EA201171228A1 - Производные хиназолиндиона, их получение и их различные терапевтические применения - Google Patents

Производные хиназолиндиона, их получение и их различные терапевтические применения

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Publication number
EA201171228A1
EA201171228A1 EA201171228A EA201171228A EA201171228A1 EA 201171228 A1 EA201171228 A1 EA 201171228A1 EA 201171228 A EA201171228 A EA 201171228A EA 201171228 A EA201171228 A EA 201171228A EA 201171228 A1 EA201171228 A1 EA 201171228A1
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Prior art keywords
therapeutic applications
derivatives
hinazolindion
receiving
different therapeutic
Prior art date
Application number
EA201171228A
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English (en)
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EA021765B1 (ru
Inventor
Анни Клосс
Кристоф Гласс
Жильбер Марсиньяк
Жан-Франсуа Нав
Бертран Виве
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Санофи
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Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=41226702&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=EA201171228(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Санофи filed Critical Санофи
Publication of EA201171228A1 publication Critical patent/EA201171228A1/ru
Publication of EA021765B1 publication Critical patent/EA021765B1/ru

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Abstract

Объектом настоящего изобретения являются производные хиназолиндиона формулы (I), где А означает атом серы или кислорода или сульфоксидную или сульфоновую группу, способы их получения и их терапевтические применения, такие как, среди прочего, в случае рака, диабета, мышечных, костных, сердечно-сосудистых заболеваний, заболеваний центральной нервной системы, заболеваний периферической нервной системы.
EA201171228A 2009-04-09 2010-04-07 Производные хиназолиндиона, их получение и их различные терапевтические применения EA021765B1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR0901760A FR2944282B1 (fr) 2009-04-09 2009-04-09 Derives de quinazolinedione, leur preparation et leurs diverses applications therapeutiques
PCT/FR2010/050664 WO2010116088A2 (fr) 2009-04-09 2010-04-07 Dérivés de quinazolinedione, leur préparation et leurs diverses applications thérapeutiques

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EA201171228A1 true EA201171228A1 (ru) 2012-05-30
EA021765B1 EA021765B1 (ru) 2015-08-31

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JP2015521177A (ja) * 2012-05-07 2015-07-27 オメロス コーポレーション Pde7インヒビターを用いる嗜癖および衝動制御障害の処置
ITMI20130646A1 (it) * 2013-04-19 2014-10-20 Univ Bologna Alma Mater Composti chinazolindionici con attività inibente sulle sirtuine
CN106146413B (zh) * 2015-04-03 2019-01-18 中南大学 2,4-(1h,3h)-喹唑啉二酮衍生物及其合成方法和用途
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GB201517217D0 (en) * 2015-09-29 2015-11-11 Astex Therapeutics Ltd And Cancer Res Technology Ltd Pharmaceutical compounds
WO2024038089A1 (en) 2022-08-18 2024-02-22 Mitodicure Gmbh Use of a therapeutic agent with phosphodiesterase-7 inhibitory activity for the treatment and prevention of diseases associated with chronic fatigue, exhaustion and/or exertional intolerance

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US20120115846A1 (en) 2012-05-10
AU2010233594A1 (en) 2011-11-03
AR076233A1 (es) 2011-05-26
CA2758233A1 (fr) 2010-10-14
TW201040148A (en) 2010-11-16
AU2010233594B2 (en) 2016-07-07
SG175130A1 (en) 2011-11-28
MX2011010639A (es) 2012-01-19
CN102459244B (zh) 2015-07-08
NZ595768A (en) 2012-12-21
SG10201401232QA (en) 2014-08-28
CL2011002522A1 (es) 2012-02-17
KR20120028872A (ko) 2012-03-23
CN102459244A (zh) 2012-05-16
US8722659B2 (en) 2014-05-13
FR2944282B1 (fr) 2013-05-03
FR2944282A1 (fr) 2010-10-15
WO2010116088A3 (fr) 2010-12-16
WO2010116088A2 (fr) 2010-10-14
JP2012523397A (ja) 2012-10-04
MA33255B1 (fr) 2012-05-02
IL215609A0 (en) 2011-12-29
UY32556A (es) 2010-11-30
JP5564101B2 (ja) 2014-07-30
EA021765B1 (ru) 2015-08-31
BRPI1014904A2 (pt) 2016-04-19
ZA201107363B (en) 2012-12-27
EP2417130A2 (fr) 2012-02-15
CO6440583A2 (es) 2012-05-15

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