EA200101235A1 - СПОСОБ ПОЛУЧЕНИЯ ЗАМЕЩЕННЫХ [1,4] ДИАЗЕПИНО [6,7,1-hi]ИНДОЛ-4-ОНОВ - Google Patents

СПОСОБ ПОЛУЧЕНИЯ ЗАМЕЩЕННЫХ [1,4] ДИАЗЕПИНО [6,7,1-hi]ИНДОЛ-4-ОНОВ

Info

Publication number
EA200101235A1
EA200101235A1 EA200101235A EA200101235A EA200101235A1 EA 200101235 A1 EA200101235 A1 EA 200101235A1 EA 200101235 A EA200101235 A EA 200101235A EA 200101235 A EA200101235 A EA 200101235A EA 200101235 A1 EA200101235 A1 EA 200101235A1
Authority
EA
Eurasian Patent Office
Prior art keywords
diazepino
indol
head
obtaining substituted
obtaining
Prior art date
Application number
EA200101235A
Other languages
English (en)
Other versions
EA004675B1 (ru
Inventor
Патрик Бернарделли
Original Assignee
Уорнер-Ламберт Компани
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Уорнер-Ламберт Компани filed Critical Уорнер-Ламберт Компани
Publication of EA200101235A1 publication Critical patent/EA200101235A1/ru
Publication of EA004675B1 publication Critical patent/EA004675B1/ru

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/06—Peri-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pulmonology (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

Abstract

Способ получения энантиомерно чистого диазепиноиндолона формулыпри котором осуществляют внутримолекулярную циклизацию продукта формулыгде А, В, X, X, Z, Z, Zи R являются такими, как они определены в описании, в присутствии катализатора, представляющего собой слабую кислоту Льюиса.Международная заявка была опубликована вместе с отчетом о международном поиске.
EA200101235A 1999-07-02 2000-06-29 СПОСОБ ПОЛУЧЕНИЯ ЗАМЕЩЕННЫХ [1,4]ДИАЗЕПИНО[6,7,1-hi]ИНДОЛ-4-ОНОВ EA004675B1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9908537A FR2795731B1 (fr) 1999-07-02 1999-07-02 PROCEDE DE PREPARATION DE [1,4] DIAZEPINO [6,7,1-hi] INDOL-4-ONES SUBSTITUEES
PCT/FR2000/001839 WO2001002403A1 (fr) 1999-07-02 2000-06-29 PROCEDE DE PREPARATION DE [1,4]DIAZEPINO[6,7,1-hi]INDOL-4-ONES SUBSTITUEES

Publications (2)

Publication Number Publication Date
EA200101235A1 true EA200101235A1 (ru) 2002-06-27
EA004675B1 EA004675B1 (ru) 2004-06-24

Family

ID=9547630

Family Applications (1)

Application Number Title Priority Date Filing Date
EA200101235A EA004675B1 (ru) 1999-07-02 2000-06-29 СПОСОБ ПОЛУЧЕНИЯ ЗАМЕЩЕННЫХ [1,4]ДИАЗЕПИНО[6,7,1-hi]ИНДОЛ-4-ОНОВ

Country Status (31)

Country Link
US (1) US6689881B1 (ru)
EP (1) EP1196418B1 (ru)
JP (1) JP2003503498A (ru)
KR (1) KR20020016644A (ru)
CN (1) CN1166668C (ru)
AP (1) AP2001002378A0 (ru)
AT (1) ATE269334T1 (ru)
AU (1) AU772966B2 (ru)
BG (1) BG106264A (ru)
BR (1) BR0012532A (ru)
CA (1) CA2376707A1 (ru)
CZ (1) CZ20014681A3 (ru)
DE (1) DE60011619D1 (ru)
DZ (1) DZ3260A1 (ru)
EA (1) EA004675B1 (ru)
EE (1) EE200100700A (ru)
FR (1) FR2795731B1 (ru)
HR (1) HRP20010952A2 (ru)
HU (1) HUP0201635A3 (ru)
IL (1) IL147364A0 (ru)
IS (1) IS6211A (ru)
MX (1) MXPA02000257A (ru)
NO (1) NO20016271L (ru)
NZ (1) NZ516287A (ru)
OA (1) OA11981A (ru)
PL (1) PL357075A1 (ru)
SK (1) SK19242001A3 (ru)
TR (1) TR200103857T2 (ru)
WO (1) WO2001002403A1 (ru)
YU (1) YU92001A (ru)
ZA (1) ZA200200114B (ru)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2006297300B2 (en) * 2005-09-29 2012-05-10 Albany Molecular Research, Inc. Process for production of delta-9-tetrahydrocannabinol
US12029718B2 (en) 2021-11-09 2024-07-09 Cct Sciences, Llc Process for production of essentially pure delta-9-tetrahydrocannabinol

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5256801A (en) 1992-08-14 1993-10-26 Napro Biotherapeutics, Inc. Processes of converting taxanes into 10-deacetylbaccatin III
US5342971A (en) 1992-12-29 1994-08-30 The Australian National University Process for the preparation of dibenzo[b,d]pyrans
GB9305806D0 (en) 1993-03-20 1993-05-05 Glaxo Spa Chemical compounds
FR2762841B1 (fr) * 1997-04-30 1999-07-02 Jouveinal Inst Rech Diazepino-indolones inhibitrices de phosphodiesterases iv

Also Published As

Publication number Publication date
CA2376707A1 (en) 2001-01-11
EP1196418A1 (fr) 2002-04-17
WO2001002403A1 (fr) 2001-01-11
MXPA02000257A (es) 2003-08-20
TR200103857T2 (tr) 2003-01-21
FR2795731B1 (fr) 2001-09-07
CN1166668C (zh) 2004-09-15
HUP0201635A3 (en) 2004-12-28
AU772966B2 (en) 2004-05-13
KR20020016644A (ko) 2002-03-04
NZ516287A (en) 2003-06-30
JP2003503498A (ja) 2003-01-28
OA11981A (fr) 2006-04-17
AU6289600A (en) 2001-01-22
IL147364A0 (en) 2002-08-14
NO20016271L (no) 2001-12-28
FR2795731A1 (fr) 2001-01-05
EP1196418B1 (fr) 2004-06-16
HRP20010952A2 (en) 2003-06-30
PL357075A1 (en) 2004-07-12
NO20016271D0 (no) 2001-12-20
CN1362960A (zh) 2002-08-07
US6689881B1 (en) 2004-02-10
AP2001002378A0 (en) 2001-12-31
DE60011619D1 (de) 2004-07-22
YU92001A (sh) 2004-09-03
CZ20014681A3 (cs) 2002-08-14
HUP0201635A2 (en) 2002-09-28
IS6211A (is) 2001-12-21
BG106264A (en) 2002-08-30
BR0012532A (pt) 2002-04-02
DZ3260A1 (fr) 2001-01-11
ATE269334T1 (de) 2004-07-15
EA004675B1 (ru) 2004-06-24
ZA200200114B (en) 2002-10-30
SK19242001A3 (sk) 2002-11-06
EE200100700A (et) 2003-04-15

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Legal Events

Date Code Title Description
MM4A Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s)

Designated state(s): AM AZ BY KZ KG MD TJ TM RU