UY32556A - Derivados de quinazolinadiona, su preparación y sus diversas aplicaciones terapeúticas - Google Patents

Derivados de quinazolinadiona, su preparación y sus diversas aplicaciones terapeúticas

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Publication number
UY32556A
UY32556A UY0001032556A UY32556A UY32556A UY 32556 A UY32556 A UY 32556A UY 0001032556 A UY0001032556 A UY 0001032556A UY 32556 A UY32556 A UY 32556A UY 32556 A UY32556 A UY 32556A
Authority
UY
Uruguay
Prior art keywords
derivatives
therapeutic applications
quinazolinadiona
preparation
various therapeutic
Prior art date
Application number
UY0001032556A
Other languages
English (en)
Inventor
Annie Clauss
Christophe Glaess
Gilbert Marciniak
Nave Jean-Francois
Bertrand Vivet
Original Assignee
Sanofi Aventis
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=41226702&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=UY32556(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Sanofi Aventis filed Critical Sanofi Aventis
Publication of UY32556A publication Critical patent/UY32556A/es

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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D407/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00
    • C07D407/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings
    • C07D407/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/517—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with carbocyclic ring systems, e.g. quinazoline, perimidine
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Abstract

La invención tiene por objeto los derivados de quinazolinadiona de fórmula general (I) con A un átomo de azufre o de oxígeno o un grupo sulfóxido o sulfona, sus procedimientos de obtención y sus aplicaciones terapéuticas tal como cáncer, diabetes, enfermedades musculares, óseas, cardiovasculares, del sistema nervioso central, del sistema nervioso periférico entre otras.
UY0001032556A 2009-04-09 2010-04-09 Derivados de quinazolinadiona, su preparación y sus diversas aplicaciones terapeúticas UY32556A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR0901760A FR2944282B1 (fr) 2009-04-09 2009-04-09 Derives de quinazolinedione, leur preparation et leurs diverses applications therapeutiques

Publications (1)

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UY32556A true UY32556A (es) 2010-11-30

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ITMI20130646A1 (it) * 2013-04-19 2014-10-20 Univ Bologna Alma Mater Composti chinazolindionici con attività inibente sulle sirtuine
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WO2010116088A3 (fr) 2010-12-16
EP2417130A2 (fr) 2012-02-15
SG10201401232QA (en) 2014-08-28
EA201171228A1 (ru) 2012-05-30
MA33255B1 (fr) 2012-05-02
KR20120028872A (ko) 2012-03-23
SG175130A1 (en) 2011-11-28
FR2944282B1 (fr) 2013-05-03
IL215609A0 (en) 2011-12-29
EA021765B1 (ru) 2015-08-31
CL2011002522A1 (es) 2012-02-17
JP5564101B2 (ja) 2014-07-30
JP2012523397A (ja) 2012-10-04
MX2011010639A (es) 2012-01-19
AU2010233594A1 (en) 2011-11-03
NZ595768A (en) 2012-12-21
WO2010116088A2 (fr) 2010-10-14
TW201040148A (en) 2010-11-16
US8722659B2 (en) 2014-05-13
US20120115846A1 (en) 2012-05-10
CN102459244B (zh) 2015-07-08
AU2010233594B2 (en) 2016-07-07
FR2944282A1 (fr) 2010-10-15
CO6440583A2 (es) 2012-05-15
BRPI1014904A2 (pt) 2016-04-19
CN102459244A (zh) 2012-05-16
AR076233A1 (es) 2011-05-26
ZA201107363B (en) 2012-12-27
CA2758233A1 (fr) 2010-10-14

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