EA200602202A1 - Фармацевтические композиции, содержащие высшие первичные спирты и эзетимиб, и способ их получения - Google Patents
Фармацевтические композиции, содержащие высшие первичные спирты и эзетимиб, и способ их полученияInfo
- Publication number
- EA200602202A1 EA200602202A1 EA200602202A EA200602202A EA200602202A1 EA 200602202 A1 EA200602202 A1 EA 200602202A1 EA 200602202 A EA200602202 A EA 200602202A EA 200602202 A EA200602202 A EA 200602202A EA 200602202 A1 EA200602202 A1 EA 200602202A1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- ezetimib
- receiving
- pharmaceutical compositions
- compositions containing
- primary alcohols
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/045—Hydroxy compounds, e.g. alcohols; Salts thereof, e.g. alcoholates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/397—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having four-membered rings, e.g. azetidine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
Landscapes
- Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Epidemiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Hematology (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Obesity (AREA)
- Diabetes (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicinal Preparation (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicines Containing Plant Substances (AREA)
Abstract
Представлены новая фармацевтическая композиция, содержащая смесь высших первичных алифатических спиртов из от 24 до 39 атомов углерода, по меньшей мере один другой органический компонент, выбранный из смол и пигментов, углеводородов, сложных эфиров, кетонов и альдегидов, и фенольных соединений, и эзетимиб, его соли, аналоги или их производные, необязательно, с фармацевтически приемлемыми вспомогательными веществами, и способ получения такой композиции. Также представлены способ лечения и использования такой композиции для снижения патологических липидных показателей, связанных с гиперлипидемией.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IN103DE2004 | 2004-01-20 | ||
PCT/IN2005/000025 WO2005067903A1 (en) | 2004-01-20 | 2005-01-19 | Pharmaceutical compositions comprising higher primary alcohols and ezetimibe and process of preparation thereof |
Publications (2)
Publication Number | Publication Date |
---|---|
EA200602202A1 true EA200602202A1 (ru) | 2007-04-27 |
EA010373B1 EA010373B1 (ru) | 2008-08-29 |
Family
ID=34779371
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EA200602202A EA010373B1 (ru) | 2004-01-20 | 2005-01-19 | Фармацевтические композиции, содержащие высшие первичные спирты и эзетимиб, и способ их получения |
Country Status (9)
Country | Link |
---|---|
US (1) | US20070027218A1 (ru) |
EP (1) | EP1755573A1 (ru) |
AP (1) | AP2006003832A0 (ru) |
AU (1) | AU2005205166B8 (ru) |
CA (1) | CA2553985A1 (ru) |
EA (1) | EA010373B1 (ru) |
RS (1) | RS20060437A (ru) |
WO (1) | WO2005067903A1 (ru) |
ZA (1) | ZA200609584B (ru) |
Families Citing this family (14)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB0215579D0 (en) | 2002-07-05 | 2002-08-14 | Astrazeneca Ab | Chemical compounds |
SA04250427A (ar) | 2003-12-23 | 2005-12-03 | استرازينيكا ايه بي | مشتقات ثاني فينيل أزيتيدون |
UY29607A1 (es) | 2005-06-20 | 2007-01-31 | Astrazeneca Ab | Compuestos quimicos |
MY148538A (en) | 2005-06-22 | 2013-04-30 | Astrazeneca Ab | Novel 2-azetidinone derivatives as cholesterol absorption inhibitors for the treatment of hyperlipidaemic conditions |
SA06270191B1 (ar) | 2005-06-22 | 2010-03-29 | استرازينيكا ايه بي | مشتقات من 2- أزيتيدينون جديدة باعتبارها مثبطات لامتصاص الكوليسترول لعلاج حالات فرط نسبة الدهون في الدم |
BRPI0708556A2 (pt) * | 2006-03-06 | 2011-05-31 | Teva Pharma | composição de ezetimiba |
TW200811098A (en) | 2006-04-27 | 2008-03-01 | Astrazeneca Ab | Chemical compounds |
CN101190873B (zh) * | 2006-11-24 | 2010-09-29 | 樊献俄 | 三十烷醇的制备方法 |
WO2008061428A1 (fr) * | 2006-11-24 | 2008-05-29 | Fan Xian E | Formulations pharmaceutiques, utilisation et élaboration du triacontanol |
WO2009158328A1 (en) * | 2008-06-23 | 2009-12-30 | Trustees Of The University Of Pennsylvania | Method for in vivo measurement of reverse cholesterol transport |
EP2216016A1 (en) * | 2009-02-06 | 2010-08-11 | LEK Pharmaceuticals d.d. | Process for the preparation of a pharmaceutical composition comprising ezetimibe |
EP2468258A1 (en) * | 2010-12-22 | 2012-06-27 | LEK Pharmaceuticals d.d. | Process for the preparation of a pharmaceutical composition comprising a low soluble pharmaceutically active ingredient |
CN104940153A (zh) * | 2015-07-23 | 2015-09-30 | 青岛蓝盛洋医药生物科技有限责任公司 | 一种治疗高血脂症的药物依折麦布组合物片剂 |
CN104958261A (zh) * | 2015-08-05 | 2015-10-07 | 青岛蓝盛洋医药生物科技有限责任公司 | 一种治疗心脑血管疾病的药物依折麦布组合物干混悬剂 |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4623667A (en) * | 1985-06-28 | 1986-11-18 | Richardson-Vicks Inc. | Topical treatment of skin inflammatory disorders |
CU22229A1 (es) * | 1992-09-29 | 1996-01-31 | Dalmer Lab Sa | Policosanol, una mezcla de alcoholes alifaticos primarios superiores para hipergregabilidad plaquetaria, los accidentes isquemicos, trombosis e incluso efectividad contra ulceras gastricas quimicamente inducidas y su proceso de obtencion de la caña de azucar. el tratamiento de complicaciones ateroscleroticas tales como la |
US6225354B1 (en) * | 1999-06-21 | 2001-05-01 | Cholesterol Control Laboratories, Inc. | High molecular weight primary aliphatic alcohols obtained from beeswax and pharmaceutical use thereof |
US6596776B2 (en) * | 1999-06-21 | 2003-07-22 | Hauser, Inc. | High molecular weight primary aliphatic alcohols obtained from natural products and uses thereof |
ATE337782T1 (de) * | 2000-08-17 | 2006-09-15 | Merck & Co Inc | Cyclopentylmodulatoren der chemokin-rezeptor- aktivität |
IL156552A0 (en) * | 2000-12-21 | 2004-01-04 | Aventis Pharma Gmbh | Diphenyl azetidinone derivatives, method for the production thereof, medicaments containing these compounds, and their use |
WO2003103632A1 (en) * | 2002-06-10 | 2003-12-18 | Elan Pharma International, Ltd. | Nanoparticulate polycosanol formulations and novel polycosanol combinations |
-
2005
- 2005-01-19 WO PCT/IN2005/000025 patent/WO2005067903A1/en active Application Filing
- 2005-01-19 EA EA200602202A patent/EA010373B1/ru not_active IP Right Cessation
- 2005-01-19 RS RSP-2006/0437A patent/RS20060437A/sr unknown
- 2005-01-19 CA CA002553985A patent/CA2553985A1/en not_active Abandoned
- 2005-01-19 ZA ZA200609584A patent/ZA200609584B/xx unknown
- 2005-01-19 AU AU2005205166A patent/AU2005205166B8/en not_active Ceased
- 2005-01-19 EP EP05709166A patent/EP1755573A1/en not_active Withdrawn
- 2005-01-19 AP AP2006003832A patent/AP2006003832A0/xx unknown
-
2006
- 2006-07-19 US US11/489,253 patent/US20070027218A1/en not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
AU2005205166B8 (en) | 2008-04-24 |
US20070027218A1 (en) | 2007-02-01 |
WO2005067903A8 (en) | 2005-11-03 |
AU2005205166A1 (en) | 2005-07-28 |
AU2005205166B2 (en) | 2008-04-03 |
WO2005067903A1 (en) | 2005-07-28 |
EP1755573A1 (en) | 2007-02-28 |
CA2553985A1 (en) | 2005-07-28 |
RS20060437A (en) | 2008-11-28 |
EA010373B1 (ru) | 2008-08-29 |
AP2006003832A0 (en) | 2006-12-31 |
ZA200609584B (en) | 2008-06-25 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
MM4A | Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s) |
Designated state(s): AM AZ BY KZ KG MD TJ TM RU |