DK374679A - PROCEDURE FOR PREPARING 7BETA-AMINOTHIAZOLYL-ACETAMIDO-3-CEPHEM-4-CARBOXYLIC ACID COMPOUNDS AND SALTS THEREOF - Google Patents
PROCEDURE FOR PREPARING 7BETA-AMINOTHIAZOLYL-ACETAMIDO-3-CEPHEM-4-CARBOXYLIC ACID COMPOUNDS AND SALTS THEREOFInfo
- Publication number
- DK374679A DK374679A DK374679A DK374679A DK374679A DK 374679 A DK374679 A DK 374679A DK 374679 A DK374679 A DK 374679A DK 374679 A DK374679 A DK 374679A DK 374679 A DK374679 A DK 374679A
- Authority
- DK
- Denmark
- Prior art keywords
- aminothiazolyl
- cephem
- acetamido
- salts
- procedure
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/587—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with aliphatic hydrocarbon radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms, said aliphatic radicals being substituted in the alpha-position to the ring by a hetero atom, e.g. with m >= 0, Z being a singly or a doubly bound hetero atom
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Communicable Diseases (AREA)
- Pharmacology & Pharmacy (AREA)
- Oncology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Cephalosporin Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
CH946878 | 1978-09-08 |
Publications (1)
Publication Number | Publication Date |
---|---|
DK374679A true DK374679A (en) | 1980-03-09 |
Family
ID=4352310
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DK374679A DK374679A (en) | 1978-09-08 | 1979-09-07 | PROCEDURE FOR PREPARING 7BETA-AMINOTHIAZOLYL-ACETAMIDO-3-CEPHEM-4-CARBOXYLIC ACID COMPOUNDS AND SALTS THEREOF |
Country Status (5)
Country | Link |
---|---|
EP (1) | EP0009008A3 (en) |
JP (1) | JPS5538392A (en) |
DK (1) | DK374679A (en) |
ES (1) | ES483986A1 (en) |
ZA (1) | ZA794749B (en) |
Families Citing this family (18)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS57154175A (en) * | 1981-03-16 | 1982-09-22 | Mitsui Toatsu Chem Inc | 2-thiazoleamine derivative, its preparation, and drug composition comprising it |
JPS5838289A (en) * | 1981-08-29 | 1983-03-05 | Meiji Seika Kaisha Ltd | Improvement of chemical process |
EP0096297B1 (en) * | 1982-06-03 | 1988-06-15 | F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft | Process for the preparation of 1-sulfo-2-oxoazetidine derivatives |
FR2550200B1 (en) * | 1983-08-01 | 1988-04-08 | Fujisawa Pharmaceutical Co | PROCESS FOR THE PREPARATION OF CEPHEM COMPOUNDS WITH ANTIMICROBIAL ACTIVITY AND NOVEL PRODUCTS THUS OBTAINED |
EP0432042B1 (en) * | 1989-12-07 | 1996-08-28 | Meiji Seika Kaisha Ltd. | Cephalosporin derivatives and their production and uses |
IL100576A (en) * | 1991-01-18 | 1995-11-27 | Eli Lilley And Company | Cephalosporin antibiotics |
JPH05132488A (en) * | 1991-08-13 | 1993-05-28 | Meiji Seika Kaisha Ltd | New cephalosporin derivative |
JP2857532B2 (en) * | 1992-03-12 | 1999-02-17 | 明治製菓株式会社 | New cephalosporin derivatives |
TW427993B (en) * | 1993-09-09 | 2001-04-01 | Fujisawa Pharmaceutical Co | New cephem compounds |
US5698547A (en) * | 1994-04-01 | 1997-12-16 | Microcide Pharmaceuticals, Inc. | Cephalosporin antibiotics |
US5688786A (en) * | 1994-04-01 | 1997-11-18 | Microcide Pharmaceuticals, Inc. | β-lactam antibiotics |
EP0754184A1 (en) * | 1994-04-01 | 1997-01-22 | Microcide Pharmaceuticals, Inc. | Cephalosporin antibiotics |
US5498777A (en) * | 1994-07-20 | 1996-03-12 | Merck & Co., Inc. | 3-thioheteroaryl cephalosporin compounds, compositions and methods of use |
WO1996017850A1 (en) * | 1994-12-09 | 1996-06-13 | Fujisawa Pharmaceutical Co., Ltd. | Cephem compounds and pharmaceutical use thereof |
JP2845789B2 (en) | 1995-12-25 | 1999-01-13 | 株式会社トクヤマ | Method for producing aminothiazoleacetic acid derivative |
AUPN801196A0 (en) * | 1996-02-12 | 1996-03-07 | Fujisawa Pharmaceutical Co., Ltd. | New cephem compounds and pharmaceutical use thereof |
US6545004B1 (en) | 1999-10-27 | 2003-04-08 | Cytokinetics, Inc. | Methods and compositions utilizing quinazolinones |
US6599893B2 (en) * | 2000-08-29 | 2003-07-29 | Essential Therapeutics, Inc. | Cephalosporin antibiotics and prodrugs thereof |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CH605997A5 (en) * | 1974-08-30 | 1978-10-13 | Ciba Geigy Ag | |
JPS53103493A (en) * | 1977-02-18 | 1978-09-08 | Takeda Chem Ind Ltd | Cephalosporin derivatives and process for their preparation |
FR2384779A1 (en) * | 1977-03-25 | 1978-10-20 | Roussel Uclaf | NEW OXIMES DERIVED FROM 3-CHLORO OR 3-METHOXY 7-AMINO THIAZOLYL ACETAMIDO CEPHALOSPORANIC, THEIR PREPARATION PROCESS AND THEIR APPLICATION AS MEDICINAL PRODUCTS |
-
1979
- 1979-09-03 EP EP79810085A patent/EP0009008A3/en not_active Withdrawn
- 1979-09-07 ES ES483986A patent/ES483986A1/en not_active Expired
- 1979-09-07 DK DK374679A patent/DK374679A/en unknown
- 1979-09-07 ZA ZA00794749A patent/ZA794749B/en unknown
- 1979-09-08 JP JP11563379A patent/JPS5538392A/en active Pending
Also Published As
Publication number | Publication date |
---|---|
EP0009008A2 (en) | 1980-03-19 |
JPS5538392A (en) | 1980-03-17 |
ES483986A1 (en) | 1980-04-16 |
ZA794749B (en) | 1980-08-27 |
EP0009008A3 (en) | 1980-05-14 |
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