DK428477A - 1h-pyrazolo (3,4-b)pyridiner og fremgangsmaade til fremstilling deraf - Google Patents

1h-pyrazolo (3,4-b)pyridiner og fremgangsmaade til fremstilling deraf

Info

Publication number
DK428477A
DK428477A DK428477A DK428477A DK428477A DK 428477 A DK428477 A DK 428477A DK 428477 A DK428477 A DK 428477A DK 428477 A DK428477 A DK 428477A DK 428477 A DK428477 A DK 428477A
Authority
DK
Denmark
Prior art keywords
pyrazolo
pyridines
manufacture
methods
Prior art date
Application number
DK428477A
Other languages
English (en)
Other versions
DK143183B (da
DK143183C (da
Inventor
J Roch
E Mueller
B Narr
J Nickl
W Haarmann
Original Assignee
Thomae Gmbh Dr K
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Thomae Gmbh Dr K filed Critical Thomae Gmbh Dr K
Publication of DK428477A publication Critical patent/DK428477A/da
Publication of DK143183B publication Critical patent/DK143183B/da
Application granted granted Critical
Publication of DK143183C publication Critical patent/DK143183C/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D213/84—Nitriles
    • C07D213/85—Nitriles in position 3

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DK428477A 1976-09-29 1977-09-28 Analogifremgangsmaade til fremstilling af 1h-pyrazolo(3,4-b)pyridiner eller fysiologisk acceptable salte deraf DK143183C (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE19762643753 DE2643753A1 (de) 1976-09-29 1976-09-29 Neue 1h-pyrazolo eckige klammer auf 3,4-b eckige klammer zu pyridine
DE2643753 1976-09-29

Publications (3)

Publication Number Publication Date
DK428477A true DK428477A (da) 1978-03-30
DK143183B DK143183B (da) 1981-07-13
DK143183C DK143183C (da) 1981-11-16

Family

ID=5989097

Family Applications (1)

Application Number Title Priority Date Filing Date
DK428477A DK143183C (da) 1976-09-29 1977-09-28 Analogifremgangsmaade til fremstilling af 1h-pyrazolo(3,4-b)pyridiner eller fysiologisk acceptable salte deraf

Country Status (21)

Country Link
US (3) US4182887A (da)
JP (1) JPS5344588A (da)
AT (1) AT359064B (da)
AU (1) AU513406B2 (da)
BE (1) BE859152A (da)
DE (1) DE2643753A1 (da)
DK (1) DK143183C (da)
ES (1) ES462700A1 (da)
FI (1) FI61899C (da)
FR (1) FR2366290A1 (da)
GB (1) GB1552730A (da)
GR (1) GR64049B (da)
IE (1) IE45700B1 (da)
IL (1) IL52997A (da)
LU (1) LU78179A1 (da)
NL (1) NL7710573A (da)
NO (1) NO147913C (da)
NZ (1) NZ185292A (da)
PT (1) PT67091B (da)
SE (1) SE7710873L (da)
ZA (1) ZA775784B (da)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2643753A1 (de) * 1976-09-29 1978-04-06 Thomae Gmbh Dr K Neue 1h-pyrazolo eckige klammer auf 3,4-b eckige klammer zu pyridine
AR036873A1 (es) * 2001-09-07 2004-10-13 Euro Celtique Sa Piridinas aril sustituidas a, composiciones farmaceuticas y el uso de las mismas para la preparacion de un medicamento
AR037233A1 (es) 2001-09-07 2004-11-03 Euro Celtique Sa Piridinas aril sustituidas, composiciones farmaceuticas y el uso de dichos compuestos para la elaboracion de un medicamento
WO2005007648A2 (en) * 2003-07-16 2005-01-27 Neurogen Corporation Biaryl piperazinyl-pyridine analogues
EP1687004A4 (en) 2003-11-10 2009-04-08 Synta Pharmaceuticals Corp PYRIDINE COMPOUNDS
KR100881240B1 (ko) 2004-07-06 2009-02-05 에프. 호프만-라 로슈 아게 Nk-1 수용체 길항제의 합성에 있어서 중간체로서사용되는 카르복스아미드 피리딘 유도체의 제조 방법
MX2007000198A (es) * 2004-07-06 2007-03-15 Hoffmann La Roche Proceso para la preparacion de derivados de carboxamida-piridina utilizados como intermediarios en la sintesis de antagonistas del receptor nk-1.
MY145822A (en) * 2004-08-13 2012-04-30 Neurogen Corp Substituted biaryl piperazinyl-pyridine analogues
US7812166B2 (en) 2004-10-29 2010-10-12 Abbott Laboratories Kinase inhibitors
DE102004061288A1 (de) * 2004-12-14 2006-06-29 Schering Ag 3-Amino-Pyrazolo[3,4b]pyridine als Inhibitoren von Proteintyrosinkinasen, deren Herstellung und Verwendung als Arzneimittel
US7725056B2 (en) * 2006-01-10 2010-05-25 Ricoh Co., Ltd. Triboelectric charging device and field assisted toner transporter
EP2137162B1 (en) 2007-03-15 2018-08-01 Novartis AG Organic compounds and their uses
US20100041663A1 (en) 2008-07-18 2010-02-18 Novartis Ag Organic Compounds as Smo Inhibitors
CA2744154A1 (en) 2008-11-20 2010-05-27 Genentech, Inc. Pyrazolopyridine pi3k inhibitor compounds and methods of use
EP2789614B1 (en) 2009-08-11 2017-04-26 Bristol-Myers Squibb Company Azaindazoles as Btk kinase modulators and use thereof
CN112313232B (zh) * 2018-05-02 2024-03-08 Jw中外制药公司 新型杂环衍生物

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2232038A1 (de) * 1972-06-30 1974-01-10 Hoechst Ag 3-amino-1h-pyrazolo eckige klammer auf 3,4-b eckige klammer zu pyridine, ihre herstellung und verwendung
DE2643753A1 (de) * 1976-09-29 1978-04-06 Thomae Gmbh Dr K Neue 1h-pyrazolo eckige klammer auf 3,4-b eckige klammer zu pyridine
US4048184A (en) * 1976-11-15 1977-09-13 E. R. Squibb & Sons, Inc. 6-Phenyl-2H-pyrazolo[3,4-b]pyridines

Also Published As

Publication number Publication date
DK143183B (da) 1981-07-13
ATA670077A (de) 1980-03-15
FI772655A7 (fi) 1978-03-30
NZ185292A (en) 1980-05-08
ES462700A1 (es) 1978-06-01
PT67091A (de) 1977-10-01
IE45700L (en) 1978-03-29
AT359064B (de) 1980-10-27
US4260621A (en) 1981-04-07
AU2903777A (en) 1979-03-29
NO773327L (no) 1978-03-30
GB1552730A (en) 1979-09-19
IL52997A0 (en) 1977-11-30
SE7710873L (sv) 1978-03-30
FI61899B (fi) 1982-06-30
NO147913B (no) 1983-03-28
PT67091B (de) 1979-09-12
BE859152A (fr) 1978-03-28
JPS5344588A (en) 1978-04-21
DK143183C (da) 1981-11-16
AU513406B2 (en) 1980-11-27
FR2366290A1 (fr) 1978-04-28
US4182887A (en) 1980-01-08
GR64049B (en) 1980-01-19
FR2366290B1 (da) 1982-07-09
IL52997A (en) 1980-09-16
FI61899C (fi) 1982-10-11
ZA775784B (en) 1979-06-27
NO147913C (no) 1983-07-06
LU78179A1 (da) 1978-11-03
NL7710573A (nl) 1978-03-31
DE2643753A1 (de) 1978-04-06
IE45700B1 (en) 1982-11-03
US4224322A (en) 1980-09-23

Similar Documents

Publication Publication Date Title
DK508077A (da) Hidtil ukendte spirolactoner og fremgangsmaade til fremstilling deraf
DK228878A (da) Pyrimidinderivater og fremgangsmaade til fremstilling deraf
DK117377A (da) Provemiddel, proveudstyr og provemetode
NZ182756A (en) 2-or3-amino-c-substituted-imidazo(1,2-a) pyridines
DK489477A (da) Pyrimido(6,1-a)isoquinolin-2-on-derivater og fremgangsmaade til fremstilling deraf
DK336878A (da) Prostaglandin-12-derivater og fremgangsmaade til fremstilling heraf
DK478677A (da) Aminoglycosidderivater og fremgangsmaade til fremstilling deraf
DK355776A (da) 4-chromanoner og fremgangsmade til disses fremstilling
DK526976A (da) Picolinsyrerivater og fremgangsmade til fremstilling heraf
DK546776A (da) Quinazolinderivater og fremgangsmade til fremstilling deraf
DK307577A (da) 5-aroyl-1,2-dihydro-3h-pyrrol (1,2-a) pyrrol-1-carboxylsyrederivater og fremgangsmade til fremstilling deraf
PT67091A (de) Neue 1h-pyrazolo(3,4-b)pyridine
NO773892L (no) Antracyklinderivater og fremgangsmaate til fremstilling derav
DK4278A (da) 4-substituerede imidazo(1,2-a)quinoxaliner og mellemproduktersamt fremgangsmaade til fremstilling deraf
DK84077A (da) Aminoalkylpyrrolbenzoxazalkaner og fremgangsmade til fremstilling deraf
DK281377A (da) Joderede isophthalamsyrederivater og fremgangsmade til fremstilling deraf
DK213176A (da) Antraquinon-bis-amidiner og fremgangsmade til fremstilling deraf
DK402776A (da) 1,2-benzisoxazolderivater og fremgangsmade til fremstilling deraf
DK297477A (da) 5-o-acylerede imidazol-4-carboxamidderivater og fremgangsmade til fremstilling deraf
DK110476A (da) 13,14-dehydro-11-deoxy-prostaglandiner og fremgangsmade til fremstilling deraf
DK228677A (da) 3,5,5-trimethylhexanoyl-ferrocen og fremgangsmade til fremstilling deraf
DK568078A (da) Thieno (2,3-c) pyridinderivater og fremgangsmaade til fremstilling deraf
DK207679A (da) Tetrahydrothiopyrano (2,3-b) indol-derivater og fremgangsmaade til fremstilling deraf
DK306776A (da) 2-benzopyranonderivater og fremgangsmade til fremstilling derag
DK168576A (da) Spunsvaeg,samt fremgangsmaade og apparat til fremstilling heraf