CO6440583A2 - Derivados de quinazolinadiona, su preparación y sus diversas aplicaciones terapéuticas - Google Patents

Derivados de quinazolinadiona, su preparación y sus diversas aplicaciones terapéuticas

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Publication number
CO6440583A2
CO6440583A2 CO11131880A CO11131880A CO6440583A2 CO 6440583 A2 CO6440583 A2 CO 6440583A2 CO 11131880 A CO11131880 A CO 11131880A CO 11131880 A CO11131880 A CO 11131880A CO 6440583 A2 CO6440583 A2 CO 6440583A2
Authority
CO
Colombia
Prior art keywords
derivatives
therapeutic applications
quinazolinadiona
preparation
various therapeutic
Prior art date
Application number
CO11131880A
Other languages
English (en)
Inventor
Annie Clauss
Christophe Glaess
Gilbert Marciniak
Jean-Francois Nave
Bertrand Vivet
Original Assignee
Sanofi Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=41226702&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CO6440583(A2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Sanofi Sa filed Critical Sanofi Sa
Publication of CO6440583A2 publication Critical patent/CO6440583A2/es

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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D407/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00
    • C07D407/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings
    • C07D407/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/517—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with carbocyclic ring systems, e.g. quinazoline, perimidine
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Abstract

La invención tiene por objeto los derivados de quinazolinadiona de fórmula general (I) con A un átomo de azufre o de oxígeno o un grupo sulfóxido o sulfona, sus procedimientos de obtención y sus aplicaciones terapéuticas tal como cáncer, diabetes, enfermedades musculares, óseas, cardiovasculares, del sistema nervioso central, del sistema nervioso periférico entre otras.
CO11131880A 2009-04-09 2011-10-06 Derivados de quinazolinadiona, su preparación y sus diversas aplicaciones terapéuticas CO6440583A2 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR0901760A FR2944282B1 (fr) 2009-04-09 2009-04-09 Derives de quinazolinedione, leur preparation et leurs diverses applications therapeutiques

Publications (1)

Publication Number Publication Date
CO6440583A2 true CO6440583A2 (es) 2012-05-15

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JP2015521177A (ja) * 2012-05-07 2015-07-27 オメロス コーポレーション Ｐｄｅ７インヒビターを用いる嗜癖および衝動制御障害の処置
ITMI20130646A1 (it) * 2013-04-19 2014-10-20 Univ Bologna Alma Mater Composti chinazolindionici con attività inibente sulle sirtuine
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NZ595768A (en) 2012-12-21
AR076233A1 (es) 2011-05-26
FR2944282A1 (fr) 2010-10-15
IL215609A0 (en) 2011-12-29
KR20120028872A (ko) 2012-03-23
EP2417130A2 (fr) 2012-02-15
JP2012523397A (ja) 2012-10-04
BRPI1014904A2 (pt) 2016-04-19
FR2944282B1 (fr) 2013-05-03
AU2010233594A1 (en) 2011-11-03
CN102459244A (zh) 2012-05-16
AU2010233594B2 (en) 2016-07-07
SG175130A1 (en) 2011-11-28
EA201171228A1 (ru) 2012-05-30
SG10201401232QA (en) 2014-08-28
CL2011002522A1 (es) 2012-02-17
CN102459244B (zh) 2015-07-08
MX2011010639A (es) 2012-01-19
ZA201107363B (en) 2012-12-27
UY32556A (es) 2010-11-30
MA33255B1 (fr) 2012-05-02
WO2010116088A2 (fr) 2010-10-14
JP5564101B2 (ja) 2014-07-30
CA2758233A1 (fr) 2010-10-14
WO2010116088A3 (fr) 2010-12-16
EA021765B1 (ru) 2015-08-31
TW201040148A (en) 2010-11-16
US8722659B2 (en) 2014-05-13

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