EA200501883A1 - Таблетки дерамциклан-фумарата - Google Patents

Таблетки дерамциклан-фумарата

Info

Publication number
EA200501883A1
EA200501883A1 EA200501883A EA200501883A EA200501883A1 EA 200501883 A1 EA200501883 A1 EA 200501883A1 EA 200501883 A EA200501883 A EA 200501883A EA 200501883 A EA200501883 A EA 200501883A EA 200501883 A1 EA200501883 A1 EA 200501883A1
Authority
EA
Eurasian Patent Office
Prior art keywords
fumarate
deramciclan
weight
deramcyclan
fumarate tablets
Prior art date
Application number
EA200501883A
Other languages
English (en)
Other versions
EA009681B1 (ru
Inventor
Паль Фекете
Ласлоне Марошхелйи
Зольт Жигмонд
Ласлоне Гора
Магдольна Левентисне Хусар
Иштванне Ямбор
Йожеф Тари
Original Assignee
Эгиш Дьёдьсердьяр Рт.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Эгиш Дьёдьсердьяр Рт. filed Critical Эгиш Дьёдьсердьяр Рт.
Publication of EA200501883A1 publication Critical patent/EA200501883A1/ru
Publication of EA009681B1 publication Critical patent/EA009681B1/ru

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/2027Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/22Anxiolytics

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Biomedical Technology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Neurology (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Adhesives Or Adhesive Processes (AREA)
  • Compositions Of Macromolecular Compounds (AREA)
  • Materials For Medical Uses (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

Изобретение относится к таблеткам, содержащим дерамциклан-фумарат формулы (I), содержащим (относительно общей массы) более чем 50 мас.% дерамциклан-фумарата, 5-20 мас.% связующего вещества, 5-20 мас.% микрокристаллической целлюлозы, имеющей средний размер частиц меньше 30 мкм, 1-10 мас.% разрыхлителя, 0,5-4 мас.% смазывающего вещества, 0,5-4 мас.% антиадгезионного вещества и 0-30 мас.% наполнителя. Дерамциклан-фумарат является известным анксиолитическим активным компонентом.
EA200501883A 2003-06-03 2004-06-03 Таблетка дерамцикланфумарата и способ её приготовления EA009681B1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
HU0301537A HUP0301537A3 (en) 2003-06-03 2003-06-03 Deramcyclane fumarate tablets and process for producing them
PCT/HU2004/000058 WO2004105743A1 (en) 2003-06-03 2004-06-03 Deramciclane-fumarate tablets

Publications (2)

Publication Number Publication Date
EA200501883A1 true EA200501883A1 (ru) 2006-06-30
EA009681B1 EA009681B1 (ru) 2008-02-28

Family

ID=90001686

Family Applications (1)

Application Number Title Priority Date Filing Date
EA200501883A EA009681B1 (ru) 2003-06-03 2004-06-03 Таблетка дерамцикланфумарата и способ её приготовления

Country Status (25)

Country Link
US (1) US20060258745A1 (ru)
EP (1) EP1628648B1 (ru)
JP (1) JP2006526603A (ru)
KR (1) KR20060015746A (ru)
CN (1) CN1832733A (ru)
AT (1) ATE381325T1 (ru)
AU (1) AU2004243240A1 (ru)
BG (1) BG109404A (ru)
BR (1) BRPI0410909A (ru)
CA (1) CA2527431A1 (ru)
CZ (1) CZ2005817A3 (ru)
DE (1) DE602004010803D1 (ru)
EA (1) EA009681B1 (ru)
HR (1) HRP20050979A2 (ru)
HU (1) HUP0301537A3 (ru)
IL (1) IL172133A0 (ru)
IS (1) IS8202A (ru)
MX (1) MXPA05013020A (ru)
NO (1) NO20056220L (ru)
PL (1) PL378540A1 (ru)
RS (1) RS20050898A (ru)
SK (1) SK51112005A3 (ru)
UA (1) UA80209C2 (ru)
WO (1) WO2004105743A1 (ru)
ZA (1) ZA200510139B (ru)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI399223B (zh) * 2006-09-15 2013-06-21 Daiichi Sankyo Co Ltd 奧美沙坦酯及氨氯地平之固體劑型
CA2937365C (en) 2016-03-29 2018-09-18 F. Hoffmann-La Roche Ag Granulate formulation of 5-methyl-1-phenyl-2-(1h)-pyridone and method of making the same
US11478467B2 (en) 2017-05-04 2022-10-25 Sreenivasarao Vepachedu Targeted drug rescue with novel compositions, combinations, and methods thereof
CN110973635B (zh) * 2019-12-26 2022-07-29 汤臣倍健股份有限公司 一种辅料组合物及益生菌片剂
CN114643014B (zh) * 2022-05-07 2024-02-13 佛山市锦厨食品科技有限公司 一种可提高颗粒状鸡精的成型速度的食品用造粒机

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HU179164B (en) * 1979-12-14 1982-08-28 Egyt Gyogyszervegyeszeti Gyar Process for producing cycloalkyl-ethers of alkanolamines
HU214588B (hu) * 1994-07-01 1998-04-28 EGIS Gyógyszergyár Rt. Eljárás bicikloheptán-származékot tartalmazó, CCK-rendszer gátló hatású gyógyászati készítmények előállítására
SI20624A (sl) * 1998-12-18 2002-02-28 Abbott Laboratories Formulacija divalproeks natrija za kontrolirano sproščanje
HUP0103017A3 (en) * 2001-07-18 2004-05-28 Egis Gyogyszergyar Nyilvanosan Pharmaceutical composition for the treatment of diseases caused by impairment of cognitive functions and its use
UA75831C2 (en) * 2002-04-29 2006-05-15 Egyt Gyogyszervegyeszeti Gyar Process for preparation of tablets from pharmaceutically active ingredients having unfavourable tabletting properties with the use of granulating liquid containing microcrystalline cellulose

Also Published As

Publication number Publication date
IL172133A0 (en) 2006-04-10
ATE381325T1 (de) 2008-01-15
BRPI0410909A (pt) 2006-06-27
HUP0301537D0 (en) 2003-08-28
EP1628648B1 (en) 2007-12-19
CA2527431A1 (en) 2004-12-09
DE602004010803D1 (de) 2008-01-31
RS20050898A (en) 2008-04-04
AU2004243240A1 (en) 2004-12-09
CN1832733A (zh) 2006-09-13
MXPA05013020A (es) 2006-03-17
CZ2005817A3 (cs) 2006-04-12
US20060258745A1 (en) 2006-11-16
SK51112005A3 (sk) 2006-06-01
BG109404A (en) 2006-11-30
HUP0301537A2 (hu) 2005-03-29
NO20056220L (no) 2006-03-02
UA80209C2 (en) 2007-08-27
PL378540A1 (pl) 2006-05-02
EA009681B1 (ru) 2008-02-28
HRP20050979A2 (en) 2006-03-31
HUP0301537A3 (en) 2005-07-28
ZA200510139B (en) 2007-03-28
EP1628648A1 (en) 2006-03-01
WO2004105743A1 (en) 2004-12-09
KR20060015746A (ko) 2006-02-20
JP2006526603A (ja) 2006-11-24
IS8202A (is) 2005-12-28

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Legal Events

Date Code Title Description
MM4A Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s)

Designated state(s): AM AZ BY KZ KG MD TJ TM RU