DK96983A - Fremgangsmaade til fremstilling af 9-dihydro-11,12-ketalderivater af erythromycin a eller epi-erythromycin a - Google Patents
Fremgangsmaade til fremstilling af 9-dihydro-11,12-ketalderivater af erythromycin a eller epi-erythromycin a Download PDFInfo
- Publication number
- DK96983A DK96983A DK96983A DK96983A DK96983A DK 96983 A DK96983 A DK 96983A DK 96983 A DK96983 A DK 96983A DK 96983 A DK96983 A DK 96983A DK 96983 A DK96983 A DK 96983A
- Authority
- DK
- Denmark
- Prior art keywords
- erythromycine
- epi
- dihydro
- preparing
- ketal derivatives
- Prior art date
Links
- ULGZDMOVFRHVEP-RWJQBGPGSA-N Erythromycin Chemical class O([C@@H]1[C@@H](C)C(=O)O[C@@H]([C@@]([C@H](O)[C@@H](C)C(=O)[C@H](C)C[C@@](C)(O)[C@H](O[C@H]2[C@@H]([C@H](C[C@@H](C)O2)N(C)C)O)[C@H]1C)(C)O)CC)[C@H]1C[C@@](C)(OC)[C@@H](O)[C@H](C)O1 ULGZDMOVFRHVEP-RWJQBGPGSA-N 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
- C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Engineering & Computer Science (AREA)
- Biochemistry (AREA)
- Molecular Biology (AREA)
- Genetics & Genomics (AREA)
- Biotechnology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- Oncology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Communicable Diseases (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US35354882 | 1982-03-01 | ||
| US06/353,548 US4382086A (en) | 1982-03-01 | 1982-03-01 | 9-Dihydro-11,12-ketal derivatives of erythromycin A and epi-erythromycin A |
Publications (4)
| Publication Number | Publication Date |
|---|---|
| DK96983D0 DK96983D0 (da) | 1983-02-28 |
| DK96983A true DK96983A (da) | 1983-09-02 |
| DK159853B DK159853B (da) | 1990-12-17 |
| DK159853C DK159853C (da) | 1991-05-13 |
Family
ID=23389607
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK096983A DK159853C (da) | 1982-03-01 | 1983-02-28 | Analogifremgangsmaade til fremstilling af 9-dihydro-11,12-o-isopropyliden-erythromycin a eller -4ae-epi-erythromycin a eller 2'-o-acylater deraf eller farmaceutisk acceptable syreadditionssalte deraf |
Country Status (8)
| Country | Link |
|---|---|
| US (1) | US4382086A (da) |
| EP (1) | EP0087916B1 (da) |
| JP (1) | JPS58159500A (da) |
| DE (1) | DE3361453D1 (da) |
| DK (1) | DK159853C (da) |
| GR (1) | GR77921B (da) |
| IE (1) | IE54431B1 (da) |
| YU (1) | YU42841B (da) |
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB8421429D0 (en) * | 1984-08-23 | 1984-09-26 | Beecham Group Plc | Chemical compounds |
| EP0184921A3 (en) * | 1984-12-08 | 1986-10-29 | Beecham Group Plc | Erythromycin derivatives |
| EP0201166B1 (en) | 1985-03-12 | 1990-02-07 | Beecham Group Plc | Erythromycin derivatives |
| US4640910A (en) * | 1985-11-12 | 1987-02-03 | Abbott Laboratories | Erythromycin A silylated compounds and method of use |
| US4681872A (en) * | 1985-11-12 | 1987-07-21 | Abbott Laboratories | Erythromycin A 11,12-carbonate and method of use |
| US5350839A (en) * | 1990-10-15 | 1994-09-27 | Taisho Pharmaceutical Co., Ltd. | 2'-position modified compound of erythromycin or its derivative |
| NZ535354A (en) | 2002-02-15 | 2008-01-31 | Merckle Gmbh | Conjugates of biologically active compounds, methods for their preparation and use, formulation and pharmaceutical applications thereof |
| EP1483579A4 (en) | 2002-02-15 | 2006-07-12 | Merckle Gmbh | CONJUGATES OF BIOLOGICALLY ACTIVE COMPOUNDS, METHODS FOR THE PREPARATION AND USE OF CONJUGATES, FORMULATION AND PHARMACEUTICAL APPLICATIONS OBTAINED FROM SUCH CONJUGATES |
| EP1482957A4 (en) * | 2002-02-15 | 2006-07-19 | Merckle Gmbh | ANTIBIOTIC CONJUGATES |
| CN100363359C (zh) * | 2002-08-29 | 2008-01-23 | 菲塞股份有限公司 | 运动内酯化合物 |
| US7211568B2 (en) * | 2003-12-18 | 2007-05-01 | Kosan Biosciences Incorporated | 9-Desoxoerythromycin compounds as prokinetic agents |
| WO2007012464A1 (en) * | 2005-07-26 | 2007-02-01 | Merckle Gmbh | Macrolide conjugates of pyrrolizine and indolizine compounds as inhibitors of 5-lipooxygenase and cyclooxygenase |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US2653899A (en) * | 1952-04-14 | 1953-09-29 | Lilly Co Eli | Erythromycin, its salts, and method of preparation |
| US3417077A (en) * | 1966-05-16 | 1968-12-17 | Lilly Co Eli | Erythromycin derivative and process for the preparation thereof |
| US3884904A (en) * | 1973-06-21 | 1975-05-20 | Abbott Lab | 11-Substituted erythromycin B derivatives |
| US3884903A (en) * | 1973-06-21 | 1975-05-20 | Abbott Lab | 4{41 -Deoxy-4{41 -oxoerythromycin B derivatives |
| US4150220A (en) * | 1977-02-04 | 1979-04-17 | Pfizer Inc. | Semi-synthetic 4"-erythromycin A derivatives |
-
1982
- 1982-03-01 US US06/353,548 patent/US4382086A/en not_active Expired - Lifetime
-
1983
- 1983-02-23 DE DE8383300937T patent/DE3361453D1/de not_active Expired
- 1983-02-23 EP EP83300937A patent/EP0087916B1/en not_active Expired
- 1983-02-23 GR GR70583A patent/GR77921B/el unknown
- 1983-02-25 YU YU459/83A patent/YU42841B/xx unknown
- 1983-02-28 IE IE410/83A patent/IE54431B1/en not_active IP Right Cessation
- 1983-02-28 DK DK096983A patent/DK159853C/da not_active IP Right Cessation
- 1983-03-01 JP JP58033682A patent/JPS58159500A/ja active Granted
Also Published As
| Publication number | Publication date |
|---|---|
| DK159853C (da) | 1991-05-13 |
| EP0087916A1 (en) | 1983-09-07 |
| YU45983A (en) | 1986-02-28 |
| DE3361453D1 (en) | 1986-01-23 |
| JPS58159500A (ja) | 1983-09-21 |
| DK159853B (da) | 1990-12-17 |
| GR77921B (da) | 1984-09-25 |
| YU42841B (en) | 1988-12-31 |
| IE54431B1 (en) | 1989-10-11 |
| JPH0142275B2 (da) | 1989-09-11 |
| US4382086A (en) | 1983-05-03 |
| IE830410L (en) | 1983-09-01 |
| DK96983D0 (da) | 1983-02-28 |
| EP0087916B1 (en) | 1985-12-11 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PUP | Patent expired |