DOP2006000028A - Pirroles sustituidos, composiciones que los contienen, proceso de fabricación y utilización - Google Patents
Pirroles sustituidos, composiciones que los contienen, proceso de fabricación y utilizaciónInfo
- Publication number
- DOP2006000028A DOP2006000028A DO2006000028A DO2006000028A DOP2006000028A DO P2006000028 A DOP2006000028 A DO P2006000028A DO 2006000028 A DO2006000028 A DO 2006000028A DO 2006000028 A DO2006000028 A DO 2006000028A DO P2006000028 A DOP2006000028 A DO P2006000028A
- Authority
- DO
- Dominican Republic
- Prior art keywords
- compositions
- manufacturing
- pirroles
- replaced
- contain
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/30—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
- C07D207/34—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pyrrole Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
Pirroles sustituidos, composiciones que los contienen, proceso de fabricación y utilización. La presente invención se refiere particularmente a la preparación de pirroles sustituidos, a las composiciones que los contienen, a su proceso de preparación, y a su utilización como medicamento, en particular como agentes anticancerígenos.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR0501354A FR2881742B1 (fr) | 2005-02-10 | 2005-02-10 | Pyrroles substitues, compositions les contenant, procede de fabrication et utilisation |
Publications (1)
Publication Number | Publication Date |
---|---|
DOP2006000028A true DOP2006000028A (es) | 2006-09-15 |
Family
ID=35478244
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DO2006000028A DOP2006000028A (es) | 2005-02-10 | 2006-02-02 | Pirroles sustituidos, composiciones que los contienen, proceso de fabricación y utilización |
Country Status (36)
Country | Link |
---|---|
US (1) | US7592365B2 (es) |
EP (1) | EP1851198B1 (es) |
JP (1) | JP2008530061A (es) |
KR (1) | KR20070101317A (es) |
CN (1) | CN101115716A (es) |
AR (1) | AR052571A1 (es) |
AT (1) | ATE419234T1 (es) |
AU (1) | AU2006212106A1 (es) |
BR (1) | BRPI0606955A2 (es) |
CA (1) | CA2596822A1 (es) |
CR (1) | CR9231A (es) |
CY (1) | CY1108916T1 (es) |
DE (1) | DE602006004566D1 (es) |
DK (1) | DK1851198T3 (es) |
DO (1) | DOP2006000028A (es) |
EA (1) | EA013060B1 (es) |
ES (1) | ES2319926T3 (es) |
FR (1) | FR2881742B1 (es) |
GT (1) | GT200600048A (es) |
HR (1) | HRP20090158T1 (es) |
IL (1) | IL184488A0 (es) |
MA (1) | MA29248B1 (es) |
MX (1) | MX2007008789A (es) |
MY (1) | MY142082A (es) |
NO (1) | NO20074528L (es) |
PA (1) | PA8661601A1 (es) |
PE (1) | PE20061086A1 (es) |
PL (1) | PL1851198T3 (es) |
PT (1) | PT1851198E (es) |
RS (1) | RS50806B (es) |
SI (1) | SI1851198T1 (es) |
TN (1) | TNSN07241A1 (es) |
TW (1) | TW200640858A (es) |
UY (1) | UY29371A1 (es) |
WO (1) | WO2006084996A1 (es) |
ZA (1) | ZA200706157B (es) |
Families Citing this family (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2881426B1 (fr) | 2005-02-03 | 2007-03-30 | Aventis Pharma Sa | Pyrolles et imidazoles substitues, compositions les contenant, procede de frabrication et utilisation |
WO2008051887A1 (en) * | 2006-10-23 | 2008-05-02 | Lexicon Pharmaceuticals, Inc. | Process for preparing 5-alkyl-7h-pyrrolo[2,3-d]pyrimidine-2-ols |
TW201111385A (en) | 2009-08-27 | 2011-04-01 | Biocryst Pharm Inc | Heterocyclic compounds as janus kinase inhibitors |
US20120244141A1 (en) | 2010-09-28 | 2012-09-27 | Boehringer Ingelheim International Gmbh | Stratification of cancer patients for susceptibility to therapy with PTK2 inhibitors |
TW202021967A (zh) * | 2018-08-14 | 2020-06-16 | 大陸商江蘇豪森藥業集團有限公司 | 凋亡信號調節激酶1抑制劑的鹽及其晶型 |
US11034669B2 (en) | 2018-11-30 | 2021-06-15 | Nuvation Bio Inc. | Pyrrole and pyrazole compounds and methods of use thereof |
Family Cites Families (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB0107901D0 (en) * | 2001-03-29 | 2001-05-23 | Cyclacel Ltd | Anti-cancer compounds |
ES2307780T3 (es) * | 2001-09-21 | 2008-12-01 | Smithkline Beecham Corporation | Compuestos quimicos. |
JP2006515828A (ja) | 2001-09-27 | 2006-06-08 | スミスクライン・ビーチャム・コーポレイション | 化学化合物 |
US20040138269A1 (en) * | 2002-10-11 | 2004-07-15 | Sugen, Inc. | Substituted pyrroles as kinase inhibitors |
GB0229581D0 (en) * | 2002-12-19 | 2003-01-22 | Cyclacel Ltd | Use |
JP4808154B2 (ja) * | 2003-03-13 | 2011-11-02 | バーテックス ファーマシューティカルズ インコーポレイテッド | プロテインキナーゼインヒビターとして有用な組成物 |
DE10354060A1 (de) * | 2003-11-19 | 2005-06-02 | Merck Patent Gmbh | Pyrrolderivate |
US7183285B2 (en) * | 2004-04-29 | 2007-02-27 | Pharmix Corp. | Compositions and treatments for inhibiting kinase and/or HMG-CoA reductase |
FR2881426B1 (fr) | 2005-02-03 | 2007-03-30 | Aventis Pharma Sa | Pyrolles et imidazoles substitues, compositions les contenant, procede de frabrication et utilisation |
-
2005
- 2005-02-10 FR FR0501354A patent/FR2881742B1/fr not_active Expired - Fee Related
-
2006
- 2006-02-02 PA PA20068661601A patent/PA8661601A1/es unknown
- 2006-02-02 PE PE2006000135A patent/PE20061086A1/es not_active Application Discontinuation
- 2006-02-02 DO DO2006000028A patent/DOP2006000028A/es unknown
- 2006-02-03 MY MYPI20060441A patent/MY142082A/en unknown
- 2006-02-08 CA CA002596822A patent/CA2596822A1/fr not_active Abandoned
- 2006-02-08 PL PL06709274T patent/PL1851198T3/pl unknown
- 2006-02-08 WO PCT/FR2006/000286 patent/WO2006084996A1/fr active Application Filing
- 2006-02-08 AR ARP060100452A patent/AR052571A1/es unknown
- 2006-02-08 AT AT06709274T patent/ATE419234T1/de active
- 2006-02-08 ES ES06709274T patent/ES2319926T3/es active Active
- 2006-02-08 DE DE602006004566T patent/DE602006004566D1/de active Active
- 2006-02-08 PT PT06709274T patent/PT1851198E/pt unknown
- 2006-02-08 DK DK06709274T patent/DK1851198T3/da active
- 2006-02-08 SI SI200630232T patent/SI1851198T1/sl unknown
- 2006-02-08 RS RSP-2009/0128A patent/RS50806B/sr unknown
- 2006-02-08 ZA ZA200706157A patent/ZA200706157B/xx unknown
- 2006-02-08 EA EA200701688A patent/EA013060B1/ru not_active IP Right Cessation
- 2006-02-08 BR BRPI0606955-0A patent/BRPI0606955A2/pt not_active IP Right Cessation
- 2006-02-08 MX MX2007008789A patent/MX2007008789A/es active IP Right Grant
- 2006-02-08 JP JP2007554598A patent/JP2008530061A/ja active Pending
- 2006-02-08 GT GT200600048A patent/GT200600048A/es unknown
- 2006-02-08 KR KR1020077018321A patent/KR20070101317A/ko not_active Application Discontinuation
- 2006-02-08 AU AU2006212106A patent/AU2006212106A1/en not_active Withdrawn
- 2006-02-08 CN CNA2006800044573A patent/CN101115716A/zh active Pending
- 2006-02-08 EP EP06709274A patent/EP1851198B1/fr active Active
- 2006-02-09 TW TW095104288A patent/TW200640858A/zh unknown
- 2006-02-10 UY UY29371A patent/UY29371A1/es unknown
-
2007
- 2007-06-26 TN TNP2007000241A patent/TNSN07241A1/fr unknown
- 2007-07-06 CR CR9231A patent/CR9231A/es not_active Application Discontinuation
- 2007-07-08 IL IL184488A patent/IL184488A0/en unknown
- 2007-08-01 US US11/832,208 patent/US7592365B2/en not_active Expired - Fee Related
- 2007-08-13 MA MA30134A patent/MA29248B1/fr unknown
- 2007-09-06 NO NO20074528A patent/NO20074528L/no not_active Application Discontinuation
-
2009
- 2009-03-17 HR HR20090158T patent/HRP20090158T1/xx unknown
- 2009-03-23 CY CY20091100344T patent/CY1108916T1/el unknown
Also Published As
Similar Documents
Publication | Publication Date | Title |
---|---|---|
UY29341A1 (es) | Pirazolo piridinas sustituidas, composiciones que las contienen, procedimiento de fabricación | |
CR9463A (es) | Pirrolinas sustituidas, composiciones que las contienen, proceso de fabricacion y utilizacion | |
UY29361A1 (es) | Pirroles e imidazoles sustituídos, composiciones que los contienen, procedimiento de fabricación y utilización | |
UY29248A1 (es) | Indoles sustituidos, composiciones que los contienen, procedimiento de fabricación y utilización | |
HN2008000188A (es) | 7- aza- indazoles sustituidos, composiciones que los contienen, procedimiento de fabricacion y su utilizacion | |
CR10247A (es) | Dimeros de derivados de artemisinina, su preparacion y su aplicacion en terapeutica | |
UY29236A1 (es) | 2-alcoxi-3,4,5-trihidroxi-alquilamidas. su preparación, composiciones que las contienen y su utilización. | |
DOP2006000015A (es) | Pirazolo piridinas sustituidas, composiciones que las contienen, procedimiento de fabricación | |
ECSP088252A (es) | 7-aza-indazoles sustituidos, composiciones que los contienen, procedimiento de fabricación y utilización | |
NI200900078A (es) | Pirazoles sustituidos, composiciones que los contienen, procedimiento de fabricación y utilización. | |
CR9231A (es) | Pirroles sustituidos, composiciones que los contienen, procesos de fabricacion y utilizacion | |
CR9115A (es) | Indoles sustituidos, composiciones que los contienen, procedimiento de fabricacion y utilizacion | |
ECSP088893A (es) | 2-alcoxi-3, 4,5-trihidroxi-alquilamida-benzazepinas, su preparación, composiciones que las contienen y utilización | |
ECSP088899A (es) | Derivados de 2-alcoxi-3,4,5-trihidroxi-alquilamida, su preparación, composiciones que las contienen y utilización | |
DOP2005000246A (es) | Indoles sustituidos, composiciones que los contienen, procedimiento de fabricacion y utilizacion | |
CR10428A (es) | 2-alcoxi-3,4,5-trihidroxi-alquilamida-benzotiazepinas, su preparacion, composiciones que las contienen y utilizacion | |
UY29235A1 (es) | Bengamidas que poseen un ciclo caprolactama sustituido, procedimiento de preparación, composiciones que las contienen y utilización | |
UY29501A1 (es) | Pirrolopiridinas sustituidas, composiciones que las contienen, proceso de fabricación y utilización |