EA201991990A1 - Фармацевтические композиции для комбинированной терапии - Google Patents
Фармацевтические композиции для комбинированной терапииInfo
- Publication number
- EA201991990A1 EA201991990A1 EA201991990A EA201991990A EA201991990A1 EA 201991990 A1 EA201991990 A1 EA 201991990A1 EA 201991990 A EA201991990 A EA 201991990A EA 201991990 A EA201991990 A EA 201991990A EA 201991990 A1 EA201991990 A1 EA 201991990A1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- pharmaceutical compositions
- combined therapy
- combination
- phenyl
- cenicrivirok
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
- A61K31/19—Carboxylic acids, e.g. valproic acid
- A61K31/192—Carboxylic acids, e.g. valproic acid having aromatic groups, e.g. sulindac, 2-aryl-propionic acids, ethacrynic acid
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4164—1,3-Diazoles
- A61K31/4178—1,3-Diazoles not condensed 1,3-diazoles and containing further heterocyclic rings, e.g. pilocarpine, nitrofurantoin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K2300/00—Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
Abstract
Настоящее изобретение относится к фармацевтической комбинации, содержащей агонист PPAR и (S,Е)-8-(4-(2-бутоксиэтокси)фенил)-1-(2-метилпропил)-N-(4-((((1-пропил)-1Н-имидазол-5-ил)метил)сульфинил)фенил)-1,2,3,4-тетрагидробензо[b]азоцин-5-карбоксамид, также известный как ценикривирок (CVC), или его производные, и её применению. Комбинация может быть полезна в комбинированной терапии для лечения воспалительных, метаболических, фиброзных и холестатических заболеваний.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP17305213 | 2017-02-24 | ||
PCT/EP2018/054588 WO2018154081A1 (en) | 2017-02-24 | 2018-02-23 | Pharmaceutical compositions for combination therapy |
Publications (1)
Publication Number | Publication Date |
---|---|
EA201991990A1 true EA201991990A1 (ru) | 2020-04-07 |
Family
ID=58231557
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EA201991990A EA201991990A1 (ru) | 2017-02-24 | 2018-02-23 | Фармацевтические композиции для комбинированной терапии |
Country Status (14)
Country | Link |
---|---|
US (1) | US11590108B2 (ru) |
EP (1) | EP3585384A1 (ru) |
JP (1) | JP2020510651A (ru) |
KR (1) | KR102633249B1 (ru) |
CN (1) | CN110418641A (ru) |
AU (1) | AU2018223976B2 (ru) |
BR (1) | BR112019017314A2 (ru) |
CA (1) | CA3051977A1 (ru) |
EA (1) | EA201991990A1 (ru) |
IL (1) | IL268708B (ru) |
MX (1) | MX2019009909A (ru) |
PH (1) | PH12019501820A1 (ru) |
SG (1) | SG11201907084VA (ru) |
WO (1) | WO2018154081A1 (ru) |
Families Citing this family (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
KR102338085B1 (ko) * | 2016-03-31 | 2021-12-10 | 장피트 | 담즙울체성 질환의 치료 방법 |
US20220133666A1 (en) * | 2016-03-31 | 2022-05-05 | Genfit | Methods of treatment of cholestatic diseases |
Family Cites Families (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
ES2339340T3 (es) | 2001-08-08 | 2010-05-19 | Tobira Therapeutics, Inc. | Compuesto biciclico, produccion y su uso. |
FR2841900B1 (fr) | 2002-07-08 | 2007-03-02 | Genfit S A | Nouveaux derives de 1,3-diphenylprop-2-en-1-one substitues, preparation et utilisations |
EA020849B1 (ru) * | 2009-11-26 | 2015-02-27 | Женфит | Применение 1,3-дифенилпроп-2-ен-1-оновых производных для лечения заболеваний печени |
SG10201909122QA (en) * | 2011-10-28 | 2019-11-28 | Lumena Pharmaceuticals Inc | Bile acid recycling inhibitors for treatment of pediatric cholestatic liver diseases |
SG10201808104RA (en) * | 2014-03-21 | 2018-10-30 | Tobira Therapeutics Inc | Cenicriviroc for the treatment of fibrosis |
EP3777863A1 (en) * | 2014-09-12 | 2021-02-17 | Tobira Therapeutics, Inc. | Cenicriviroc combination therapy for the treatment of fibrosis |
EP3349751A4 (en) | 2015-09-16 | 2019-05-22 | Tobira Therapeutics, Inc. | CENICRIVIROC COMBINATION THERAPY FOR THE TREATMENT OF FIBROSIS |
KR102338085B1 (ko) * | 2016-03-31 | 2021-12-10 | 장피트 | 담즙울체성 질환의 치료 방법 |
AU2017249603B2 (en) | 2016-04-11 | 2022-12-01 | Genfit | Methods of treatment for cholestatic and fibrotic diseases |
JOP20190040A1 (ar) * | 2016-09-14 | 2019-03-10 | Novartis Ag | توليفة من ناهضات fxr |
SG11201906041QA (en) | 2017-01-27 | 2019-08-27 | Genfit | Pharmaceutical compositions for combination therapy |
-
2018
- 2018-02-23 AU AU2018223976A patent/AU2018223976B2/en active Active
- 2018-02-23 KR KR1020197027007A patent/KR102633249B1/ko active IP Right Grant
- 2018-02-23 CN CN201880013686.4A patent/CN110418641A/zh active Pending
- 2018-02-23 JP JP2019546127A patent/JP2020510651A/ja active Pending
- 2018-02-23 MX MX2019009909A patent/MX2019009909A/es unknown
- 2018-02-23 CA CA3051977A patent/CA3051977A1/en active Pending
- 2018-02-23 WO PCT/EP2018/054588 patent/WO2018154081A1/en unknown
- 2018-02-23 EA EA201991990A patent/EA201991990A1/ru unknown
- 2018-02-23 US US16/485,025 patent/US11590108B2/en active Active
- 2018-02-23 EP EP18705945.6A patent/EP3585384A1/en not_active Withdrawn
- 2018-02-23 SG SG11201907084VA patent/SG11201907084VA/en unknown
- 2018-02-23 BR BR112019017314A patent/BR112019017314A2/pt not_active Application Discontinuation
-
2019
- 2019-08-06 PH PH12019501820A patent/PH12019501820A1/en unknown
- 2019-08-14 IL IL268708A patent/IL268708B/en unknown
Also Published As
Publication number | Publication date |
---|---|
CN110418641A (zh) | 2019-11-05 |
US11590108B2 (en) | 2023-02-28 |
US20190388394A1 (en) | 2019-12-26 |
AU2018223976A1 (en) | 2019-09-05 |
IL268708A (en) | 2019-10-31 |
CA3051977A1 (en) | 2018-08-30 |
JP2020510651A (ja) | 2020-04-09 |
KR102633249B1 (ko) | 2024-02-02 |
KR20190119097A (ko) | 2019-10-21 |
MX2019009909A (es) | 2019-10-14 |
BR112019017314A2 (pt) | 2020-04-14 |
SG11201907084VA (en) | 2019-09-27 |
IL268708B (en) | 2022-05-01 |
PH12019501820A1 (en) | 2020-09-14 |
WO2018154081A1 (en) | 2018-08-30 |
AU2018223976B2 (en) | 2023-08-17 |
EP3585384A1 (en) | 2020-01-01 |
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