FI800252A - PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ANALYTICAL BAR 4-AMINO-2-PIPERIDINOKINAZOLINE - Google Patents

PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ANALYTICAL BAR 4-AMINO-2-PIPERIDINOKINAZOLINE

Info

Publication number
FI800252A
FI800252A FI800252A FI800252A FI800252A FI 800252 A FI800252 A FI 800252A FI 800252 A FI800252 A FI 800252A FI 800252 A FI800252 A FI 800252A FI 800252 A FI800252 A FI 800252A
Authority
FI
Finland
Prior art keywords
piperidinokinazoline
amino
procedure
preparation
bar
Prior art date
Application number
FI800252A
Other languages
Finnish (fi)
Other versions
FI63936C (en
FI63936B (en
Inventor
Simon Fraser Campbell
John Christopher Danilewicz
Colin William Greengrass
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of FI800252A publication Critical patent/FI800252A/en
Application granted granted Critical
Publication of FI63936B publication Critical patent/FI63936B/en
Publication of FI63936C publication Critical patent/FI63936C/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D211/00Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/40Oxygen atoms
    • C07D211/44Oxygen atoms attached in position 4
    • C07D211/46Oxygen atoms attached in position 4 having a hydrogen atom as the second substituent in position 4
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
FI800252A 1979-01-31 1980-01-29 ANALOGIFICATION OF FRAMSTATION OF AV 4-AMINO-2- (4- (PHENYL SUBSTITUTES ALCOXY) PIPERIDINO) QUINAZOLINE ANVAENDBARA SAOSOMANTIHYPERTENSIVA MEDEL FI63936C (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB7903398 1979-01-31
GB7903398 1979-01-31

Publications (3)

Publication Number Publication Date
FI800252A true FI800252A (en) 1980-08-01
FI63936B FI63936B (en) 1983-05-31
FI63936C FI63936C (en) 1983-09-12

Family

ID=10502852

Family Applications (1)

Application Number Title Priority Date Filing Date
FI800252A FI63936C (en) 1979-01-31 1980-01-29 ANALOGIFICATION OF FRAMSTATION OF AV 4-AMINO-2- (4- (PHENYL SUBSTITUTES ALCOXY) PIPERIDINO) QUINAZOLINE ANVAENDBARA SAOSOMANTIHYPERTENSIVA MEDEL

Country Status (28)

Country Link
JP (1) JPS55104278A (en)
AR (1) AR222208A1 (en)
AT (1) AT373595B (en)
BE (1) BE881448A (en)
CA (1) CA1131636A (en)
CS (1) CS231970B2 (en)
DD (1) DD148720A5 (en)
DE (1) DE3003323A1 (en)
DK (1) DK540879A (en)
ES (1) ES488129A0 (en)
FI (1) FI63936C (en)
FR (1) FR2447919A1 (en)
GR (1) GR73626B (en)
HU (1) HU184233B (en)
IE (1) IE800178L (en)
IL (1) IL59252A (en)
IT (1) IT1149902B (en)
LU (1) LU82115A1 (en)
NL (1) NL8000571A (en)
NO (1) NO800230L (en)
NZ (1) NZ192744A (en)
PH (1) PH15436A (en)
PL (1) PL121890B1 (en)
PT (1) PT70749A (en)
SE (1) SE8000699L (en)
SU (1) SU895291A3 (en)
YU (1) YU22980A (en)
ZA (1) ZA80557B (en)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2483920A1 (en) * 1980-06-09 1981-12-11 Synthelabo Antihypertensive piperidino quinazoline(s) - prepd. from benzyloxy piperidine and a 2:halo-4:amino 6,7-di:methoxy quinazoline
ES515338A0 (en) * 1981-09-09 1983-11-01 Orion Yhtymae Oy "METHOD FOR THE PREPARATION OF SUBSTITUTED PIPERIDINYLQUINAZOLIDINES".
US5280032A (en) * 1989-02-14 1994-01-18 Toyama Chemical Co., Ltd. 1,2-ethanediol derivative and salt thereof, process for producing the same, and cerebral function-improving agent comprising the same
US9458131B2 (en) * 2011-11-08 2016-10-04 Emory University Compounds and compositions used to epigenetically transform cells and methods related thereto

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1088068A (en) * 1977-11-16 1980-10-21 Simon F. Campbell Piperidino-quinazolines
GB2021108B (en) * 1978-05-18 1982-07-21 Pfizer Ltd 6,7 - di - 4 - amino - 2 - quinazolines

Also Published As

Publication number Publication date
PH15436A (en) 1983-01-18
FI63936C (en) 1983-09-12
HU184233B (en) 1984-07-30
SE8000699L (en) 1980-08-01
ES8101583A1 (en) 1980-12-16
FI63936B (en) 1983-05-31
IT8019537A0 (en) 1980-01-29
CS60780A2 (en) 1984-01-16
FR2447919A1 (en) 1980-08-29
LU82115A1 (en) 1980-04-23
NO800230L (en) 1980-08-01
CS231970B2 (en) 1985-01-16
JPS55104278A (en) 1980-08-09
NZ192744A (en) 1984-03-30
NL8000571A (en) 1980-08-04
IT1149902B (en) 1986-12-10
CA1131636A (en) 1982-09-14
JPS5728711B2 (en) 1982-06-18
YU22980A (en) 1983-02-28
ZA80557B (en) 1981-08-26
AT373595B (en) 1984-02-10
IL59252A (en) 1983-11-30
IE800178L (en) 1980-07-31
PT70749A (en) 1980-02-01
BE881448A (en) 1980-07-30
DE3003323A1 (en) 1980-08-14
DK540879A (en) 1980-08-01
AR222208A1 (en) 1981-04-30
IL59252A0 (en) 1980-05-30
AU5502480A (en) 1980-08-07
FR2447919B1 (en) 1983-02-11
DD148720A5 (en) 1981-06-10
PL121890B1 (en) 1982-06-30
SU895291A3 (en) 1981-12-30
GR73626B (en) 1984-03-26
ATA46980A (en) 1983-06-15
PL221683A1 (en) 1980-12-01
ES488129A0 (en) 1980-12-16

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Legal Events

Date Code Title Description
MM Patent lapsed

Owner name: PFIZER CORPORATION