DK540879A - METHOD OF PREPARING 4-AMINO-2-PIPERIDINOQUINAZOLINE DERIVATIVES AND SALTS THEREOF - Google Patents

METHOD OF PREPARING 4-AMINO-2-PIPERIDINOQUINAZOLINE DERIVATIVES AND SALTS THEREOF

Info

Publication number
DK540879A
DK540879A DK540879A DK540879A DK540879A DK 540879 A DK540879 A DK 540879A DK 540879 A DK540879 A DK 540879A DK 540879 A DK540879 A DK 540879A DK 540879 A DK540879 A DK 540879A
Authority
DK
Denmark
Prior art keywords
piperidinoquinazoline
derivatives
salts
amino
preparing
Prior art date
Application number
DK540879A
Other languages
Danish (da)
Inventor
S F Campbell
J C Danilewicz
C W Greengrass
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of DK540879A publication Critical patent/DK540879A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D211/00Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/40Oxygen atoms
    • C07D211/44Oxygen atoms attached in position 4
    • C07D211/46Oxygen atoms attached in position 4 having a hydrogen atom as the second substituent in position 4
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
DK540879A 1979-01-31 1979-12-18 METHOD OF PREPARING 4-AMINO-2-PIPERIDINOQUINAZOLINE DERIVATIVES AND SALTS THEREOF DK540879A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB7903398 1979-01-31

Publications (1)

Publication Number Publication Date
DK540879A true DK540879A (en) 1980-08-01

Family

ID=10502852

Family Applications (1)

Application Number Title Priority Date Filing Date
DK540879A DK540879A (en) 1979-01-31 1979-12-18 METHOD OF PREPARING 4-AMINO-2-PIPERIDINOQUINAZOLINE DERIVATIVES AND SALTS THEREOF

Country Status (28)

Country Link
JP (1) JPS55104278A (en)
AR (1) AR222208A1 (en)
AT (1) AT373595B (en)
BE (1) BE881448A (en)
CA (1) CA1131636A (en)
CS (1) CS231970B2 (en)
DD (1) DD148720A5 (en)
DE (1) DE3003323A1 (en)
DK (1) DK540879A (en)
ES (1) ES488129A0 (en)
FI (1) FI63936C (en)
FR (1) FR2447919A1 (en)
GR (1) GR73626B (en)
HU (1) HU184233B (en)
IE (1) IE800178L (en)
IL (1) IL59252A (en)
IT (1) IT1149902B (en)
LU (1) LU82115A1 (en)
NL (1) NL8000571A (en)
NO (1) NO800230L (en)
NZ (1) NZ192744A (en)
PH (1) PH15436A (en)
PL (1) PL121890B1 (en)
PT (1) PT70749A (en)
SE (1) SE8000699L (en)
SU (1) SU895291A3 (en)
YU (1) YU22980A (en)
ZA (1) ZA80557B (en)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2483920A1 (en) * 1980-06-09 1981-12-11 Synthelabo Antihypertensive piperidino quinazoline(s) - prepd. from benzyloxy piperidine and a 2:halo-4:amino 6,7-di:methoxy quinazoline
ES8405389A1 (en) * 1981-09-09 1983-11-01 Orion Yhtymae Oy Substituted piperidinyl quinazolines.
US5280032A (en) * 1989-02-14 1994-01-18 Toyama Chemical Co., Ltd. 1,2-ethanediol derivative and salt thereof, process for producing the same, and cerebral function-improving agent comprising the same
US9458131B2 (en) * 2011-11-08 2016-10-04 Emory University Compounds and compositions used to epigenetically transform cells and methods related thereto

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1088068A (en) * 1977-11-16 1980-10-21 Simon F. Campbell Piperidino-quinazolines
GB2021108B (en) * 1978-05-18 1982-07-21 Pfizer Ltd 6,7 - di - 4 - amino - 2 - quinazolines

Also Published As

Publication number Publication date
IT1149902B (en) 1986-12-10
IL59252A0 (en) 1980-05-30
DE3003323A1 (en) 1980-08-14
HU184233B (en) 1984-07-30
FR2447919B1 (en) 1983-02-11
ES8101583A1 (en) 1980-12-16
PT70749A (en) 1980-02-01
SE8000699L (en) 1980-08-01
ES488129A0 (en) 1980-12-16
PH15436A (en) 1983-01-18
FI800252A (en) 1980-08-01
GR73626B (en) 1984-03-26
JPS55104278A (en) 1980-08-09
BE881448A (en) 1980-07-30
PL221683A1 (en) 1980-12-01
FI63936B (en) 1983-05-31
CS60780A2 (en) 1984-01-16
NO800230L (en) 1980-08-01
FR2447919A1 (en) 1980-08-29
AR222208A1 (en) 1981-04-30
IL59252A (en) 1983-11-30
YU22980A (en) 1983-02-28
DD148720A5 (en) 1981-06-10
CS231970B2 (en) 1985-01-16
NL8000571A (en) 1980-08-04
FI63936C (en) 1983-09-12
CA1131636A (en) 1982-09-14
PL121890B1 (en) 1982-06-30
ZA80557B (en) 1981-08-26
LU82115A1 (en) 1980-04-23
NZ192744A (en) 1984-03-30
AT373595B (en) 1984-02-10
IT8019537A0 (en) 1980-01-29
JPS5728711B2 (en) 1982-06-18
IE800178L (en) 1980-07-31
AU5502480A (en) 1980-08-07
SU895291A3 (en) 1981-12-30
ATA46980A (en) 1983-06-15

Similar Documents

Publication Publication Date Title
DK471479A (en) PROCEDURE FOR PREPARING IMIDAZOLD DERIVATIVES AND SALTS THEREOF
DK531479A (en) PROCEDURE FOR PREPARING IMIDAZOLD DERIVATIVES AND SALTS THEREOF
DK23981A (en) AGMATIN DERIVATIVES AND SALTS THEREOF THEIR PREPARATION AND APPLICATION
DK157301C (en) ANALOGY PROCEDURE FOR THE PREPARATION OF HYDANTOINE DERIVATIVES AND SALTS THEREOF
DK149842C (en) METHOD FOR PREPARING D-CAMPHORATE OF L-CARNITINAMIDE AND D-CAMPHORATE OF D-CARNITINAMIDE
DK140480A (en) METHOD OF PREPARING MERCAPTOACYLDIPEPTIDES
DK229980A (en) METHOD OF PREPARING N-HETEROCYCLYL-THIENAMYCINES
DK374679A (en) PROCEDURE FOR PREPARING 7BETA-AMINOTHIAZOLYL-ACETAMIDO-3-CEPHEM-4-CARBOXYLIC ACID COMPOUNDS AND SALTS THEREOF
DK149586C (en) PROCEDURE FOR PREPARING 1-AMINO-CYCLOPROPAN-CARBOXYLIC ACID AND DERIVATIVES THEREOF
DK437480A (en) PROCEDURE FOR PREPARING BENZODIAZEPINE DERIVATIVES AND SALTS THEREOF
DK263180A (en) METHOD OF PREPARING SUBSTITUTED 2-NITRO-5-PHENOXY BENZO ACIDS AND SALTS THEREOF
DK232080A (en) METHOD OF PREPARING HYDROXYAMINOEBURNAND DERIVATIVES
DK300781A (en) METHOD OF PREPARING HALOGENPHENYLPYRIDYLLYLAMINE DERIVATIVES
DK333179A (en) PROCEDURE FOR PREPARING SUBSTITUTED ANTHRANIC ACID AMOIDS AND SALTS THEREOF
DK567778A (en) PROCEDURE FOR THE PREPARATION OF QUATERAN AMMONIUM SALTS OF PHENYLPROPYLAMINES AND PHENYLBUTYLAMINES
DK316178A (en) PROCEDURE FOR THE PREPARATION OF BENZOPYRANE DERIVATIVES ESPECIALLY 3-OXALOAMINO-4-OXO4H-1-BENZOPYRANE DERIVATIVES AND SALTS THEREOF
DK469879A (en) ADENOSINTRIPHOSPHATE DERIVATIVES AND SALTS THEREOF
DK540879A (en) METHOD OF PREPARING 4-AMINO-2-PIPERIDINOQUINAZOLINE DERIVATIVES AND SALTS THEREOF
DK333279A (en) PROCEDURE FOR THE PREPARATION OF THIOS-SUBSTITUTED DIAZACYCLOALKENES AND SALTS THEREOF
DK319178A (en) PROCEDURE FOR THE PREPARATION OF ACYLAMIDO-2-CEPHEM-4-CARBOXYLIC ACID COMPOUNDS AND SALTS
DK196878A (en) PROCEDURE FOR THE PREPARATION OF PHENYLGLYCIN DERIVATIVES AND SALTS THEREOF
DK183880A (en) METHOD FOR PREPARING HYDROXYDER DERIVATIVES OF ISOPROPYRIMIDINE
DK286779A (en) PROCEDURE FOR PREPARING 7BETA-AMINOTHIAZOLYL-ACETAMIDO-3-CEPHEM-4-CARBOXYLIC ACID COMPOUNDS AND SALTS THEREOF
DK337182A (en) PROCEDURE FOR PREPARING 4-AMINO-BUTYRAMIDE AND SALTS THEREOF
DK257280A (en) METHOD OF PREPARING 3-THIENYLMALONIC ACID AND SALTS THEREOF

Legal Events

Date Code Title Description
ATS Application withdrawn