AU2010232995C1 - Dental anesthetic comprising tetracaine and a vasoconstrictor for intranasal administration - Google Patents
Dental anesthetic comprising tetracaine and a vasoconstrictor for intranasal administration Download PDFInfo
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- AU2010232995C1 AU2010232995C1 AU2010232995A AU2010232995A AU2010232995C1 AU 2010232995 C1 AU2010232995 C1 AU 2010232995C1 AU 2010232995 A AU2010232995 A AU 2010232995A AU 2010232995 A AU2010232995 A AU 2010232995A AU 2010232995 C1 AU2010232995 C1 AU 2010232995C1
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- pharmaceutical composition
- nasal
- tetracaine
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- 229960002372 tetracaine Drugs 0.000 title claims abstract description 73
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- WYWIFABBXFUGLM-UHFFFAOYSA-N oxymetazoline Chemical group CC1=CC(C(C)(C)C)=C(O)C(C)=C1CC1=NCCN1 WYWIFABBXFUGLM-UHFFFAOYSA-N 0.000 claims description 52
- 210000003928 nasal cavity Anatomy 0.000 claims description 48
- 210000005036 nerve Anatomy 0.000 claims description 33
- WVDDGKGOMKODPV-UHFFFAOYSA-N Benzyl alcohol Chemical group OCC1=CC=CC=C1 WVDDGKGOMKODPV-UHFFFAOYSA-N 0.000 claims description 30
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- Oil, Petroleum & Natural Gas (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Priority Applications (1)
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|---|---|---|---|
| AU2015242984A AU2015242984B2 (en) | 2009-04-03 | 2015-10-13 | Dental Anesthetic Comprising Tetracaine and a Vasoconstrictor For Intranasal Administration |
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| US16668009P | 2009-04-03 | 2009-04-03 | |
| US61/166,680 | 2009-04-03 | ||
| PCT/US2010/001002 WO2010114622A1 (en) | 2009-04-03 | 2010-04-02 | Dental anesthetic comprising tetracaine and a vasoconstrictor for intranasal administration |
Related Child Applications (1)
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| AU2015242984A Division AU2015242984B2 (en) | 2009-04-03 | 2015-10-13 | Dental Anesthetic Comprising Tetracaine and a Vasoconstrictor For Intranasal Administration |
Publications (3)
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| AU2015242984A Expired - Fee Related AU2015242984B2 (en) | 2009-04-03 | 2015-10-13 | Dental Anesthetic Comprising Tetracaine and a Vasoconstrictor For Intranasal Administration |
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| PT (1) | PT2413899T (enExample) |
| WO (1) | WO2010114622A1 (enExample) |
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Families Citing this family (12)
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| JP5788864B2 (ja) | 2009-04-03 | 2015-10-07 | セイント レナタス， エルエルシー | 鼻腔内投与用のテトラカインおよび血管収縮薬を含む歯科用麻酔剤 |
| NZ629475A (en) | 2012-09-28 | 2017-03-31 | St Renatus Llc | Pharmaceutical composition comprising benzyl alcohol for the treatment of migraines |
| WO2015103450A1 (en) * | 2014-01-01 | 2015-07-09 | Real Time Imaging Technologies, Llc | Improved local anesthetic solution for dental and/or contrast media use |
| AU2015277272A1 (en) * | 2014-06-16 | 2017-01-12 | Loewi LLC | Methods of anesthetizing nerve tissue in the trigeminal nerve pathway and medical uses thereof |
| EA201791448A1 (ru) * | 2014-12-23 | 2017-11-30 | СТ. РЕНАТУС, ЭлЭлСи | Анестетик на основе тетракаина |
| WO2016115117A1 (en) | 2015-01-12 | 2016-07-21 | Real Time Imaging Technologies, Llc | Low-dose x-ray imaging system |
| US10039830B2 (en) * | 2016-03-04 | 2018-08-07 | Cetylite Industries, Inc. | Topical anesthetic composition |
| WO2017210390A1 (en) * | 2016-06-01 | 2017-12-07 | St. Renatus, Llc | Intranasal dental anesthetic |
| CA3122363A1 (en) | 2018-12-19 | 2020-06-25 | Nortic Holdings Inc. | Therapeutic composition of intranasal lidocaine |
| CN111494310A (zh) * | 2020-04-29 | 2020-08-07 | 周晓玲 | 一种局部麻醉药物的制备及使用方法 |
| EP4648760A1 (en) * | 2023-01-13 | 2025-11-19 | Smilanich, Michael D. | Composition for local anesthesia and uses thereof |
| GB2628149A (en) * | 2023-03-16 | 2024-09-18 | Lee Nathaniel Wurie | Nasal spray for performing sphenopalatine ganglion block |
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| US3832460A (en) * | 1971-03-19 | 1974-08-27 | C Kosti | Anesthetic-vasoconstrictor-antihistamine composition for the treatment of hypertrophied oral tissue |
| US5585398A (en) * | 1994-07-15 | 1996-12-17 | Ernst; Amy A. | Topical anesthetic comprising lidocaine, adrenaline, and tetracaine, and its method of use |
| US6413499B1 (en) * | 2000-01-06 | 2002-07-02 | Bryan M. Clay | Methods and kits for maxillary dental anesthesia by means of a nasal deliverable anesthetic |
| US20040131665A1 (en) * | 1999-10-22 | 2004-07-08 | Wepfer Scott T. | Topical anesthetic formulation |
| JP2004196786A (ja) * | 2002-12-03 | 2004-07-15 | Taisho Pharmaceut Co Ltd | 難溶性抗ウイルス成分含有水溶性外用剤組成物 |
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| US5209724A (en) | 1988-04-11 | 1993-05-11 | Dhaliwal Avtar S | Composite anesthetic article and method of use |
| AU4673993A (en) | 1992-07-28 | 1994-02-14 | Procter & Gamble Company, The | Pharmaceutical composition for topical use containing a crosslinked cationic polymer and an alkoxylated ether |
| US5854269A (en) | 1993-11-19 | 1998-12-29 | Schering-Plough Healthcare Products, Inc. | Nasal spray compositions |
| US6075059A (en) | 1999-02-24 | 2000-06-13 | The Ohio State University | Compositions for dental anesthesia |
| US20040045546A1 (en) | 2002-09-05 | 2004-03-11 | Peirce Management, Llc | Pharmaceutical delivery system for oral inhalation through nebulization consisting of inert substrate impregnated with substance (S) to be solubilized or suspended prior to use |
| ES2223277B1 (es) * | 2003-06-19 | 2006-03-01 | Fernando Bouffard Fita | Composicion anestesica para administracion topica. |
| WO2005065696A1 (en) | 2004-01-01 | 2005-07-21 | Panacea Biotec Ltd. | Pharmaceutical compositions comprising an extract of euphorbia prostrata |
| US20060052305A1 (en) * | 2004-05-10 | 2006-03-09 | Nastech Pharmaceutical Company Inc. | Method of treating osteoporosis using intranasal parathyroid hormone |
| WO2007050543A2 (en) | 2005-10-24 | 2007-05-03 | Collegium Pharmaceutical, Inc. | Topical pharmaceutical foam composition |
| US9252862B2 (en) | 2008-09-17 | 2016-02-02 | Qualcomm Incorporated | MIMO preamble for initial access with an unknown number of transmit antennas |
| JP5788864B2 (ja) * | 2009-04-03 | 2015-10-07 | セイント レナタス， エルエルシー | 鼻腔内投与用のテトラカインおよび血管収縮薬を含む歯科用麻酔剤 |
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2010
- 2010-04-02 JP JP2012503429A patent/JP5788864B2/ja not_active Expired - Fee Related
- 2010-04-02 CN CN201080020599.5A patent/CN102421416B/zh not_active Expired - Fee Related
- 2010-04-02 CA CA2757032A patent/CA2757032C/en active Active
- 2010-04-02 KR KR1020117026165A patent/KR101747979B1/ko not_active Expired - Fee Related
- 2010-04-02 PT PT107141194T patent/PT2413899T/pt unknown
- 2010-04-02 EP EP10714119.4A patent/EP2413899B1/en active Active
- 2010-04-02 DK DK10714119.4T patent/DK2413899T3/da active
- 2010-04-02 PL PL10714119T patent/PL2413899T3/pl unknown
- 2010-04-02 KR KR1020177005466A patent/KR20170026639A/ko not_active Ceased
- 2010-04-02 CN CN201410169695.6A patent/CN103932973B/zh not_active Expired - Fee Related
- 2010-04-02 NZ NZ595376A patent/NZ595376A/xx unknown
- 2010-04-02 NZ NZ612063A patent/NZ612063A/en not_active IP Right Cessation
- 2010-04-02 MX MX2011010445A patent/MX2011010445A/es active IP Right Grant
- 2010-04-02 WO PCT/US2010/001002 patent/WO2010114622A1/en not_active Ceased
- 2010-04-02 AU AU2010232995A patent/AU2010232995C1/en not_active Ceased
- 2010-04-02 US US13/262,704 patent/US8580282B2/en not_active Expired - Fee Related
- 2010-04-02 BR BRPI1010303A patent/BRPI1010303A2/pt not_active IP Right Cessation
- 2010-04-02 ES ES10714119T patent/ES2861064T3/es active Active
- 2010-04-02 EA EA201171215A patent/EA024184B1/ru not_active IP Right Cessation
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2011
- 2011-09-26 ZA ZA2011/07011A patent/ZA201107011B/en unknown
- 2011-10-02 IL IL215489A patent/IL215489A0/en unknown
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2013
- 2013-09-13 US US14/027,033 patent/US9308191B2/en not_active Expired - Fee Related
- 2013-12-11 ZA ZA2013/09321A patent/ZA201309321B/en unknown
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2014
- 2014-10-15 JP JP2014210422A patent/JP2015034167A/ja not_active Withdrawn
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2015
- 2015-10-13 AU AU2015242984A patent/AU2015242984B2/en not_active Expired - Fee Related
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2016
- 2016-03-02 US US15/058,324 patent/US9855247B2/en active Active
- 2016-11-15 JP JP2016222091A patent/JP2017031226A/ja active Pending
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2017
- 2017-04-18 US US15/490,011 patent/US10456377B2/en active Active
- 2017-04-27 US US15/498,986 patent/US20170326111A1/en not_active Abandoned
- 2017-04-27 US US15/498,991 patent/US10420750B2/en active Active
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2020
- 2020-05-12 US US16/872,657 patent/US20200268715A1/en not_active Abandoned
Patent Citations (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3832460A (en) * | 1971-03-19 | 1974-08-27 | C Kosti | Anesthetic-vasoconstrictor-antihistamine composition for the treatment of hypertrophied oral tissue |
| US5585398A (en) * | 1994-07-15 | 1996-12-17 | Ernst; Amy A. | Topical anesthetic comprising lidocaine, adrenaline, and tetracaine, and its method of use |
| US20040131665A1 (en) * | 1999-10-22 | 2004-07-08 | Wepfer Scott T. | Topical anesthetic formulation |
| US6413499B1 (en) * | 2000-01-06 | 2002-07-02 | Bryan M. Clay | Methods and kits for maxillary dental anesthesia by means of a nasal deliverable anesthetic |
| JP2004196786A (ja) * | 2002-12-03 | 2004-07-15 | Taisho Pharmaceut Co Ltd | 難溶性抗ウイルス成分含有水溶性外用剤組成物 |
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