CR9115A - Indoles sustituidos, composiciones que los contienen, procedimiento de fabricacion y utilizacion - Google Patents
Indoles sustituidos, composiciones que los contienen, procedimiento de fabricacion y utilizacionInfo
- Publication number
- CR9115A CR9115A CR9115A CR9115A CR9115A CR 9115 A CR9115 A CR 9115A CR 9115 A CR9115 A CR 9115A CR 9115 A CR9115 A CR 9115A CR 9115 A CR9115 A CR 9115A
- Authority
- CR
- Costa Rica
- Prior art keywords
- indoles
- compositions
- replaced
- contain
- manufacturing
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
- C07D209/42—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
- A61K31/404—Indoles, e.g. pindolol
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B55/00—Racemisation; Complete or partial inversion
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/07—Optical isomers
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/09—Geometrical isomers
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Indole Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Abstract
La presente invencion se refiere particularmente a la preparacion de indoles sustituidos, a las composiciones que los contienen, a su procedimiento de preparacion, y a su utilizacion como medicamento, en particular como agentes anticancerigenos. Formula (I).
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR0412966A FR2878849B1 (fr) | 2004-12-06 | 2004-12-06 | Indoles substitues, compositions les contenant, procede de fabrication et utilisation |
US65046505P | 2005-02-07 | 2005-02-07 |
Publications (1)
Publication Number | Publication Date |
---|---|
CR9115A true CR9115A (es) | 2007-10-23 |
Family
ID=38792212
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CR9115A CR9115A (es) | 2004-12-06 | 2007-05-09 | Indoles sustituidos, composiciones que los contienen, procedimiento de fabricacion y utilizacion |
Country Status (9)
Country | Link |
---|---|
JP (1) | JP2008532926A (es) |
KR (1) | KR20070100277A (es) |
BR (1) | BRPI0515811A (es) |
CR (1) | CR9115A (es) |
EA (1) | EA012613B1 (es) |
IL (1) | IL183438A0 (es) |
MA (1) | MA29026B1 (es) |
MX (1) | MX2007006764A (es) |
NO (1) | NO20073015L (es) |
Families Citing this family (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE102005037499A1 (de) * | 2005-08-09 | 2007-02-15 | Merck Patent Gmbh | Pyrazolderivate |
JP7323218B2 (ja) * | 2019-02-18 | 2023-08-08 | 深▲チェン▼市塔吉瑞生物医薬有限公司 | 置換された縮合芳香環誘導体、その組成物、およびそれらの使用 |
Family Cites Families (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
KR19990022369A (ko) * | 1995-06-07 | 1999-03-25 | 스테판 이반스-프레크 | 어뎁터 단백질/티로신 카이나제 상호작용을 방해하는 조성물과그 방법 |
US6376529B1 (en) * | 1995-06-07 | 2002-04-23 | Peng Cho Tang | Mono- and bis-indolylquinones and prophylactic and therapeutic uses thereof |
JP4623962B2 (ja) * | 2001-10-22 | 2011-02-02 | ザ・リサーチ・ファウンデーション・オブ・ステイト・ユニバーシティ・オブ・ニューヨーク | タンパク質キナーゼおよびホスファターゼ阻害剤、それらを設計する方法、ならびにそれらを使用する方法 |
DK1539742T3 (da) * | 2002-06-24 | 2006-12-27 | Schering Corp | Indolderivater, der er nyttige som histamin H3-antagonister |
FR2842526B1 (fr) * | 2002-07-16 | 2007-07-13 | Aventis Pharma Sa | Compositions pharmaceutiques contenant un derive de 3-guanidinocarbonyl-1-heteroaryl-indole, procede de preparation a titre de medicaments |
JP2004149429A (ja) * | 2002-10-29 | 2004-05-27 | Takeda Chem Ind Ltd | インドール化合物およびその用途 |
-
2005
- 2005-12-02 JP JP2007543884A patent/JP2008532926A/ja active Pending
- 2005-12-02 BR BRPI0515811-7A patent/BRPI0515811A/pt not_active IP Right Cessation
- 2005-12-02 EA EA200701227A patent/EA012613B1/ru not_active IP Right Cessation
- 2005-12-02 KR KR1020077015482A patent/KR20070100277A/ko not_active Application Discontinuation
- 2005-12-02 MX MX2007006764A patent/MX2007006764A/es unknown
-
2007
- 2007-05-09 CR CR9115A patent/CR9115A/es unknown
- 2007-05-17 MA MA29913A patent/MA29026B1/fr unknown
- 2007-05-27 IL IL183438A patent/IL183438A0/en unknown
- 2007-06-13 NO NO20073015A patent/NO20073015L/no not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
BRPI0515811A (pt) | 2008-08-05 |
JP2008532926A (ja) | 2008-08-21 |
MX2007006764A (es) | 2007-08-15 |
NO20073015L (no) | 2007-08-28 |
EA012613B1 (ru) | 2009-10-30 |
MA29026B1 (fr) | 2007-11-01 |
EA200701227A1 (ru) | 2007-10-26 |
KR20070100277A (ko) | 2007-10-10 |
IL183438A0 (en) | 2007-09-20 |
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