DK374679A - PROCEDURE FOR PREPARING 7BETA-AMINOTHIAZOLYL-ACETAMIDO-3-CEPHEM-4-CARBOXYLIC ACID COMPOUNDS AND SALTS THEREOF - Google Patents

PROCEDURE FOR PREPARING 7BETA-AMINOTHIAZOLYL-ACETAMIDO-3-CEPHEM-4-CARBOXYLIC ACID COMPOUNDS AND SALTS THEREOF

Info

Publication number
DK374679A
DK374679A DK374679A DK374679A DK374679A DK 374679 A DK374679 A DK 374679A DK 374679 A DK374679 A DK 374679A DK 374679 A DK374679 A DK 374679A DK 374679 A DK374679 A DK 374679A
Authority
DK
Denmark
Prior art keywords
aminothiazolyl
cephem
acetamido
salts
procedure
Prior art date
Application number
DK374679A
Other languages
Danish (da)
Inventor
P Schneider
R Wiederkehr
P Wenk
R Scartazzini
Original Assignee
Ciba Geigy Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ciba Geigy Ag filed Critical Ciba Geigy Ag
Publication of DK374679A publication Critical patent/DK374679A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D277/00Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/587Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with aliphatic hydrocarbon radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms, said aliphatic radicals being substituted in the alpha-position to the ring by a hetero atom, e.g. with m >= 0, Z being a singly or a doubly bound hetero atom
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Cephalosporin Compounds (AREA)
DK374679A 1978-09-08 1979-09-07 PROCEDURE FOR PREPARING 7BETA-AMINOTHIAZOLYL-ACETAMIDO-3-CEPHEM-4-CARBOXYLIC ACID COMPOUNDS AND SALTS THEREOF DK374679A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH946878 1978-09-08

Publications (1)

Publication Number Publication Date
DK374679A true DK374679A (en) 1980-03-09

Family

ID=4352310

Family Applications (1)

Application Number Title Priority Date Filing Date
DK374679A DK374679A (en) 1978-09-08 1979-09-07 PROCEDURE FOR PREPARING 7BETA-AMINOTHIAZOLYL-ACETAMIDO-3-CEPHEM-4-CARBOXYLIC ACID COMPOUNDS AND SALTS THEREOF

Country Status (5)

Country Link
EP (1) EP0009008A3 (en)
JP (1) JPS5538392A (en)
DK (1) DK374679A (en)
ES (1) ES483986A1 (en)
ZA (1) ZA794749B (en)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS57154175A (en) * 1981-03-16 1982-09-22 Mitsui Toatsu Chem Inc 2-thiazoleamine derivative, its preparation, and drug composition comprising it
JPS5838289A (en) * 1981-08-29 1983-03-05 Meiji Seika Kaisha Ltd Improvement of chemical process
EP0096297B1 (en) * 1982-06-03 1988-06-15 F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft Process for the preparation of 1-sulfo-2-oxoazetidine derivatives
FR2550200B1 (en) * 1983-08-01 1988-04-08 Fujisawa Pharmaceutical Co PROCESS FOR THE PREPARATION OF CEPHEM COMPOUNDS WITH ANTIMICROBIAL ACTIVITY AND NOVEL PRODUCTS THUS OBTAINED
EP0432042B1 (en) * 1989-12-07 1996-08-28 Meiji Seika Kaisha Ltd. Cephalosporin derivatives and their production and uses
IL100576A (en) * 1991-01-18 1995-11-27 Eli Lilley And Company Cephalosporin antibiotics
JPH05132488A (en) * 1991-08-13 1993-05-28 Meiji Seika Kaisha Ltd New cephalosporin derivative
JP2857532B2 (en) * 1992-03-12 1999-02-17 明治製菓株式会社 New cephalosporin derivatives
TW427993B (en) * 1993-09-09 2001-04-01 Fujisawa Pharmaceutical Co New cephem compounds
US5698547A (en) * 1994-04-01 1997-12-16 Microcide Pharmaceuticals, Inc. Cephalosporin antibiotics
US5688786A (en) * 1994-04-01 1997-11-18 Microcide Pharmaceuticals, Inc. β-lactam antibiotics
EP0754184A1 (en) * 1994-04-01 1997-01-22 Microcide Pharmaceuticals, Inc. Cephalosporin antibiotics
US5498777A (en) * 1994-07-20 1996-03-12 Merck & Co., Inc. 3-thioheteroaryl cephalosporin compounds, compositions and methods of use
WO1996017850A1 (en) * 1994-12-09 1996-06-13 Fujisawa Pharmaceutical Co., Ltd. Cephem compounds and pharmaceutical use thereof
JP2845789B2 (en) 1995-12-25 1999-01-13 株式会社トクヤマ Method for producing aminothiazoleacetic acid derivative
AUPN801196A0 (en) * 1996-02-12 1996-03-07 Fujisawa Pharmaceutical Co., Ltd. New cephem compounds and pharmaceutical use thereof
US6545004B1 (en) 1999-10-27 2003-04-08 Cytokinetics, Inc. Methods and compositions utilizing quinazolinones
US6599893B2 (en) * 2000-08-29 2003-07-29 Essential Therapeutics, Inc. Cephalosporin antibiotics and prodrugs thereof

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH605997A5 (en) * 1974-08-30 1978-10-13 Ciba Geigy Ag
JPS53103493A (en) * 1977-02-18 1978-09-08 Takeda Chem Ind Ltd Cephalosporin derivatives and process for their preparation
FR2384779A1 (en) * 1977-03-25 1978-10-20 Roussel Uclaf NEW OXIMES DERIVED FROM 3-CHLORO OR 3-METHOXY 7-AMINO THIAZOLYL ACETAMIDO CEPHALOSPORANIC, THEIR PREPARATION PROCESS AND THEIR APPLICATION AS MEDICINAL PRODUCTS

Also Published As

Publication number Publication date
EP0009008A2 (en) 1980-03-19
JPS5538392A (en) 1980-03-17
ES483986A1 (en) 1980-04-16
ZA794749B (en) 1980-08-27
EP0009008A3 (en) 1980-05-14

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