EA024184B1 - Стоматологическое анестезирующее средство для интраназального введения, содержащее тетракаин и вазоконстриктор - Google Patents
Стоматологическое анестезирующее средство для интраназального введения, содержащее тетракаин и вазоконстриктор Download PDFInfo
- Publication number
- EA024184B1 EA024184B1 EA201171215A EA201171215A EA024184B1 EA 024184 B1 EA024184 B1 EA 024184B1 EA 201171215 A EA201171215 A EA 201171215A EA 201171215 A EA201171215 A EA 201171215A EA 024184 B1 EA024184 B1 EA 024184B1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- pharmaceutical composition
- specified
- tetracaine
- subject
- nasal
- Prior art date
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4164—1,3-Diazoles
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- A61K31/21—Esters, e.g. nitroglycerine, selenocyanates
- A61K31/215—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
- A61K31/235—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids having an aromatic ring attached to a carboxyl group
- A61K31/24—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids having an aromatic ring attached to a carboxyl group having an amino or nitro group
- A61K31/245—Amino benzoic acid types, e.g. procaine, novocaine
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
- A61K47/10—Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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- A61K9/0012—Galenical forms characterised by the site of application
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- A61M—DEVICES FOR INTRODUCING MEDIA INTO, OR ONTO, THE BODY; DEVICES FOR TRANSDUCING BODY MEDIA OR FOR TAKING MEDIA FROM THE BODY; DEVICES FOR PRODUCING OR ENDING SLEEP OR STUPOR
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Landscapes
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- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
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- Anesthesiology (AREA)
- Emergency Medicine (AREA)
- Otolaryngology (AREA)
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- Chemical Kinetics & Catalysis (AREA)
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- Heart & Thoracic Surgery (AREA)
- Hematology (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Oil, Petroleum & Natural Gas (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (2)
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|---|---|---|---|
| US16668009P | 2009-04-03 | 2009-04-03 | |
| PCT/US2010/001002 WO2010114622A1 (en) | 2009-04-03 | 2010-04-02 | Dental anesthetic comprising tetracaine and a vasoconstrictor for intranasal administration |
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| EA201171215A1 EA201171215A1 (ru) | 2012-07-30 |
| EA024184B1 true EA024184B1 (ru) | 2016-08-31 |
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| MX (1) | MX2011010445A (enExample) |
| NZ (2) | NZ595376A (enExample) |
| PL (1) | PL2413899T3 (enExample) |
| PT (1) | PT2413899T (enExample) |
| WO (1) | WO2010114622A1 (enExample) |
| ZA (2) | ZA201107011B (enExample) |
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| JP5788864B2 (ja) | 2009-04-03 | 2015-10-07 | セイント レナタス， エルエルシー | 鼻腔内投与用のテトラカインおよび血管収縮薬を含む歯科用麻酔剤 |
| NZ629475A (en) | 2012-09-28 | 2017-03-31 | St Renatus Llc | Pharmaceutical composition comprising benzyl alcohol for the treatment of migraines |
| WO2015103450A1 (en) * | 2014-01-01 | 2015-07-09 | Real Time Imaging Technologies, Llc | Improved local anesthetic solution for dental and/or contrast media use |
| AU2015277272A1 (en) * | 2014-06-16 | 2017-01-12 | Loewi LLC | Methods of anesthetizing nerve tissue in the trigeminal nerve pathway and medical uses thereof |
| EA201791448A1 (ru) * | 2014-12-23 | 2017-11-30 | СТ. РЕНАТУС, ЭлЭлСи | Анестетик на основе тетракаина |
| WO2016115117A1 (en) | 2015-01-12 | 2016-07-21 | Real Time Imaging Technologies, Llc | Low-dose x-ray imaging system |
| US10039830B2 (en) * | 2016-03-04 | 2018-08-07 | Cetylite Industries, Inc. | Topical anesthetic composition |
| WO2017210390A1 (en) * | 2016-06-01 | 2017-12-07 | St. Renatus, Llc | Intranasal dental anesthetic |
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| CN111494310A (zh) * | 2020-04-29 | 2020-08-07 | 周晓玲 | 一种局部麻醉药物的制备及使用方法 |
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