DK96983D0 - Fremgangsmade til fremstilling af 9-dihydro-11,12-ketalderivater af erythromycin a eller epi-erythromycin a - Google Patents

Fremgangsmade til fremstilling af 9-dihydro-11,12-ketalderivater af erythromycin a eller epi-erythromycin a

Info

Publication number
DK96983D0
DK96983D0 DK0969/83A DK96983A DK96983D0 DK 96983 D0 DK96983 D0 DK 96983D0 DK 0969/83 A DK0969/83 A DK 0969/83A DK 96983 A DK96983 A DK 96983A DK 96983 D0 DK96983 D0 DK 96983D0
Authority
DK
Denmark
Prior art keywords
erythromycine
epi
dihydro
preparing
ketal derivatives
Prior art date
Application number
DK0969/83A
Other languages
English (en)
Other versions
DK96983A (da
DK159853C (da
DK159853B (da
Inventor
James Robert Hauske
Frank Christian Sciavolino
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of DK96983D0 publication Critical patent/DK96983D0/da
Publication of DK96983A publication Critical patent/DK96983A/da
Publication of DK159853B publication Critical patent/DK159853B/da
Application granted granted Critical
Publication of DK159853C publication Critical patent/DK159853C/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DK096983A 1982-03-01 1983-02-28 Analogifremgangsmaade til fremstilling af 9-dihydro-11,12-o-isopropyliden-erythromycin a eller -4ae-epi-erythromycin a eller 2'-o-acylater deraf eller farmaceutisk acceptable syreadditionssalte deraf DK159853C (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US35354882 1982-03-01
US06/353,548 US4382086A (en) 1982-03-01 1982-03-01 9-Dihydro-11,12-ketal derivatives of erythromycin A and epi-erythromycin A

Publications (4)

Publication Number Publication Date
DK96983D0 true DK96983D0 (da) 1983-02-28
DK96983A DK96983A (da) 1983-09-02
DK159853B DK159853B (da) 1990-12-17
DK159853C DK159853C (da) 1991-05-13

Family

ID=23389607

Family Applications (1)

Application Number Title Priority Date Filing Date
DK096983A DK159853C (da) 1982-03-01 1983-02-28 Analogifremgangsmaade til fremstilling af 9-dihydro-11,12-o-isopropyliden-erythromycin a eller -4ae-epi-erythromycin a eller 2'-o-acylater deraf eller farmaceutisk acceptable syreadditionssalte deraf

Country Status (8)

Country Link
US (1) US4382086A (da)
EP (1) EP0087916B1 (da)
JP (1) JPS58159500A (da)
DE (1) DE3361453D1 (da)
DK (1) DK159853C (da)
GR (1) GR77921B (da)
IE (1) IE54431B1 (da)
YU (1) YU42841B (da)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8421429D0 (en) * 1984-08-23 1984-09-26 Beecham Group Plc Chemical compounds
EP0184921A3 (en) * 1984-12-08 1986-10-29 Beecham Group Plc Erythromycin derivatives
DK109886A (da) 1985-03-12 1986-09-13 Beecham Group Plc Erythromycinderivater
US4681872A (en) * 1985-11-12 1987-07-21 Abbott Laboratories Erythromycin A 11,12-carbonate and method of use
US4640910A (en) * 1985-11-12 1987-02-03 Abbott Laboratories Erythromycin A silylated compounds and method of use
CA2094060A1 (en) * 1990-10-15 1992-04-16 Toshifumi Asaka 2'-position modified compound of erythromycin or its derivative
WO2003070254A1 (en) * 2002-02-15 2003-08-28 Sympore Gmbh Antibiotic conjugates
US20040005641A1 (en) * 2002-02-15 2004-01-08 Michael Burnet Conjugates of biologically active compounds, methods for their preparation and use, formulation and pharmaceutical applications thereof
US7579324B2 (en) 2002-02-15 2009-08-25 C-A-I-R Biosciences Gmbh Conjugates of biologically active compounds, methods for their preparation and use, formulation and pharmaceutical applications thereof
JP4796300B2 (ja) * 2002-08-29 2011-10-19 ファイザー インコーポレイテッド モチライド化合物
US7211568B2 (en) * 2003-12-18 2007-05-01 Kosan Biosciences Incorporated 9-Desoxoerythromycin compounds as prokinetic agents
CN101228171A (zh) * 2005-07-26 2008-07-23 默克勒有限公司 作为5-脂氧化酶和环加氧酶抑制剂的吡咯里嗪和中氮茚化合物的大环内酯偶联物

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2653899A (en) * 1952-04-14 1953-09-29 Lilly Co Eli Erythromycin, its salts, and method of preparation
US3417077A (en) * 1966-05-16 1968-12-17 Lilly Co Eli Erythromycin derivative and process for the preparation thereof
US3884903A (en) * 1973-06-21 1975-05-20 Abbott Lab 4{41 -Deoxy-4{41 -oxoerythromycin B derivatives
US3884904A (en) * 1973-06-21 1975-05-20 Abbott Lab 11-Substituted erythromycin B derivatives
US4150220A (en) * 1977-02-04 1979-04-17 Pfizer Inc. Semi-synthetic 4"-erythromycin A derivatives

Also Published As

Publication number Publication date
DE3361453D1 (en) 1986-01-23
JPS58159500A (ja) 1983-09-21
US4382086A (en) 1983-05-03
EP0087916A1 (en) 1983-09-07
DK96983A (da) 1983-09-02
JPH0142275B2 (da) 1989-09-11
EP0087916B1 (en) 1985-12-11
YU45983A (en) 1986-02-28
YU42841B (en) 1988-12-31
IE830410L (en) 1983-09-01
GR77921B (da) 1984-09-25
IE54431B1 (en) 1989-10-11
DK159853C (da) 1991-05-13
DK159853B (da) 1990-12-17

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