080182899A1 (es)
EP (1) EP1928448B1 (es)
JP (1) JP2009508829A (es)
KR (1) KR20080064115A (es)
CN (1) CN101267814A (es)
AR (1) AR055436A1 (es)
AT (1) ATE441407T1 (es)
AU (1) AU2006293801A1 (es)
BR (1) BRPI0616197A2 (es)
CA (1) CA2620235A1 (es)
CR (1) CR9768A (es)
DE (1) DE602006008964D1 (es)
EA (1) EA200800870A1 (es)
EC (1) ECSP088275A (es)
FR (1) FR2890862B1 (es)
IL (1) IL189755A0 (es)
MA (1) MA30002B1 (es)
NO (1) NO20081723L (es)
NZ (1) NZ566310A (es)
TN (1) TNSN08095A1 (es)
TW (1) TW200744571A (es)
WO (1) WO2007034056A1 (es)
ZA (1) ZA200802544B (es)

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4018895A (en) * 1974-01-10 1977-04-19 Eli Lilly And Company Aryloxyphenylpropylamines in treating depression
FR2669821A1 (fr) * 1990-12-04 1992-06-05 Sanofi Sa Utilisation de phenylethanolaminotetralines pour la preparation de medicaments destines au traitement de la depression.
US5288749A (en) * 1991-12-20 1994-02-22 Abbott Laboratories Tertiary and secondary amines as alpha-2 antagonists and serotonin uptake inhibitors
US6288749B1 (en) * 1996-11-16 2001-09-11 Altec Lansing Technologies, Inc. Computer system with remote television display
SE9703375D0 (sv) * 1997-09-18 1997-09-18 Astra Ab A new combination
FR2826651B1 (fr) * 2001-06-28 2005-09-02 Sanofi Synthelabo Forme cristalline d'une phenylethanolamine, sa preparation et compositions pharmaceutiques la contenant
EP1675582A1 (en) * 2003-09-12 2006-07-05 Warner-Lambert Company LLC Combination comprising an alpha-2-delta ligand and an ssri and/or snri for treatment of depression and anxiety disorders

Also Published As

Publication number Publication date
MA30002B1 (fr) 2008-12-01
CA2620235A1 (fr) 2007-03-29
EP1928448A1 (fr) 2008-06-11
IL189755A0 (en) 2008-12-29
FR2890862A1 (fr) 2007-03-23
ZA200802544B (en) 2009-08-26
TW200744571A (en) 2007-12-16
NZ566310A (en) 2010-03-26
JP2009508829A (ja) 2009-03-05
EA200800870A1 (ru) 2008-08-29
CN101267814A (zh) 2008-09-17
BRPI0616197A2 (pt) 2011-06-14
AU2006293801A1 (en) 2007-03-29
DE602006008964D1 (de) 2009-10-15
AR055436A1 (es) 2007-08-22
KR20080064115A (ko) 2008-07-08
WO2007034056A1 (fr) 2007-03-29
FR2890862B1 (fr) 2008-01-25
NO20081723L (no) 2008-05-29
EP1928448B1 (fr) 2009-09-02
TNSN08095A1 (en) 2009-07-14
CR9768A (es) 2008-09-23
ATE441407T1 (de) 2009-09-15
US20080182899A1 (en) 2008-07-31

Similar Documents

Publication Publication Date Title
ECSP088222A (es) Agonistas de receptores adrenérgicos alfa2c funcionalmente selectivos
NZ740644A (en) Glucagon receptor agonists
ECSP088221A (es) Agonistas adrenoreceptores alfa2c
ECSP12012317A (es) Marcadores predictivos útiles en el tratamiento del síndrome frágil x (fxs)
CL2007003791A1 (es) Compuestos derivados de piperidina, inhibidores de la proteina quinasa; composicion farmaceutica que comprende a dichos compuestos; y su uso para inhibir el crecimiento celular anormal.
NI200900081U (es) Anticuerpos agonistas de trkb y sus usos.
CL2011001073A1 (es) Compuestos derivados de 1-[{pirrolidin-3-il}-carbonil]-5-(piperazin-1-ilcarbonil)-pirrolidin, agonistas de los receptores de la melanocortina; composicion farmaceutica; utiles en el tratamiento de la obesidad, diabetes, inflamacion y disfusion erectil.
ECSP11011417A (es) Anticuerpos anti-fgfr3 y métodos que los utilizan
DK2049475T3 (da) Cyclohexyl-substituerede pyrrolidinoner som inhibitorer af 11-beta-hydroxysteroid dehydrogenase1
UY32183A (es) Combinacion de una insulina y un agonista de glp-1
CL2007003793A1 (es) Metodo para inhibir union del receptor de muerte 6 (dr6) a la proteina precursora amiloide (app) que comprende uno o mas antagonistas del dr6; uso de dichos antagonistas; metodo para identificar una molecula de interes que inhibe la union del dr6 a l
CL2007001451A1 (es) Compuestos derivados de [1,2,3]-tiazol-4-ilmetoxilo, agonista del receptor farnesoide x (fxr); composicion farmaceutica que comprende a dichos compuestos; y su uso para tratar dislipidemia y enfermedades relacionadas.
DK2027096T3 (da) Substituerede arylimidazoloner og -triazoloner som inhibitorer for vasopressinreceptorerne
NO20073396L (no) Farmasoytiske kombinasjoner av en angiotensinreceptorantagonist og en NEP-inhibitor
MA28902B1 (fr) Agonistes des recepteurs beta2 adrenergiques diaminiques
DE602007012072D1 (de) Orantagonisten
CR20110421A (es) Agonistas y antagonistas del receptor de s1p, y métodos de uso de los mismos
CL2008002159A1 (es) Compuestos derivados de n-(((1r, 4r)-4-aminociclohexil)metil) sulfonaminas sustituidas con heterociclos, antagonistas del receptor npy y5; composicion farmaceutica que comprende a dichos compuestos, utiles para tratar anorexia y obesidad.
CL2010000214A1 (es) Metodos de tratamiento para inhibir la corrosion a base de azufre de una superficie, que comprende contactar a dicha superficie con una composicion que comprende aguarras.
DK1989196T3 (da) Piperidinoylpyrrolidiner som melanocortin-type 4-receptoragonister
CL2007001391A1 (es) Compuestos derivados de pirrolidinas sustituidas, inhibidores del factor xa y/o inhibidores sobre la serina proteasa; composicion farmaceutica que comprende a dichos compuestos; proedimiento para preparar la composicon farmaceutica; y uso de los compuestos preparar un medicamneto con un efecto antitrombotico
MX2010008875A (es) Agonistas nicotinicos alfa 7 y antipsicoticos.
AR059445A1 (es) Composiciones de antimicoticos ramnolipidicos y metodos de uso relacionados
DK2407451T3 (da) N,N-substituerede 3-aminopyrrolidin-forbindelser anvendelige som monoamin-genoptagelseshæmmere
ECSP099579A (es) Agonistas de adrenoreceptores alfa2c funcionalmente selectivos