DK530681A - Hidtil ukendte laegemidler paa basis af derivater af 1-(4-quinolyl)-2-(4-piperidyl)-ethanol eller 1-(4-quinolyl)-3-(4-piperidyl)-propanol - Google Patents

Hidtil ukendte laegemidler paa basis af derivater af 1-(4-quinolyl)-2-(4-piperidyl)-ethanol eller 1-(4-quinolyl)-3-(4-piperidyl)-propanol

Info

Publication number
DK530681A
DK530681A DK530681A DK530681A DK530681A DK 530681 A DK530681 A DK 530681A DK 530681 A DK530681 A DK 530681A DK 530681 A DK530681 A DK 530681A DK 530681 A DK530681 A DK 530681A
Authority
DK
Denmark
Prior art keywords
piperidyl
quinolyl
propanol
ethanol
derivatives
Prior art date
Application number
DK530681A
Other languages
Danish (da)
English (en)
Inventor
C Gueremy
M Mestre
C Renault
Original Assignee
Pharmindustrie
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pharmindustrie filed Critical Pharmindustrie
Publication of DK530681A publication Critical patent/DK530681A/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/06Antiarrhythmics

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Hydrogenated Pyridines (AREA)
DK530681A 1980-12-05 1981-11-30 Hidtil ukendte laegemidler paa basis af derivater af 1-(4-quinolyl)-2-(4-piperidyl)-ethanol eller 1-(4-quinolyl)-3-(4-piperidyl)-propanol DK530681A (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR8025829A FR2495470A1 (fr) 1980-12-05 1980-12-05 Nouveaux medicaments a base de derives de (quinolyl-4)-1 (piperidyl-4)-2 ethanol ou (quinolyl-4)-1 (piperidyl-4)-3 propanol

Publications (1)

Publication Number Publication Date
DK530681A true DK530681A (da) 1982-06-06

Family

ID=9248697

Family Applications (1)

Application Number Title Priority Date Filing Date
DK530681A DK530681A (da) 1980-12-05 1981-11-30 Hidtil ukendte laegemidler paa basis af derivater af 1-(4-quinolyl)-2-(4-piperidyl)-ethanol eller 1-(4-quinolyl)-3-(4-piperidyl)-propanol

Country Status (18)

Country Link
US (1) US4613607A (xx)
EP (1) EP0053964B1 (xx)
JP (1) JPS57122081A (xx)
AR (1) AR231289A1 (xx)
AT (1) AT378958B (xx)
AU (1) AU548800B2 (xx)
CA (1) CA1261841A (xx)
DE (1) DE3174581D1 (xx)
DK (1) DK530681A (xx)
ES (1) ES8303397A1 (xx)
FR (1) FR2495470A1 (xx)
GR (1) GR76939B (xx)
HU (1) HU187480B (xx)
IL (1) IL64201A (xx)
MA (1) MA19348A1 (xx)
NO (1) NO159532C (xx)
PT (1) PT74081B (xx)
ZA (1) ZA818387B (xx)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL8100877A (nl) * 1981-02-23 1982-09-16 Acf Chemiefarma Nv Farmaceutisch preparaaat met als werkzaam bestanddeel een chinolinederivaat, werkwijze voor de bereiding van een dergelijk preparaat, nieuwe chinolinederivaten en werkwijze voor de bereiding ervan.
FR2560877B1 (fr) * 1984-03-09 1986-09-05 Rhone Poulenc Sante Derives de (quinolyl-4)-1 (piperidyl-4)-2 ethanamine et de (quinolyl-4)-1 (piperidyl-4)-3 propanamine, procedes pour leur preparation et medicaments les contenant
GB9819382D0 (en) * 1998-09-04 1998-10-28 Cerebrus Ltd Chemical compounds I
GB9917408D0 (en) * 1999-07-23 1999-09-22 Smithkline Beecham Plc Compounds
GB9917406D0 (en) 1999-07-23 1999-09-22 Smithkline Beecham Plc Compounds
US6376514B1 (en) * 2000-10-17 2002-04-23 The Procter & Gamble Co. Substituted six-membered heterocyclic compounds useful for treating multidrug resistance and compositions and methods thereof
US6693099B2 (en) * 2000-10-17 2004-02-17 The Procter & Gamble Company Substituted piperazine compounds optionally containing a quinolyl moiety for treating multidrug resistance
TW200406410A (en) 2002-01-29 2004-05-01 Glaxo Group Ltd Compounds
AU2008249745B2 (en) * 2007-05-09 2012-01-12 Pfizer Inc. Substituted heterocyclic derivatives and compositions and their pharmaceutical use as antibacterials

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE330813C (de) * 1918-03-08 1920-12-18 Ver Chininfabriken Zimmer & Co Verfahren zur Darstellung von Alkoholen und Aminoalkoholen der Chinolinreihe
US3914235A (en) * 1968-07-02 1975-10-21 Hoffmann La Roche Processes and intermediates for quinine, quinidine, isomers and derivatives thereof
FR2177511A1 (en) * 1972-03-28 1973-11-09 Omnium Chimique Sa Quinolyl pipiridylethyl ketones - with vasodilatory and antispasmodic activity
GB1441244A (en) * 1972-11-17 1976-06-30 Rech Et Dapplications Scient S Derivatives of quinoline and method of preparing the same
US3953453A (en) * 1973-12-07 1976-04-27 Hoffmann-La Roche Inc. Trifluoromethyl substituted analogs of quinine and quinidine
PT66682B (pt) * 1976-06-18 1978-11-15 Ind Biolog Francaise /(quinolyl-4)-propyl-1/-4 piperidines leur preparation et leur utilisation comme medicaments /(quinolyl-4)-propyl/-4 piperidines leur preparation et leur utilisation comme medicaments
FR2354771A1 (fr) * 1976-06-18 1978-01-13 Mar Pha Etu Expl Marques ((quinolyl-4)-3 propyl-1) -4 piperidines, leur preparation et leur utilisation comme medicaments
NL7908030A (nl) * 1979-11-01 1981-06-01 Acf Chemiefarma Nv Nieuwe chinolinederivaten en farmaceutische preparaten die een dergelijke verbinding bevatten, alsmede werk- wijze voor het bereiden van deze verbindingen.
NL7908031A (nl) * 1979-11-01 1981-06-01 Acf Chemiefarma Nv Nieuwe chinolinederivaten en farmaceutische preparaten die een dergelijke verbinding bevatten, alsmede werk- wijze voor het bereiden van deze verbindingen.
FR2471981A1 (fr) * 1979-12-21 1981-06-26 Pharmindustrie Nouveaux derives de la (piperidyl-4)-2 (quinolyl-4)-1 ethanone, produits intermediaires et procedes pour leur preparation, et leur utilisation comme medicaments
US4442107A (en) * 1980-03-06 1984-04-10 Acf Chemiefarma N.V. Quinoline derivatives, pharmaceutical compositions containing such compounds, and methods for treating cardiovascular conditions with them
GR74482B (xx) * 1980-03-06 1984-06-28 Acf Chemiefarma Nv
NL8001369A (nl) * 1980-03-06 1981-10-01 Acf Chemiefarma Nv Nieuwe chinolinederivaten en farmaceutische preparaten die een dergelijke verbinding bevatten, alsmede werkwijze voor het bereiden van deze verbindingen.
IL62240A0 (en) * 1980-03-06 1981-05-20 Acf Chemiefarma Nv Novel quinoline derivatives,pharmaceutical compositions containing such compounds,and methods for the preparation of these compounds
FR2477544A1 (fr) * 1980-03-07 1981-09-11 Pharmindustrie Nouveaux derives de la chloro-3 quinoleine, procedes pour leur preparation, et leur utilisation comme medicaments
FR2485014A1 (fr) * 1980-06-20 1981-12-24 Pharmindustrie Nouveaux derives de (quinolyl-2, -3 ou -4)-1 (piperidyl ou pyrrolidinyl-2 ou -3)-2 ou -3 ethanone ou propanone, procedes pour leur preparation, et leur utilisation comme medicaments

Also Published As

Publication number Publication date
GR76939B (xx) 1984-09-04
DE3174581D1 (en) 1986-06-12
NO814157L (no) 1982-06-07
FR2495470A1 (fr) 1982-06-11
US4613607A (en) 1986-09-23
JPS6337111B2 (xx) 1988-07-22
EP0053964B1 (fr) 1986-05-07
HU187480B (en) 1986-01-28
MA19348A1 (fr) 1982-07-01
IL64201A (en) 1985-09-29
ZA818387B (en) 1982-10-27
AU548800B2 (en) 1986-01-02
JPS57122081A (en) 1982-07-29
AU7828081A (en) 1982-06-10
PT74081A (fr) 1982-01-01
ATA517781A (de) 1985-03-15
PT74081B (fr) 1983-05-11
AR231289A1 (es) 1984-10-31
AT378958B (de) 1985-10-25
ES507758A0 (es) 1983-02-01
ES8303397A1 (es) 1983-02-01
NO159532B (no) 1988-10-03
NO159532C (no) 1989-01-11
EP0053964A1 (fr) 1982-06-16
FR2495470B1 (xx) 1983-06-10
IL64201A0 (en) 1982-02-28
CA1261841A (fr) 1989-09-26

Similar Documents

Publication Publication Date Title
DK157301C (da) Analogifremgangsmaade til fremstilling af hydantoinderivater og salte deraf
NO159531C (no) Analogifremgangsmaate for fremstilling av farmasoeytisk aktive karbostyrilderivater.
FI811350L (fi) Aminocyklopentanalkensyror och -estrar samt framstaellning och farmaceutiska preparat av dessa
DK13082A (da) Analogifremgangsmaade til fremstilling af n-(2-pyridyl)-2-methyl-4-hydroxy-2h-1,2-benzothiazin-3-carboxamid-1,1-dioxid-derivater
DK160561C (da) Analogifremgangsmaade til fremstilling af 3-aminopregn-5-enderivater eller salte deraf
DK530681A (da) Hidtil ukendte laegemidler paa basis af derivater af 1-(4-quinolyl)-2-(4-piperidyl)-ethanol eller 1-(4-quinolyl)-3-(4-piperidyl)-propanol
DK493083D0 (da) Fremgangsmaade til fremstilling af 4-oxo-1,4-dihydfremgangsmade til fremstilling af 4-oxo-1,4-dihydronicotinsyrederivater eller salte deraf ronicotinsyrederivater eller salte deraf
DK130382A (da) Fremgangsmaade til fremstilling af quinolinderivater eller salte deraf
DK514182A (da) Fremgangsmaade til fremstilling af n-substituerede 2-pyridylindoler eller n-oxider eller salte deraf
FI822373A0 (fi) Saett och anordning foer uppvaermning av foer industriella aendamaol avsedd processluft
NL7902211A (nl) Werkwijze voor het hanteren van polymeer-brij.
AR231134A1 (es) Procedimiento para obtener derivados de 4-(sulfamoilfenil)-2-(hidroxi-o aciloxi-fenilimino)-tiazolina
NO800910L (no) Nye derivater av 2-(2-pyridyl)tetrahydrotiofen.
DK164288C (da) Maskinopvaskemiddel paa basis af chlorisocyanuratderivat samt fremgangsmaade til fremstilling af et saadant middel
NO157652C (no) Fremgangsmaate for fremstilling av 3-pikolin.
DK224381A (da) Fremgangsmaade til fremstilling af benzazolderivater eller salte deraf
NO154193C (no) Fremgangsmaate for fremstilling av monohydratisert picotamid
DK149823C (da) Fremgangsmaade til fremstilling af kijanimicin eller farmaceutisk acceptable salte heraf
NO821806L (no) Prosedyre for bestemmelse av belegningshastigheter
SE8007240L (sv) Anordning for overforing av serveringsbrickor och liknande
DK7483A (da) Fremgangsmaade til fremstilling af 6-aminoalkylpencillansyre-1,1-dioxider samt derivater deraf
FI813913L (fi) 1,2-dihydro-5-(pyridinyl)nikotinamidderivat och deras framstaellning
DK151797C (da) Analogifremgangsmaade til fremstilling af terbutalinderivater eller terapeutisk acceptable salte deraf
FI844951A0 (fi) Nya 2-(1-imidazolyl)-etanol-derivat.
AR229111A1 (es) Procedimiento para la preparacion de nicotinatos de 4-(fenilalquiloxi 4-sustituido)fenilalquilo

Legal Events

Date Code Title Description
AHB Application shelved due to non-payment