EA202092540A1 - Комбинации для лечения рака - Google Patents
Комбинации для лечения ракаInfo
- Publication number
- EA202092540A1 EA202092540A1 EA202092540A EA202092540A EA202092540A1 EA 202092540 A1 EA202092540 A1 EA 202092540A1 EA 202092540 A EA202092540 A EA 202092540A EA 202092540 A EA202092540 A EA 202092540A EA 202092540 A1 EA202092540 A1 EA 202092540A1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- combinations
- cancer treatment
- acceptable salt
- pharmaceutically
- pentaazaheptacyclo
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/415—1,2-Diazoles
- A61K31/4155—1,2-Diazoles non condensed and containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/415—1,2-Diazoles
- A61K31/4162—1,2-Diazoles condensed with heterocyclic ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/4985—Pyrazines or piperazines ortho- or peri-condensed with heterocyclic ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K2300/00—Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Oncology (AREA)
- Hematology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
Раскрыты способы лечения рака, включающие введение 17-хлор-5,13,14,22-тетраметил-28-окса-2,9-дитиа-5,6,12,13,22-пентаазагептацикло[27.7.1.14,7.011,15.016,21.020,24.030,35]октатриаконта-1(37),4(38),6,11,14,16,18,20,23,29,31,33,35-тридекаен-23-карбоновой кислоты, ее фармацевтически приемлемой соли и акалабрутиниба или его фармацевтически приемлемой соли.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US201862664356P | 2018-04-30 | 2018-04-30 | |
PCT/IB2019/053491 WO2019211721A1 (en) | 2018-04-30 | 2019-04-29 | Combinations for treating cancer |
Publications (1)
Publication Number | Publication Date |
---|---|
EA202092540A1 true EA202092540A1 (ru) | 2021-03-17 |
Family
ID=66794041
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EA202092540A EA202092540A1 (ru) | 2018-04-30 | 2019-04-29 | Комбинации для лечения рака |
Country Status (14)
Country | Link |
---|---|
US (1) | US20210030718A1 (ru) |
EP (1) | EP3787620A1 (ru) |
JP (1) | JP2021522246A (ru) |
KR (1) | KR20210005182A (ru) |
CN (1) | CN112040944A (ru) |
AU (1) | AU2019263026B2 (ru) |
BR (1) | BR112020022020A2 (ru) |
CA (1) | CA3097486A1 (ru) |
EA (1) | EA202092540A1 (ru) |
MA (1) | MA52499A (ru) |
MX (1) | MX2020011453A (ru) |
SG (1) | SG11202010528XA (ru) |
TW (1) | TW202014184A (ru) |
WO (1) | WO2019211721A1 (ru) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
MX2022005250A (es) * | 2019-11-04 | 2022-06-08 | Astrazeneca Ab | Combinaciones terapeuticas de acalabrutinib y capivasertib para tratar neoplasias malignas de linfocitos b. |
CN115052880A (zh) * | 2019-12-18 | 2022-09-13 | 芝诺管理公司 | 大环化合物 |
KR20240019283A (ko) | 2021-06-11 | 2024-02-14 | 길리애드 사이언시즈, 인코포레이티드 | Mcl-1 저해제와 항암제의 병용 |
US11931424B2 (en) | 2021-06-11 | 2024-03-19 | Gilead Sciences, Inc. | Combination MCL-1 inhibitors with anti-body drug conjugates |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
MY192354A (en) | 2011-07-19 | 2022-08-17 | Merck Sharp & Dohme | 4-imidazopyridazin-1-yl-benzamides and 4-imidazotriazin-1-yl-benzamides as btk-inhibitors |
AU2015300966A1 (en) * | 2014-08-08 | 2017-02-16 | Janssen Pharmaceutica Nv | Bruton's tyrosine kinase inhibitor combinations and uses thereof |
CO2018008759A2 (es) * | 2016-04-22 | 2018-09-20 | Astrazeneca Ab | Inhibidores de mcl-1 y métodos de uso de los mismos |
CN107056786B (zh) * | 2016-10-14 | 2019-05-07 | 苏州明锐医药科技有限公司 | 阿卡替尼的制备方法 |
-
2019
- 2019-03-05 TW TW108107170A patent/TW202014184A/zh unknown
- 2019-04-29 SG SG11202010528XA patent/SG11202010528XA/en unknown
- 2019-04-29 MA MA052499A patent/MA52499A/fr unknown
- 2019-04-29 KR KR1020207034122A patent/KR20210005182A/ko unknown
- 2019-04-29 CA CA3097486A patent/CA3097486A1/en active Pending
- 2019-04-29 AU AU2019263026A patent/AU2019263026B2/en not_active Ceased
- 2019-04-29 US US17/047,931 patent/US20210030718A1/en not_active Abandoned
- 2019-04-29 CN CN201980028857.5A patent/CN112040944A/zh active Pending
- 2019-04-29 EP EP19729355.8A patent/EP3787620A1/en not_active Withdrawn
- 2019-04-29 EA EA202092540A patent/EA202092540A1/ru unknown
- 2019-04-29 JP JP2020559437A patent/JP2021522246A/ja not_active Withdrawn
- 2019-04-29 BR BR112020022020-5A patent/BR112020022020A2/pt not_active IP Right Cessation
- 2019-04-29 MX MX2020011453A patent/MX2020011453A/es unknown
- 2019-04-29 WO PCT/IB2019/053491 patent/WO2019211721A1/en unknown
Also Published As
Publication number | Publication date |
---|---|
MX2020011453A (es) | 2020-12-07 |
KR20210005182A (ko) | 2021-01-13 |
SG11202010528XA (en) | 2020-11-27 |
JP2021522246A (ja) | 2021-08-30 |
EP3787620A1 (en) | 2021-03-10 |
CN112040944A (zh) | 2020-12-04 |
US20210030718A1 (en) | 2021-02-04 |
AU2019263026A1 (en) | 2020-12-17 |
CA3097486A1 (en) | 2019-11-07 |
WO2019211721A1 (en) | 2019-11-07 |
BR112020022020A2 (pt) | 2021-02-02 |
MA52499A (fr) | 2021-04-14 |
AU2019263026B2 (en) | 2022-06-30 |
TW202014184A (zh) | 2020-04-16 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
EA202092540A1 (ru) | Комбинации для лечения рака | |
ZA202202097B (en) | Amino pyrimidine ssao inhibitors | |
PH12020551043A1 (en) | Compounds, compositions, and methods for treatment of diseases involving acidic or hypoxic diseased tissues | |
EA201792191A1 (ru) | Комбинированная терапия fgfr/pd-1 для лечения злокачественной опухоли | |
EA201892075A1 (ru) | Комбинации ингибиторов lsd1 для применения для лечения солидных опухолей | |
EA201991622A1 (ru) | Комплексная терапия для лечения рака | |
AU2018278311A1 (en) | IRE1 small molecule inhibitors | |
MX2021005075A (es) | Metodos para el tratamiento de cancer de prostata resistente a la castracion y sensible a la castracion. | |
EA201891399A1 (ru) | Бипиразолильные производные, пригодные для лечения аутоиммунных заболеваний | |
EA202192122A1 (ru) | Соединения, обладающие активностью индуцирования ферроптоза, и способы их применения | |
BR112017026061A2 (pt) | composto, uso de um composto, e, método de tratamento de uma infecção viral | |
EA201990400A1 (ru) | Соединения и композиции и их применение | |
EA201991688A1 (ru) | Фармацевтические комбинации для лечения рака | |
MX2021007247A (es) | Derivados de rapamicina. | |
EA202193276A1 (ru) | Способы лечения холангиокарциномы | |
ZA202206308B (en) | Ezetimibe and curcumin for use in cancer treatment | |
EA202191192A1 (ru) | Кристаллические соли ингибитора плазменного калликреина | |
EA201892311A1 (ru) | Производные 2-анилинопиримидина в качестве терапевтических агентов для лечения рака мозга | |
EA202091112A1 (ru) | Сокристаллы, фармацевтические композиции на их основе и способы лечения, предусматривающие их применение | |
ZA202106519B (en) | Caspase inhibitors and methods of use thereof | |
ZA202103975B (en) | Methods of treating disease with magl inhibitors | |
EA202090266A1 (ru) | Ингибиторы mpo для применения в медицине | |
MX2021000935A (es) | Composiciones y metodos terapeuticos para el tratamiento de cancer pancreatico con acido 6,8-bis(bencilsulfanil)octanoico. | |
EA201650085A1 (ru) | Способ лечения опухолевого заболевания и способ селективного ингибирования роста опухолевых клеток с помощью производного хиноксалин-1,4-диоксида | |
WO2018211324A8 (en) | Prodrugs for the treatment of disease |