DK1989196T3 - Piperidinoylpyrrolidiner som melanocortin-type 4-receptoragonister - Google Patents

Piperidinoylpyrrolidiner som melanocortin-type 4-receptoragonister

Info

Publication number
DK1989196T3
DK1989196T3 DK07705650.5T DK07705650T DK1989196T3 DK 1989196 T3 DK1989196 T3 DK 1989196T3 DK 07705650 T DK07705650 T DK 07705650T DK 1989196 T3 DK1989196 T3 DK 1989196T3
Authority
DK
Denmark
Prior art keywords
piperidinoylpyrrolidines
receptor agonists
melanocortin type
melanocortin
type
Prior art date
Application number
DK07705650.5T
Other languages
English (en)
Inventor
Mark David Andrews
Alan Daniel Brown
Mark Ian Lansdell
Nicholas William Summerhill
Original Assignee
Pfizer Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Ltd filed Critical Pfizer Ltd
Application granted granted Critical
Publication of DK1989196T3 publication Critical patent/DK1989196T3/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
DK07705650.5T 2006-02-23 2007-02-19 Piperidinoylpyrrolidiner som melanocortin-type 4-receptoragonister DK1989196T3 (da)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US77629506P 2006-02-23 2006-02-23
US88784007P 2007-02-02 2007-02-02
PCT/IB2007/000456 WO2007096763A2 (en) 2006-02-23 2007-02-19 Melanocortin type 4 receptor agonist piperidinoylpyrrolidines

Publications (1)

Publication Number Publication Date
DK1989196T3 true DK1989196T3 (da) 2013-04-15

Family

ID=38169450

Family Applications (1)

Application Number Title Priority Date Filing Date
DK07705650.5T DK1989196T3 (da) 2006-02-23 2007-02-19 Piperidinoylpyrrolidiner som melanocortin-type 4-receptoragonister

Country Status (22)

Country Link
US (1) US8138188B2 (da)
EP (1) EP1989196B1 (da)
KR (1) KR101036981B1 (da)
AP (1) AP2008004602A0 (da)
AU (1) AU2007219236B2 (da)
BR (1) BRPI0708264A2 (da)
CA (1) CA2642922C (da)
CR (1) CR10219A (da)
DK (1) DK1989196T3 (da)
EA (1) EA200801738A1 (da)
EC (1) ECSP088688A (da)
ES (1) ES2402581T3 (da)
HK (1) HK1126489A1 (da)
IL (1) IL193279A (da)
MA (1) MA30228B1 (da)
ME (1) MEP6808A (da)
MX (1) MX2008010899A (da)
NO (1) NO20083480L (da)
RS (1) RS20080371A (da)
SG (1) SG185849A1 (da)
TN (1) TNSN08337A1 (da)
WO (1) WO2007096763A2 (da)

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EP2025674A1 (de) 2007-08-15 2009-02-18 sanofi-aventis Substituierte Tetrahydronaphthaline, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel
US8848656B2 (en) 2007-11-16 2014-09-30 Qualcomm Incorporated Utilizing broadcast signals to convey restricted association information
US9603062B2 (en) 2007-11-16 2017-03-21 Qualcomm Incorporated Classifying access points using pilot identifiers
US8737295B2 (en) 2007-11-16 2014-05-27 Qualcomm Incorporated Sector identification using sector parameters signatures
US8902867B2 (en) 2007-11-16 2014-12-02 Qualcomm Incorporated Favoring access points in wireless communications
EP2103614A1 (en) * 2008-03-18 2009-09-23 Santhera Pharmaceuticals (Schweiz) AG Substituted imidazopyrimidine, imidazopyrazine and imidazopyridazine derivatives as melanocortin-4 receptor modulators
US8588773B2 (en) 2008-08-04 2013-11-19 Qualcomm Incorporated System and method for cell search and selection in a wireless communication system
UA99555C2 (en) 2008-11-12 2012-08-27 Элджи Лайф Саенсез Лтд. Melanocortin receptor agonists
ES2494015T3 (es) * 2009-11-18 2014-09-12 Helsinn Healthcare Sa Composiciones para tratar nauseas y vómitos de origen central
EP2722045B1 (en) 2009-11-18 2016-07-06 Helsinn Healthcare SA Compositions for treating centrally mediated nausea and vomiting
WO2012120052A1 (de) 2011-03-08 2012-09-13 Sanofi Mit carbozyklen oder heterozyklen substituierte oxathiazinderivate, verfahren zu deren herstellung, diese verbindungen enthaltende arzneimittel und deren verwendung
EP2683700B1 (de) 2011-03-08 2015-02-18 Sanofi Tetrasubstituierte oxathiazinderivate, verfahren zu deren herstellung, ihre verwendung als medikament sowie sie enthaltendes arzneimittel und deren verwendung
EP2683705B1 (de) 2011-03-08 2015-04-22 Sanofi Di- und trisubstituierte oxathiazinderivate, verfahren zu deren herstellung, ihre verwendung als medikament sowie sie enthaltendes arzneimittel und deren verwendung
US8828995B2 (en) 2011-03-08 2014-09-09 Sanofi Branched oxathiazine derivatives, method for the production thereof, use thereof as medicine and drug containing said derivatives and use thereof
WO2012120055A1 (de) 2011-03-08 2012-09-13 Sanofi Di- und trisubstituierte oxathiazinderivate, verfahren zu deren herstellung, ihre verwendung als medikament sowie sie enthaltendes arzneimittel und deren verwendung
ES2753227T3 (es) 2015-08-04 2020-04-07 Astellas Pharma Inc Derivado de piperazina
EP4161927A1 (en) 2020-06-09 2023-04-12 Pfizer Inc. Spiro compounds as melanocortin 4 receptor antagonists and uses thereof
WO2023105387A1 (en) 2021-12-06 2023-06-15 Pfizer Inc. Melanocortin 4 receptor antagonists and uses thereof

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US7649002B2 (en) 2004-02-04 2010-01-19 Pfizer Inc (3,5-dimethylpiperidin-1yl)(4-phenylpyrrolidin-3-yl)methanone derivatives as MCR4 agonists
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ES2421920T3 (es) 2008-08-06 2013-09-06 Pfizer Ltd Compuestos de diazepina y diazocano como agonistas de MC4

Also Published As

Publication number Publication date
SG185849A1 (en) 2012-12-28
WO2007096763A2 (en) 2007-08-30
EA200801738A1 (ru) 2008-12-30
HK1126489A1 (en) 2009-09-04
IL193279A (en) 2012-12-31
ES2402581T3 (es) 2013-05-06
MA30228B1 (fr) 2009-02-02
CR10219A (es) 2008-09-23
NO20083480L (no) 2008-09-10
RS20080371A (en) 2009-07-15
KR20080095918A (ko) 2008-10-29
BRPI0708264A2 (pt) 2011-05-24
CA2642922A1 (en) 2007-08-30
TNSN08337A1 (fr) 2009-12-29
EP1989196A2 (en) 2008-11-12
IL193279A0 (en) 2009-02-11
AU2007219236B2 (en) 2012-06-21
CA2642922C (en) 2011-08-02
US20090036459A1 (en) 2009-02-05
AP2008004602A0 (en) 2008-10-31
MEP6808A (xx) 2010-02-10
KR101036981B1 (ko) 2011-05-25
EP1989196B1 (en) 2013-02-13
WO2007096763A3 (en) 2007-10-18
ECSP088688A (es) 2008-10-31
MX2008010899A (es) 2008-11-27
US8138188B2 (en) 2012-03-20
AU2007219236A1 (en) 2007-08-30

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