DK93986A - Substituerede benzimidazolderivater, fremgangsmaader til fremstillingheraf, mellemprodukter, der er anvendelige ved deres fremstilling samt farmaceutiske midler indeholdende dem - Google Patents

Substituerede benzimidazolderivater, fremgangsmaader til fremstillingheraf, mellemprodukter, der er anvendelige ved deres fremstilling samt farmaceutiske midler indeholdende dem Download PDF

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Publication number
DK93986A
DK93986A DK93986A DK93986A DK93986A DK 93986 A DK93986 A DK 93986A DK 93986 A DK93986 A DK 93986A DK 93986 A DK93986 A DK 93986A DK 93986 A DK93986 A DK 93986A
Authority
DK
Denmark
Prior art keywords
intermediates
substituted
applicable
preparation
pharmaceutical agents
Prior art date
Application number
DK93986A
Other languages
Danish (da)
English (en)
Other versions
DK93986D0 (da
Inventor
Robert John Ife
Thomas Henry Brown
Original Assignee
Smith Kline French Lab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB858505615A external-priority patent/GB8505615D0/en
Priority claimed from GB858531605A external-priority patent/GB8531605D0/en
Application filed by Smith Kline French Lab filed Critical Smith Kline French Lab
Publication of DK93986D0 publication Critical patent/DK93986D0/da
Publication of DK93986A publication Critical patent/DK93986A/da

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/32One oxygen, sulfur or nitrogen atom
    • C07D239/42One nitrogen atom
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D491/00Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
DK93986A 1985-03-05 1986-02-28 Substituerede benzimidazolderivater, fremgangsmaader til fremstillingheraf, mellemprodukter, der er anvendelige ved deres fremstilling samt farmaceutiske midler indeholdende dem DK93986A (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB858505615A GB8505615D0 (en) 1985-03-05 1985-03-05 Heterocyclic compounds
GB858531605A GB8531605D0 (en) 1985-12-23 1985-12-23 Heterocyclic compounds

Publications (2)

Publication Number Publication Date
DK93986D0 DK93986D0 (da) 1986-02-28
DK93986A true DK93986A (da) 1986-09-06

Family

ID=26288907

Family Applications (2)

Application Number Title Priority Date Filing Date
DK8600939D DK8600939A (no) 1985-03-05
DK93986A DK93986A (da) 1985-03-05 1986-02-28 Substituerede benzimidazolderivater, fremgangsmaader til fremstillingheraf, mellemprodukter, der er anvendelige ved deres fremstilling samt farmaceutiske midler indeholdende dem

Family Applications Before (1)

Application Number Title Priority Date Filing Date
DK8600939D DK8600939A (no) 1985-03-05

Country Status (16)

Country Link
US (2) US4777172A (no)
EP (1) EP0198583A1 (no)
CN (1) CN86102398A (no)
AU (1) AU578141B2 (no)
DK (2) DK93986A (no)
ES (1) ES8707949A1 (no)
FI (1) FI860909A (no)
GR (1) GR860596B (no)
HU (1) HU195962B (no)
IL (1) IL78026A (no)
JO (1) JO1443B1 (no)
NO (1) NO860830L (no)
NZ (1) NZ215362A (no)
PH (2) PH23115A (no)
PT (1) PT82135B (no)
ZW (1) ZW4786A1 (no)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0174717B1 (en) * 1984-07-06 1992-01-22 FISONS plc Benzimidazoles, and their production formulation and use as gastric acid secretion inhibitors
DE3723327A1 (de) * 1987-07-15 1989-02-02 Hoechst Ag Substituierte thienoimidazol-derivate, verfahren zu ihrer herstellung, sie enthaltende pharmazeutische zubereitungen und ihre verwendung als magensaeuresekretionshemmer, magenschutzmittel sowie als medikament gegen intestinale entzuendungen
DE4025387A1 (de) * 1990-08-10 1992-02-13 Hoechst Ag Substituierte pyrimidin-derivate, verfahren zu ihrer herstellung und ihre verwendung als reagenzien
US6780880B1 (en) 1999-08-26 2004-08-24 Robert R. Whittle FT-Raman spectroscopic measurement
US6316020B1 (en) 1999-08-26 2001-11-13 Robert R. Whittle Pharmaceutical formulations
US6262086B1 (en) 1999-08-26 2001-07-17 Robert R. Whittle Pharmaceutical unit dosage form
US6262085B1 (en) 1999-08-26 2001-07-17 Robert R. Whittle Alkoxy substituted Benzimidazole compounds, pharmaceutical preparations containing the same, and methods of using the same
US6312712B1 (en) 1999-08-26 2001-11-06 Robert R. Whittle Method of improving bioavailability
US6312723B1 (en) 1999-08-26 2001-11-06 Robert R. Whittle Pharmaceutical unit dosage form
US6326384B1 (en) 1999-08-26 2001-12-04 Robert R. Whittle Dry blend pharmaceutical unit dosage form
US6268385B1 (en) 1999-08-26 2001-07-31 Robert R. Whittle Dry blend pharmaceutical formulations
US6369087B1 (en) 1999-08-26 2002-04-09 Robert R. Whittle Alkoxy substituted benzimidazole compounds, pharmaceutical preparations containing the same, and methods of using the same

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE416649B (sv) * 1974-05-16 1981-01-26 Haessle Ab Forfarande for framstellning av foreningar som paverkar magsyrasekretionen
US4359465A (en) * 1980-07-28 1982-11-16 The Upjohn Company Methods for treating gastrointestinal inflammation
EP0174717B1 (en) * 1984-07-06 1992-01-22 FISONS plc Benzimidazoles, and their production formulation and use as gastric acid secretion inhibitors
EP0178438A1 (en) * 1984-09-19 1986-04-23 Beecham Group Plc Novel compounds
FR2593178B1 (fr) * 1986-01-20 1988-04-29 Esteve Labor Dr Derives de 2-benzimidazolylalkylthio (ou sulfinyle ou sulfonyle) leur preparation et leur application en tant que medicaments.

Also Published As

Publication number Publication date
DK8600939A (no) 1986-09-06
AU5412986A (en) 1986-09-11
HUT40111A (en) 1986-11-28
HU195962B (en) 1988-08-29
PH23115A (en) 1989-04-19
CN86102398A (zh) 1986-11-12
US4777172A (en) 1988-10-11
US4820708A (en) 1989-04-11
ES552617A0 (es) 1987-09-01
FI860909A0 (fi) 1986-03-04
PT82135B (en) 1988-06-24
NZ215362A (en) 1989-01-06
IL78026A (en) 1990-07-26
DK93986D0 (da) 1986-02-28
GR860596B (en) 1986-06-26
PT82135A (en) 1986-04-01
ES8707949A1 (es) 1987-09-01
ZW4786A1 (en) 1987-09-16
AU578141B2 (en) 1988-10-13
FI860909A (fi) 1986-09-06
NO860830L (no) 1986-09-08
PH23532A (en) 1989-08-25
JO1443B1 (en) 1988-03-10
EP0198583A1 (en) 1986-10-22

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