DK451888A - C12-modificerede erythromycin-a-derivater og fremgangsmaade til fremstilling deraf samt forbindelser til anvendelse som udgangsmateriale ved fremgangsmaaden - Google Patents

C12-modificerede erythromycin-a-derivater og fremgangsmaade til fremstilling deraf samt forbindelser til anvendelse som udgangsmateriale ved fremgangsmaaden

Info

Publication number
DK451888A
DK451888A DK451888A DK451888A DK451888A DK 451888 A DK451888 A DK 451888A DK 451888 A DK451888 A DK 451888A DK 451888 A DK451888 A DK 451888A DK 451888 A DK451888 A DK 451888A
Authority
DK
Denmark
Prior art keywords
derivatives
procedures
preparing
modified erythromycin
erythromycin
Prior art date
Application number
DK451888A
Other languages
Danish (da)
English (en)
Other versions
DK451888D0 (da
Inventor
James Robert Hauske
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of DK451888D0 publication Critical patent/DK451888D0/da
Publication of DK451888A publication Critical patent/DK451888A/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Communicable Diseases (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
DK451888A 1987-08-14 1988-08-12 C12-modificerede erythromycin-a-derivater og fremgangsmaade til fremstilling deraf samt forbindelser til anvendelse som udgangsmateriale ved fremgangsmaaden DK451888A (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US07/085,446 US4857641A (en) 1987-08-14 1987-08-14 C.12 modified erythromycin A derivatives

Publications (2)

Publication Number Publication Date
DK451888D0 DK451888D0 (da) 1988-08-12
DK451888A true DK451888A (da) 1989-02-15

Family

ID=22191650

Family Applications (1)

Application Number Title Priority Date Filing Date
DK451888A DK451888A (da) 1987-08-14 1988-08-12 C12-modificerede erythromycin-a-derivater og fremgangsmaade til fremstilling deraf samt forbindelser til anvendelse som udgangsmateriale ved fremgangsmaaden

Country Status (12)

Country Link
US (1) US4857641A (el)
EP (1) EP0303471B1 (el)
JP (1) JPH0667957B2 (el)
AT (1) ATE69235T1 (el)
CA (1) CA1296718C (el)
DE (1) DE3866057D1 (el)
DK (1) DK451888A (el)
ES (1) ES2037838T3 (el)
FI (1) FI88925C (el)
GR (1) GR3002962T3 (el)
IE (1) IE61042B1 (el)
PT (1) PT88254B (el)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL99995A (en) * 1990-11-21 1997-11-20 Roussel Uclaf Erythromycin derivatives, their preparation and pharmaceutical compositions containing them
US6060234A (en) * 1991-01-17 2000-05-09 Abbott Laboratories Polyketide derivatives and recombinant methods for making same
US6063561A (en) * 1991-01-17 2000-05-16 Abbott Laboratories Polyketide derivatives and recombinant methods for making same
US5217960A (en) * 1991-05-03 1993-06-08 Abbott Laboratories Erythromycin derivatives
CA2451391A1 (en) 2001-07-03 2003-01-16 Chiron Corporation C12 modified erythromycin macrolides and ketolides having antibacterial activity
JP4796300B2 (ja) * 2002-08-29 2011-10-19 ファイザー インコーポレイテッド モチライド化合物
JP2006524706A (ja) 2003-04-25 2006-11-02 カイロン コーポレイション 新規なケトライド誘導体
CA2523134A1 (en) 2003-04-25 2004-11-11 Chiron Corporation Pyridyl substituted ketolide antibiotics
US7211568B2 (en) * 2003-12-18 2007-05-01 Kosan Biosciences Incorporated 9-Desoxoerythromycin compounds as prokinetic agents

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3864347A (en) * 1968-07-02 1975-02-04 Hoffmann La Roche {60 {8 3(R)-alkyl-4(R) piperidyl methyl{9 -{62 -(6,7 substituted-4 quinolyl)-2-alkanoyloxy propane and racemates
US4672056A (en) * 1985-11-12 1987-06-09 Abbott Laboratories Erythromycin A derivatives and method of use
US4686207A (en) * 1985-11-12 1987-08-11 Abbott Laboratories Erythromycin A 11,12-carbonates and method of use

Also Published As

Publication number Publication date
IE61042B1 (en) 1994-09-07
FI88925B (fi) 1993-04-15
DK451888D0 (da) 1988-08-12
ATE69235T1 (de) 1991-11-15
PT88254A (pt) 1989-06-30
FI88925C (fi) 1993-07-26
IE882475L (en) 1989-02-14
PT88254B (pt) 1995-03-01
ES2037838T3 (es) 1993-07-01
GR3002962T3 (en) 1993-01-25
DE3866057D1 (en) 1991-12-12
US4857641A (en) 1989-08-15
JPH01100189A (ja) 1989-04-18
EP0303471A3 (en) 1989-10-25
FI883759A0 (fi) 1988-08-12
FI883759A (fi) 1989-02-15
JPH0667957B2 (ja) 1994-08-31
EP0303471A2 (en) 1989-02-15
EP0303471B1 (en) 1991-11-06
CA1296718C (en) 1992-03-03

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Legal Events

Date Code Title Description
AHB Application shelved due to non-payment