ECSP077649A - Piridazinonilos macrociclicos como inhibidores de serina proteasa de hepatitis c - Google Patents
Piridazinonilos macrociclicos como inhibidores de serina proteasa de hepatitis cInfo
- Publication number
- ECSP077649A ECSP077649A EC2007007649A ECSP077649A ECSP077649A EC SP077649 A ECSP077649 A EC SP077649A EC 2007007649 A EC2007007649 A EC 2007007649A EC SP077649 A ECSP077649 A EC SP077649A EC SP077649 A ECSP077649 A EC SP077649A
- Authority
- EC
- Ecuador
- Prior art keywords
- hepatitis
- serine protease
- compounds
- piridazinonilos
- macrociclicos
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/08—Tripeptides
- C07K5/0802—Tripeptides with the first amino acid being neutral
- C07K5/0804—Tripeptides with the first amino acid being neutral and aliphatic
- C07K5/0808—Tripeptides with the first amino acid being neutral and aliphatic the side chain containing 2 to 4 carbon atoms, e.g. Val, Ile, Leu
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US49984406A | 2006-08-04 | 2006-08-04 | |
US11/832,893 US7718612B2 (en) | 2007-08-02 | 2007-08-02 | Pyridazinonyl macrocyclic hepatitis C serine protease inhibitors |
Publications (1)
Publication Number | Publication Date |
---|---|
ECSP077649A true ECSP077649A (es) | 2008-03-26 |
Family
ID=39033583
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EC2007007649A ECSP077649A (es) | 2006-08-04 | 2007-08-06 | Piridazinonilos macrociclicos como inhibidores de serina proteasa de hepatitis c |
Country Status (4)
Country | Link |
---|---|
CO (1) | CO6020004A1 (fr) |
EC (1) | ECSP077649A (fr) |
PE (1) | PE20080539A1 (fr) |
WO (1) | WO2008019303A2 (fr) |
Families Citing this family (26)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
MY140680A (en) | 2002-05-20 | 2010-01-15 | Bristol Myers Squibb Co | Hepatitis c virus inhibitors |
TWI387603B (zh) | 2005-07-20 | 2013-03-01 | Merck Sharp & Dohme | Hcv ns3蛋白酶抑制劑 |
ES2356776T3 (es) | 2005-10-11 | 2011-04-13 | Intermune, Inc. | Compuestos y métodos para inhibir la replicación del virus de la hepatitis. |
RU2008152171A (ru) | 2006-07-05 | 2010-08-10 | Интермьюн, Инк. (Us) | Новые ингибиторы вирусной репликации гепатита с |
US8207341B2 (en) | 2008-09-04 | 2012-06-26 | Bristol-Myers Squibb Company | Process or synthesizing substituted isoquinolines |
UY32099A (es) | 2008-09-11 | 2010-04-30 | Enanta Pharm Inc | Inhibidores macrocíclicos de serina proteasas de hepatitis c |
TW201040181A (en) | 2009-04-08 | 2010-11-16 | Idenix Pharmaceuticals Inc | Macrocyclic serine protease inhibitors |
WO2010135748A1 (fr) * | 2009-05-22 | 2010-11-25 | Sequoia Pharmaceuticals Inc. | Inhibiteurs de la protéase ns3 du virus de l'hépatite c bimacrocyclique |
US8232246B2 (en) | 2009-06-30 | 2012-07-31 | Abbott Laboratories | Anti-viral compounds |
TW201117812A (en) | 2009-08-05 | 2011-06-01 | Idenix Pharmaceuticals Inc | Macrocyclic serine protease inhibitors |
US8933110B2 (en) | 2010-01-25 | 2015-01-13 | Enanta Pharmaceuticals, Inc. | Hepatitis C virus inhibitors |
US8785487B2 (en) | 2010-01-25 | 2014-07-22 | Enanta Pharmaceuticals, Inc. | Hepatitis C virus inhibitors |
EP2658859A4 (fr) | 2010-12-30 | 2014-07-30 | Enanta Pharm Inc | Inhibiteurs macrocycliques de sérine protéase d'hépatite c |
BR112013016480A2 (pt) | 2010-12-30 | 2016-09-20 | Abbvie Inc | macrocíclo da fenantridina inibadores da protease da serina da hepatite c |
US9353100B2 (en) | 2011-02-10 | 2016-05-31 | Idenix Pharmaceuticals Llc | Macrocyclic serine protease inhibitors, pharmaceutical compositions thereof, and their use for treating HCV infections |
US8957203B2 (en) | 2011-05-05 | 2015-02-17 | Bristol-Myers Squibb Company | Hepatitis C virus inhibitors |
US10201584B1 (en) | 2011-05-17 | 2019-02-12 | Abbvie Inc. | Compositions and methods for treating HCV |
US8691757B2 (en) | 2011-06-15 | 2014-04-08 | Bristol-Myers Squibb Company | Hepatitis C virus inhibitors |
RS55592B1 (sr) | 2012-10-19 | 2017-06-30 | Bristol Myers Squibb Co | 9-metil supstituisani heksadekahidrociklopropa(e)pirolo(1,2-a)(1,4)diazaciklopentadecinil karbamat derivati kao nestrukturalni 3 (ns3) proteazni inhibitori za lečenje infekcijavirusom hepatitisa c |
WO2014070964A1 (fr) | 2012-11-02 | 2014-05-08 | Bristol-Myers Squibb Company | Inhibiteurs du virus de l'hépatite c |
EP2914598B1 (fr) | 2012-11-02 | 2017-10-18 | Bristol-Myers Squibb Company | Inhibiteurs du virus de l'hépatite c |
US9643999B2 (en) | 2012-11-02 | 2017-05-09 | Bristol-Myers Squibb Company | Hepatitis C virus inhibitors |
WO2014070974A1 (fr) | 2012-11-05 | 2014-05-08 | Bristol-Myers Squibb Company | Inhibiteurs du virus de l'hépatite c |
US9310374B2 (en) * | 2012-11-16 | 2016-04-12 | Redwood Bioscience, Inc. | Hydrazinyl-indole compounds and methods for producing a conjugate |
US9580463B2 (en) | 2013-03-07 | 2017-02-28 | Bristol-Myers Squibb Company | Hepatitis C virus inhibitors |
WO2015103490A1 (fr) | 2014-01-03 | 2015-07-09 | Abbvie, Inc. | Formes galéniques antivirales solides |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US7601709B2 (en) * | 2003-02-07 | 2009-10-13 | Enanta Pharmaceuticals, Inc. | Macrocyclic hepatitis C serine protease inhibitors |
KR100940619B1 (ko) * | 2003-02-07 | 2010-02-05 | 이난타 파마슈티칼스, 인코포레이티드 | 마크로사이클릭 씨형 간염 세린 단백효소 억제제 |
US20040180815A1 (en) * | 2003-03-07 | 2004-09-16 | Suanne Nakajima | Pyridazinonyl macrocyclic hepatitis C serine protease inhibitors |
-
2007
- 2007-08-03 WO PCT/US2007/075146 patent/WO2008019303A2/fr active Application Filing
- 2007-08-06 CO CO07080060A patent/CO6020004A1/es not_active Application Discontinuation
- 2007-08-06 PE PE2007001036A patent/PE20080539A1/es not_active Application Discontinuation
- 2007-08-06 EC EC2007007649A patent/ECSP077649A/es unknown
Also Published As
Publication number | Publication date |
---|---|
WO2008019303A3 (fr) | 2008-10-30 |
CO6020004A1 (es) | 2009-03-31 |
WO2008019303A2 (fr) | 2008-02-14 |
PE20080539A1 (es) | 2008-05-16 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
DOP2019000218A (es) | Inhibidores de las proteasas de serina del vhc derivados de prolinas macrocíclicas | |
ECSP077648A (es) | Tetrazolilos macrociclicos como inhibidores de serina proteasa de hepatitis c | |
ECSP077649A (es) | Piridazinonilos macrociclicos como inhibidores de serina proteasa de hepatitis c | |
AR061238A1 (es) | Compuestos de oxilmilo macrociclico inhibidores de proteasa de hepatitis c | |
UY30391A1 (es) | Compuesto de oximilo aciclico inhibidores de proteasa de hepatitis c | |
ECSP10010254A (es) | Compuestos que contienen quinoxalina como inhibidores del virus de la hepatitis c | |
UY30437A1 (es) | Quinoxalinil macroceclicos inhibidores de serina proteasa del virus de la hepatitis c | |
CO6571891A2 (es) | Inhibidores del virus de la hepatitis c. | |
CO2020002980A2 (es) | Agentes antivirales contra la hepatitis b. | |
UY28423A1 (es) | Inhibidores de proteasas serinas, en especial proteasa ns3-ns4a del vhc.- | |
MX2010010276A (es) | Compuestos macrociclicos fluorinados como inhibidores del virus de hepatitis c. | |
DOP2013000238A (es) | Derivados de nucleosidos 2'-sustituidos y metodos de uso de los mismos para el tratamiento de enfermedades virales | |
ECSP088258A (es) | Inhibidores de serina proteasas | |
UY28500A1 (es) | Inhibidores de proteasas de serina, en particular proteasa ns3-ns4a del vhc. | |
MX2010006210A (es) | Inhibidores de serina proteasa de hcv de tripeptido fluorado. | |
MX2010006518A (es) | Inhibidores de serina proteasa de hepatitis c de oximil macrociclica. | |
MX2011012155A (es) | Compuestos macrociclicos como inhibidores del virus de hepatitis c. | |
MX2010008109A (es) | Tripéptidos difluorizados como inhibidores de proteasa de serina de virus de hepatitis c (hcv). | |
MX2010008108A (es) | Inhibidores de proteasa de serina de tripéptido de virus de hepatitis c (hcv) que contienen heteroarilo. | |
TH139657A (th) | สารยับยั้ง hcv เซอรีนโปรติเอสที่ให้มาโครไซคลิกโพรลีน |