EA202190752A1 - Получение ингибитора семикарбазид-чувствительной аминоксидазы и его применение - Google Patents

Получение ингибитора семикарбазид-чувствительной аминоксидазы и его применение

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EA202190752A1
EA202190752A1 EA202190752A EA202190752A EA202190752A1 EA 202190752 A1 EA202190752 A1 EA 202190752A1 EA 202190752 A EA202190752 A EA 202190752A EA 202190752 A EA202190752 A EA 202190752A EA 202190752 A1 EA202190752 A1 EA 202190752A1
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Eurasian Patent Office
Prior art keywords
preparation
application
inhibitor
aminoxidase
semicarbazide
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EA202190752A
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English (en)
Inventor
Шэнъян Лю
Цзяньвэнь Ден
Чжиюн Фэн
Лэй Цзян
Чжи Цяо
Кэ Шан
Сяопин Се
Сюэли Сюй
Юань Сюй
Хайся Чжао
Original Assignee
Шанхай Инновабио Фармасьютикалс Ко., Лтд.
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Application filed by Шанхай Инновабио Фармасьютикалс Ко., Лтд. filed Critical Шанхай Инновабио Фармасьютикалс Ко., Лтд.
Publication of EA202190752A1 publication Critical patent/EA202190752A1/ru

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    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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Abstract

Предложен препарат ингибитора семикарбазид-чувствительной аминоксидазы и его применение. В частности, изобретение представляет собой соединение, показанное в формуле I, или его стереоизомер, или рацемат, или фармацевтически приемлемую соль. Также раскрыто, что указанное выше соединение может ингибировать семикарбазид-чувствительную аминоксидазу.
EA202190752A 2018-09-25 2019-09-25 Получение ингибитора семикарбазид-чувствительной аминоксидазы и его применение EA202190752A1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CN201811119234.2A CN110938059A (zh) 2018-09-25 2018-09-25 胺基脲敏感性胺氧化酶抑制剂制备及其应用
PCT/CN2019/107972 WO2020063696A1 (zh) 2018-09-25 2019-09-25 胺基脲敏感性胺氧化酶抑制剂制备及其应用

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EA202190752A1 true EA202190752A1 (ru) 2021-08-24

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US (1) US20220081426A1 (ru)
EP (1) EP3858827A4 (ru)
JP (2) JP2022501393A (ru)
KR (1) KR102649362B1 (ru)
CN (2) CN110938059A (ru)
AU (1) AU2019347947B2 (ru)
CA (1) CA3114243A1 (ru)
EA (1) EA202190752A1 (ru)
WO (1) WO2020063696A1 (ru)

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KR20190110740A (ko) 2018-03-21 2019-10-01 주식회사유한양행 신규의 아릴 또는 헤테로아릴 트라이아졸론 유도체 또는 이의 염 및 이를 포함하는 약학 조성물
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TW202039486A (zh) 2018-12-14 2020-11-01 南韓商柳韓洋行股份有限公司 三唑并吡啶-3-酮化物或其鹽及包含彼之醫藥組合物
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JP2023130361A (ja) 2023-09-20
CN112839940B (zh) 2023-12-22
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