EA201892265A1 - Способы лечения офтальмологических заболеваний - Google Patents

Способы лечения офтальмологических заболеваний

Info

Publication number
EA201892265A1
EA201892265A1 EA201892265A EA201892265A EA201892265A1 EA 201892265 A1 EA201892265 A1 EA 201892265A1 EA 201892265 A EA201892265 A EA 201892265A EA 201892265 A EA201892265 A EA 201892265A EA 201892265 A1 EA201892265 A1 EA 201892265A1
Authority
EA
Eurasian Patent Office
Prior art keywords
treatment
methods
ophthalmic diseases
ophthalmic
diseases
Prior art date
Application number
EA201892265A
Other languages
English (en)
Russian (ru)
Inventor
Дуглас Майкл Акерманн
Джеймс Лудин
Кеннет Дж. Манделл
Original Assignee
Ойстер Поинт Фарма, Инк.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ойстер Поинт Фарма, Инк. filed Critical Ойстер Поинт Фарма, Инк.
Publication of EA201892265A1 publication Critical patent/EA201892265A1/ru

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/436—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a six-membered ring having oxygen as a ring hetero atom, e.g. rapamycin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/12—Cyclic peptides, e.g. bacitracins; Polymyxins; Gramicidins S, C; Tyrocidins A, B or C
    • A61K38/13—Cyclosporins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0043—Nose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A61P27/04—Artificial tears; Irrigation solutions

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Ophthalmology & Optometry (AREA)
  • Otolaryngology (AREA)
  • Immunology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
EA201892265A 2016-04-07 2017-04-06 Способы лечения офтальмологических заболеваний EA201892265A1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201662319648P 2016-04-07 2016-04-07
PCT/US2017/026385 WO2017177024A1 (en) 2016-04-07 2017-04-06 Methods of treating ocular conditions

Publications (1)

Publication Number Publication Date
EA201892265A1 true EA201892265A1 (ru) 2019-04-30

Family

ID=58549326

Family Applications (1)

Application Number Title Priority Date Filing Date
EA201892265A EA201892265A1 (ru) 2016-04-07 2017-04-06 Способы лечения офтальмологических заболеваний

Country Status (19)

Country Link
US (3) US10709707B2 (cg-RX-API-DMAC10.html)
EP (2) EP3970724A1 (cg-RX-API-DMAC10.html)
JP (3) JP7090551B2 (cg-RX-API-DMAC10.html)
KR (2) KR102512777B1 (cg-RX-API-DMAC10.html)
CN (3) CN114533737B (cg-RX-API-DMAC10.html)
AU (1) AU2017248276B2 (cg-RX-API-DMAC10.html)
DK (1) DK3439661T3 (cg-RX-API-DMAC10.html)
EA (1) EA201892265A1 (cg-RX-API-DMAC10.html)
ES (1) ES2893126T3 (cg-RX-API-DMAC10.html)
IL (3) IL299204A (cg-RX-API-DMAC10.html)
MX (2) MX385698B (cg-RX-API-DMAC10.html)
MY (1) MY199237A (cg-RX-API-DMAC10.html)
NZ (1) NZ746468A (cg-RX-API-DMAC10.html)
PH (1) PH12018502154A1 (cg-RX-API-DMAC10.html)
PT (1) PT3439661T (cg-RX-API-DMAC10.html)
SG (1) SG11201808650QA (cg-RX-API-DMAC10.html)
TW (2) TWI876258B (cg-RX-API-DMAC10.html)
WO (1) WO2017177024A1 (cg-RX-API-DMAC10.html)
ZA (1) ZA201807438B (cg-RX-API-DMAC10.html)

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US9145396B2 (en) 2008-12-01 2015-09-29 Targacept, Inc. Synthesis and novel salt forms of (R)-5-((E)-2-pyrrolidin-3ylvinyl)pyrimidine
CN107106542B (zh) 2014-10-20 2020-05-08 奥伊斯特普安生物制药公司 治疗眼部病状的方法
NZ746468A (en) * 2016-04-07 2023-06-30 Oyster Point Pharma Inc Methods of treating ocular conditions
WO2020014217A1 (en) 2018-07-10 2020-01-16 Oyster Point Pharma, Inc. Methods of treating ocular conditions
EP3820443A1 (en) 2018-07-10 2021-05-19 Oyster Point Pharma, Inc. Combinations of positive allosteric modulators and nicotinic acetylcholine receptor agonists for treating ocular conditions
EP4142734B1 (en) * 2020-04-28 2025-08-20 Oyster Point Pharma, Inc. Local administration of nicotinic acetylcholine receptor agonists for the inhibition of coronavirus infections
JP2024517459A (ja) * 2021-05-07 2024-04-22 オイスター ポイント ファーマ インコーポレイテッド ベクター及びニコチン作動薬の併用療法
WO2026080563A1 (en) 2024-10-09 2026-04-16 Oyster Point Pharma, Inc. Simpinicline oral formations and use thereof

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US6277855B1 (en) 2000-04-21 2001-08-21 Inspire Pharmaceuticals, Inc. Method of treating dry eye disease with nicotinic acetylcholine receptor agonists
US20030008892A1 (en) 2001-07-09 2003-01-09 Pfizer Inc. Pharmaceutical composition and method of modulating cholinergic function in a mammal
IL161326A0 (en) 2001-11-29 2004-09-27 Pfizer Prod Inc Succinic acid salts of 5,8,14-triazatetracyclo'10.3.1.0<2,11>.0<4,9>-hexadeca-2 (11),3,5,7,9-pentaene and pharmaceutical compositions thereof
AU2003269413A1 (en) 2002-11-01 2004-05-25 Pharmacia & Upjohn Company Llc Nicotinic acetylcholine agonists in the treatment of glaucoma and retinal neuropathy
US7098331B2 (en) 2003-03-05 2006-08-29 Targacept, Inc. Arylvinylazacycloalkane compounds and methods of preparation and use thereof
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IL266097B (en) * 2008-12-01 2022-07-01 Oyster Point Pharma Inc Mono-orotate acid addition salt of r(–5–)–e(–2–)pyrrolidine––3ylvinyl)pyrimidine
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CN107106542B (zh) 2014-10-20 2020-05-08 奥伊斯特普安生物制药公司 治疗眼部病状的方法
NZ746468A (en) 2016-04-07 2023-06-30 Oyster Point Pharma Inc Methods of treating ocular conditions

Also Published As

Publication number Publication date
JP2024103594A (ja) 2024-08-01
KR20190005859A (ko) 2019-01-16
US20190201397A1 (en) 2019-07-04
CN114533737B (zh) 2024-05-31
PH12018502154A1 (en) 2019-07-08
US10709707B2 (en) 2020-07-14
WO2017177024A8 (en) 2018-11-08
DK3439661T3 (da) 2021-10-18
TWI790997B (zh) 2023-02-01
MX2018012230A (es) 2019-03-28
CN109310692A (zh) 2019-02-05
TW201737917A (zh) 2017-11-01
ES2893126T3 (es) 2022-02-08
ZA201807438B (en) 2024-09-25
KR102512777B1 (ko) 2023-03-23
EP3439661A1 (en) 2019-02-13
IL290069B1 (en) 2023-01-01
AU2017248276A1 (en) 2018-11-22
US20250000861A1 (en) 2025-01-02
JP2019513759A (ja) 2019-05-30
WO2017177024A1 (en) 2017-10-12
EP3970724A1 (en) 2022-03-23
ES2893126T8 (es) 2022-05-23
MX385698B (es) 2025-03-18
TWI876258B (zh) 2025-03-11
CN114432313A (zh) 2022-05-06
EP3439661B1 (en) 2021-08-04
IL299204A (en) 2023-02-01
IL290069A (en) 2022-03-01
PT3439661T (pt) 2021-09-30
IL290069B2 (en) 2023-05-01
CN114533737A (zh) 2022-05-27
BR112018070497A2 (pt) 2019-01-29
NZ785093A (en) 2024-07-05
JP7090551B2 (ja) 2022-06-24
TW202320785A (zh) 2023-06-01
MX2021010399A (es) 2022-01-18
IL262102B (en) 2022-03-01
SG11201808650QA (en) 2018-10-30
MY199237A (en) 2023-10-22
CN109310692B (zh) 2022-01-25
JP2022120125A (ja) 2022-08-17
US20200345734A1 (en) 2020-11-05
IL262102A (en) 2018-11-29
NZ746468A (en) 2023-06-30
AU2017248276B2 (en) 2023-07-13
CA3020170A1 (en) 2017-10-12
KR20230010813A (ko) 2023-01-19
KR102485299B1 (ko) 2023-01-06

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