EA200700065A1 - Быстрораспадающаяся диспергирующаяся во рту композиция, содержащая совместно обработанные неволокнистые частицы полиолов и силицифицированную микрокристаллическую целлюлозу - Google Patents
Быстрораспадающаяся диспергирующаяся во рту композиция, содержащая совместно обработанные неволокнистые частицы полиолов и силицифицированную микрокристаллическую целлюлозуInfo
- Publication number
- EA200700065A1 EA200700065A1 EA200700065A EA200700065A EA200700065A1 EA 200700065 A1 EA200700065 A1 EA 200700065A1 EA 200700065 A EA200700065 A EA 200700065A EA 200700065 A EA200700065 A EA 200700065A EA 200700065 A1 EA200700065 A1 EA 200700065A1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- polyols
- microcrystalline cellulose
- silicified microcrystalline
- compositions containing
- fiber particles
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
- A61K9/0056—Mouth soluble or dispersible forms; Suckable, eatable, chewable coherent forms; Forms rapidly disintegrating in the mouth; Lozenges; Lollipops; Bite capsules; Baked products; Baits or other oral forms for animals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
- A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
- A61K9/2077—Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Zoology (AREA)
- Nutrition Science (AREA)
- Physiology (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Medicinal Preparation (AREA)
- Adhesives Or Adhesive Processes (AREA)
- Polysaccharides And Polysaccharide Derivatives (AREA)
Abstract
В заявке описаны новые быстрораспадающиеся фармацевтические композиции, применимые в качестве диспергирующихся во рту таблеток. Композиция, предлагаемая в настоящем изобретении, включает гранулы, содержащие по меньшей мере одно активное вещество, быстрорастворяющийся инертный наполнитель на основе совместно обработанных сахаридов или полиолов, в котором частицы инертного наполнителя обладают неволокнистой микроструктурой, и силицифицированную микрокристаллическую целлюлозу.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
SI200400199 | 2004-07-01 | ||
PCT/EP2005/007091 WO2006002937A1 (en) | 2004-07-01 | 2005-06-30 | Rapidly disintegrating orodispersible composition containing nonfilamentous coprocessed polyols particles and silicified microcrystalline cellulose |
Publications (2)
Publication Number | Publication Date |
---|---|
EA200700065A1 true EA200700065A1 (ru) | 2007-08-31 |
EA013211B1 EA013211B1 (ru) | 2010-04-30 |
Family
ID=34971960
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EA200700065A EA013211B1 (ru) | 2004-07-01 | 2005-06-30 | Быстрораспадающаяся диспергирующаяся во рту лекарственная форма и способ ее приготовления |
Country Status (6)
Country | Link |
---|---|
EP (1) | EP1773292B1 (ru) |
AT (1) | ATE424814T1 (ru) |
DE (1) | DE602005013232D1 (ru) |
EA (1) | EA013211B1 (ru) |
SI (1) | SI1773292T1 (ru) |
WO (1) | WO2006002937A1 (ru) |
Families Citing this family (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2010109019A1 (en) | 2009-03-26 | 2010-09-30 | Royal College Of Surgeons In Ireland | Orodispersible tablets |
WO2011151018A2 (en) * | 2010-06-01 | 2011-12-08 | Cargill, Incorporated | Orodispersible tablets of erythritol and isomalt |
CN102525944A (zh) * | 2012-01-11 | 2012-07-04 | 扬子江药业集团广州海瑞药业有限公司 | 枸地氯雷他定颗粒及其制备方法 |
CN104224733B (zh) * | 2014-09-30 | 2016-08-17 | 蔡伦 | 一种氯雷他定颗粒剂及其制备方法 |
TN2017000497A1 (en) | 2015-06-18 | 2019-04-12 | Mithra Pharmaceuticals S A | Orodispersible dosage unit containing an estetrol component |
MX2017016276A (es) | 2015-06-18 | 2018-06-19 | Mithra Pharmaceuticals S A | Unidad de dosificacion orodispersable que contiene un componente estetrol. |
CN107115307A (zh) * | 2017-06-01 | 2017-09-01 | 江苏黄河药业股份有限公司 | 一种氯雷他定片剂及其制备方法 |
TWI801561B (zh) | 2018-04-19 | 2023-05-11 | 比利時商依思特拉私人有限責任公司 | 化合物及其用於緩解絕經相關症狀的用途 |
JOP20200260A1 (ar) | 2018-04-19 | 2019-10-19 | Estetra Sprl | مركبات واستخداماتها للتخفيف من الأعراض المصاحبة لانقطاع الطمث |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5585115A (en) * | 1995-01-09 | 1996-12-17 | Edward H. Mendell Co., Inc. | Pharmaceutical excipient having improved compressability |
US7118765B2 (en) * | 2001-12-17 | 2006-10-10 | Spi Pharma, Inc. | Co-processed carbohydrate system as a quick-dissolve matrix for solid dosage forms |
-
2005
- 2005-06-30 AT AT05757758T patent/ATE424814T1/de not_active IP Right Cessation
- 2005-06-30 EP EP05757758A patent/EP1773292B1/en active Active
- 2005-06-30 DE DE602005013232T patent/DE602005013232D1/de active Active
- 2005-06-30 EA EA200700065A patent/EA013211B1/ru not_active IP Right Cessation
- 2005-06-30 WO PCT/EP2005/007091 patent/WO2006002937A1/en active Application Filing
- 2005-06-30 SI SI200530701T patent/SI1773292T1/sl unknown
Also Published As
Publication number | Publication date |
---|---|
EA013211B1 (ru) | 2010-04-30 |
SI1773292T1 (sl) | 2009-10-31 |
EP1773292B1 (en) | 2009-03-11 |
WO2006002937A1 (en) | 2006-01-12 |
ATE424814T1 (de) | 2009-03-15 |
EP1773292A1 (en) | 2007-04-18 |
DE602005013232D1 (de) | 2009-04-23 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
EA200700065A1 (ru) | Быстрораспадающаяся диспергирующаяся во рту композиция, содержащая совместно обработанные неволокнистые частицы полиолов и силицифицированную микрокристаллическую целлюлозу | |
HRP20090194T1 (en) | Dry granulated composition comprising emtricitabine and tenofovir df | |
EA200801926A1 (ru) | Таблетки парацетамола с быстрым высвобождением | |
BR0205509A (pt) | Composição compreendendo partìculas finas de liberação prolongada para comprimidos de rápida desintegração na cavidade bucal e método de fabricação da mesma | |
TN2009000093A1 (en) | Pharmaceutical compositions comprising nilotinib or its salt | |
SG165315A1 (en) | Alpha2c adrenoreceptor agonists | |
ATE493972T1 (de) | Gemeinsam aufbereitete mikrokristalline cellulose und zuckeralkohol als hilfsstoff für tablettenformulierungen | |
NO20090554L (no) | Farmasoytiske preparater av memantin | |
EA200801275A1 (ru) | Стабилизированные составы карбоната лантана | |
MX2009004362A (es) | Compuestos mediante benzoilo amino heterociclilo util en el tratamiento de una enfermedad a traves de glk. | |
WO2008017867A3 (en) | Antiretroviral solid oral composition with at least one water insoluble polymer | |
MX2009004439A (es) | Composicion de ibuprofeno. | |
MY139086A (en) | Use of debranched starch in extrusion-spheronization pharmaceutical pellets | |
MXPA05014082A (es) | Acidos biariloximetilarenocarboxilicos. | |
MA27816A1 (fr) | Comprimes de domperidone rapidement hydrodispersables | |
PL2020864T3 (pl) | Sprasowana guma do żucia i sposób jej wytwarzania | |
EA201001108A1 (ru) | Диспергируемые во рту таблетки, содержащие основание эсциталопрама, и способ их получения | |
UA95088C2 (ru) | Композиция, которая содержит наночастички связанные с биосовместимым полимером противоракового агента и снижает аллопецию при химиотерапии, способ ее получения | |
CL2007000789A1 (es) | Compuestos derivados de malonamida, inhibidores de la gamma-secretasa; proceso de preparacion; composicion farmaceutica; y su uso en el tratamiento de la enfermedad de alzheimer. | |
NO20054417L (no) | Fremgangsmate for fremstilling av farmasoytiske preperater i form av fibratholdige tabletter og de derved fremstilte tabletter | |
JP2007161706A (ja) | 安中散含有錠剤 | |
EA200700207A1 (ru) | Твёрдая фармацевтическая композиция, включающая миртазапин | |
BRPI0513005A (pt) | composições contendo nicorandil, processo de preparo e utilização | |
BR0211439A (pt) | Composição de carga sinergìstica e comprimido farmacêutico | |
EA200701525A1 (ru) | Фармацевтическая полимерная композиция для перорального введения тербуталина сульфата с контролируемым высвобождением |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
MM4A | Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s) |
Designated state(s): AM AZ BY KZ KG MD TJ TM |
|
MM4A | Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s) |
Designated state(s): RU |