DOP2006000028A - Pirroles sustituidos, composiciones que los contienen, proceso de fabricación y utilización - Google Patents

Pirroles sustituidos, composiciones que los contienen, proceso de fabricación y utilización

Info

Publication number
DOP2006000028A
DOP2006000028A DO2006000028A DO2006000028A DOP2006000028A DO P2006000028 A DOP2006000028 A DO P2006000028A DO 2006000028 A DO2006000028 A DO 2006000028A DO 2006000028 A DO2006000028 A DO 2006000028A DO P2006000028 A DOP2006000028 A DO P2006000028A
Authority
DO
Dominican Republic
Prior art keywords
compositions
manufacturing
pirroles
replaced
contain
Prior art date
Application number
DO2006000028A
Other languages
English (en)
Inventor
Michel Tabart
Eric Bacque
Baptiste Ronan
Pascal Desmazeau
Fabrice Viviani
Catherine Souaille
Jean-Philippe Letallec
Original Assignee
Aventis Pharma Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=35478244&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DOP2006000028(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Aventis Pharma Sa filed Critical Aventis Pharma Sa
Publication of DOP2006000028A publication Critical patent/DOP2006000028A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D207/00Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/30Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
    • C07D207/34Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pyrrole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

Pirroles sustituidos, composiciones que los contienen, proceso de fabricación y utilización. La presente invención se refiere particularmente a la preparación de pirroles sustituidos, a las composiciones que los contienen, a su proceso de preparación, y a su utilización como medicamento, en particular como agentes anticancerígenos.
DO2006000028A 2005-02-10 2006-02-02 Pirroles sustituidos, composiciones que los contienen, proceso de fabricación y utilización DOP2006000028A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR0501354A FR2881742B1 (fr) 2005-02-10 2005-02-10 Pyrroles substitues, compositions les contenant, procede de fabrication et utilisation

Publications (1)

Publication Number Publication Date
DOP2006000028A true DOP2006000028A (es) 2006-09-15

Family

ID=35478244

Family Applications (1)

Application Number Title Priority Date Filing Date
DO2006000028A DOP2006000028A (es) 2005-02-10 2006-02-02 Pirroles sustituidos, composiciones que los contienen, proceso de fabricación y utilización

Country Status (36)

Country Link
US (1) US7592365B2 (es)
EP (1) EP1851198B1 (es)
JP (1) JP2008530061A (es)
KR (1) KR20070101317A (es)
CN (1) CN101115716A (es)
AR (1) AR052571A1 (es)
AT (1) ATE419234T1 (es)
AU (1) AU2006212106A1 (es)
BR (1) BRPI0606955A2 (es)
CA (1) CA2596822A1 (es)
CR (1) CR9231A (es)
CY (1) CY1108916T1 (es)
DE (1) DE602006004566D1 (es)
DK (1) DK1851198T3 (es)
DO (1) DOP2006000028A (es)
EA (1) EA013060B1 (es)
ES (1) ES2319926T3 (es)
FR (1) FR2881742B1 (es)
GT (1) GT200600048A (es)
HR (1) HRP20090158T1 (es)
IL (1) IL184488A0 (es)
MA (1) MA29248B1 (es)
MX (1) MX2007008789A (es)
MY (1) MY142082A (es)
NO (1) NO20074528L (es)
PA (1) PA8661601A1 (es)
PE (1) PE20061086A1 (es)
PL (1) PL1851198T3 (es)
PT (1) PT1851198E (es)
RS (1) RS50806B (es)
SI (1) SI1851198T1 (es)
TN (1) TNSN07241A1 (es)
TW (1) TW200640858A (es)
UY (1) UY29371A1 (es)
WO (1) WO2006084996A1 (es)
ZA (1) ZA200706157B (es)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2881426B1 (fr) 2005-02-03 2007-03-30 Aventis Pharma Sa Pyrolles et imidazoles substitues, compositions les contenant, procede de frabrication et utilisation
WO2008051887A1 (en) * 2006-10-23 2008-05-02 Lexicon Pharmaceuticals, Inc. Process for preparing 5-alkyl-7h-pyrrolo[2,3-d]pyrimidine-2-ols
TW201111385A (en) 2009-08-27 2011-04-01 Biocryst Pharm Inc Heterocyclic compounds as janus kinase inhibitors
US20120244141A1 (en) 2010-09-28 2012-09-27 Boehringer Ingelheim International Gmbh Stratification of cancer patients for susceptibility to therapy with PTK2 inhibitors
TW202021967A (zh) * 2018-08-14 2020-06-16 大陸商江蘇豪森藥業集團有限公司 凋亡信號調節激酶1抑制劑的鹽及其晶型
US11034669B2 (en) 2018-11-30 2021-06-15 Nuvation Bio Inc. Pyrrole and pyrazole compounds and methods of use thereof

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0107901D0 (en) * 2001-03-29 2001-05-23 Cyclacel Ltd Anti-cancer compounds
ES2307780T3 (es) * 2001-09-21 2008-12-01 Smithkline Beecham Corporation Compuestos quimicos.
JP2006515828A (ja) 2001-09-27 2006-06-08 スミスクライン・ビーチャム・コーポレイション 化学化合物
US20040138269A1 (en) * 2002-10-11 2004-07-15 Sugen, Inc. Substituted pyrroles as kinase inhibitors
GB0229581D0 (en) * 2002-12-19 2003-01-22 Cyclacel Ltd Use
JP4808154B2 (ja) * 2003-03-13 2011-11-02 バーテックス ファーマシューティカルズ インコーポレイテッド プロテインキナーゼインヒビターとして有用な組成物
DE10354060A1 (de) * 2003-11-19 2005-06-02 Merck Patent Gmbh Pyrrolderivate
US7183285B2 (en) * 2004-04-29 2007-02-27 Pharmix Corp. Compositions and treatments for inhibiting kinase and/or HMG-CoA reductase
FR2881426B1 (fr) 2005-02-03 2007-03-30 Aventis Pharma Sa Pyrolles et imidazoles substitues, compositions les contenant, procede de frabrication et utilisation

Also Published As

Publication number Publication date
SI1851198T1 (sl) 2009-06-30
CA2596822A1 (fr) 2006-08-17
IL184488A0 (en) 2007-10-31
PL1851198T3 (pl) 2009-06-30
BRPI0606955A2 (pt) 2009-07-28
US7592365B2 (en) 2009-09-22
WO2006084996A1 (fr) 2006-08-17
JP2008530061A (ja) 2008-08-07
TW200640858A (en) 2006-12-01
EA200701688A1 (ru) 2007-12-28
NO20074528L (no) 2007-10-31
RS50806B (sr) 2010-08-31
CY1108916T1 (el) 2014-07-02
ES2319926T3 (es) 2009-05-14
TNSN07241A1 (en) 2008-11-21
ATE419234T1 (de) 2009-01-15
DK1851198T3 (da) 2009-05-04
MX2007008789A (es) 2007-09-11
EP1851198B1 (fr) 2008-12-31
MY142082A (en) 2010-08-30
ZA200706157B (en) 2008-11-26
AR052571A1 (es) 2007-03-21
PA8661601A1 (es) 2006-09-08
US20080167368A1 (en) 2008-07-10
AU2006212106A1 (en) 2006-08-17
EA013060B1 (ru) 2010-02-26
CN101115716A (zh) 2008-01-30
UY29371A1 (es) 2006-10-02
FR2881742A1 (fr) 2006-08-11
EP1851198A1 (fr) 2007-11-07
KR20070101317A (ko) 2007-10-16
MA29248B1 (fr) 2008-02-01
GT200600048A (es) 2006-07-03
PT1851198E (pt) 2009-03-26
FR2881742B1 (fr) 2007-09-07
HRP20090158T1 (en) 2009-05-31
DE602006004566D1 (de) 2009-02-12
CR9231A (es) 2007-10-23
PE20061086A1 (es) 2006-11-30

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