DK3672976T3 - Bcl-2-hæmmere - Google Patents

Bcl-2-hæmmere Download PDF

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Publication number
DK3672976T3
DK3672976T3 DK18765259.9T DK18765259T DK3672976T3 DK 3672976 T3 DK3672976 T3 DK 3672976T3 DK 18765259 T DK18765259 T DK 18765259T DK 3672976 T3 DK3672976 T3 DK 3672976T3
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Prior art keywords
bcl
inhibitors
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DK18765259.9T
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English (en)
Inventor
Yi Chen
Yan Lou
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Guangzhou Lupeng Pharmaceutical Company Ltd
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Publication of DK3672976T3 publication Critical patent/DK3672976T3/da

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D498/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/12Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
    • C07D498/14Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/53751,4-Oxazines, e.g. morpholine
    • A61K31/53831,4-Oxazines, e.g. morpholine ortho- or peri-condensed with heterocyclic ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • A61K31/542Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame ortho- or peri-condensed with heterocyclic ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/02Antineoplastic agents specific for leukemia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/04Antineoplastic agents specific for metastasis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D513/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/12Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains three hetero rings
    • C07D513/14Ortho-condensed systems
    • GPHYSICS
    • G01MEASURING; TESTING
    • G01NINVESTIGATING OR ANALYSING MATERIALS BY DETERMINING THEIR CHEMICAL OR PHYSICAL PROPERTIES
    • G01N21/00Investigating or analysing materials by the use of optical means, i.e. using sub-millimetre waves, infrared, visible or ultraviolet light
    • G01N21/75Systems in which material is subjected to a chemical reaction, the progress or the result of the reaction being investigated
    • G01N21/76Chemiluminescence; Bioluminescence
    • G01N21/763Bioluminescence

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Immunology (AREA)
  • Oncology (AREA)
  • Hematology (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Diabetes (AREA)
  • Physics & Mathematics (AREA)
  • Plasma & Fusion (AREA)
  • Obesity (AREA)
  • Psychiatry (AREA)
  • Endocrinology (AREA)
  • Emergency Medicine (AREA)
  • Analytical Chemistry (AREA)
  • Biochemistry (AREA)
  • General Physics & Mathematics (AREA)
  • Pathology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
DK18765259.9T 2017-08-23 2018-08-22 Bcl-2-hæmmere DK3672976T3 (da)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201762549081P 2017-08-23 2017-08-23
US201862615007P 2018-01-09 2018-01-09
PCT/US2018/047444 WO2019040573A1 (en) 2017-08-23 2018-08-22 Bcl-2 inhibitors

Publications (1)

Publication Number Publication Date
DK3672976T3 true DK3672976T3 (da) 2024-03-04

Family

ID=63490700

Family Applications (2)

Application Number Title Priority Date Filing Date
DK18765259.9T DK3672976T3 (da) 2017-08-23 2018-08-22 Bcl-2-hæmmere
DK18765254.0T DK3672975T3 (da) 2017-08-23 2018-08-22 Kondenserede, heterocykliske derivater som bcl-2-hæmmere til behandling af neoplastiske sygdomme

Family Applications After (1)

Application Number Title Priority Date Filing Date
DK18765254.0T DK3672975T3 (da) 2017-08-23 2018-08-22 Kondenserede, heterocykliske derivater som bcl-2-hæmmere til behandling af neoplastiske sygdomme

Country Status (15)

Country Link
US (7) US11365206B2 (da)
EP (3) EP3672975B1 (da)
JP (2) JP7467331B2 (da)
KR (2) KR102680163B1 (da)
CN (4) CN116425771A (da)
AU (2) AU2018321496B2 (da)
CA (2) CA3073446A1 (da)
DK (2) DK3672976T3 (da)
ES (2) ES2948287T3 (da)
FI (2) FI3672975T3 (da)
IL (1) IL272762B2 (da)
MX (2) MX2020002033A (da)
SG (1) SG11202001553UA (da)
WO (2) WO2019040573A1 (da)
ZA (1) ZA202001301B (da)

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MX2020002033A (es) 2017-08-23 2020-08-20 Guangzhou Lupeng Pharmaceutical Company Ltd Derivados heterociclicos condensados como inhibidores de bcl-2 para el tratamiento de enfermedades neoplasticas.
MX2020011495A (es) 2018-04-29 2021-01-15 Beigene Ltd Inhibidores de bcl-2.
WO2020041405A1 (en) 2018-08-22 2020-02-27 Newave Pharmaceutical Inc. Bcl-2 inhibitors
WO2020140005A2 (en) 2018-12-29 2020-07-02 Newave Pharmaceutical Inc. Bcl-2 inhibitors
US20220372042A1 (en) * 2019-10-03 2022-11-24 Newave Pharmaceutical Inc. Condensed heterocycles as bcl-2 inhibitors
WO2021083135A1 (en) * 2019-10-28 2021-05-06 Beigene, Ltd. Bcl-2 INHIBITORS
WO2021133817A1 (en) 2019-12-27 2021-07-01 Guangzhou Lupeng Pharmaceutical Company Ltd. 1h-pyrrolo[2,3-b]pyridine derivatives as bcl-2 inhibitors for the treatment of neoplastic and autoimmune diseases
US12552784B2 (en) 2019-12-27 2026-02-17 Newave Pharmaceutical Inc. 1H-pyrrolo[2,3-b]pyridine derivatives as BCL-2 inhibitors for the treatment of neoplastic and autoimmune diseases
CN115484933A (zh) * 2020-02-24 2022-12-16 广州麓鹏制药有限公司 含有bcl2抑制剂的热熔挤出固体分散体
KR20230002419A (ko) 2020-04-15 2023-01-05 베이진 엘티디 Bcl-2 억제제
US20240166646A1 (en) 2020-12-22 2024-05-23 Newave Pharmaceutical Inc. 1h-pyrrolo[2,3-b]pyridine derivatives as bcl-2 inhibitors for the treatment of neoplastic and autoimmune diseases
CN113694059B (zh) * 2021-03-24 2023-09-26 浙江大学 Nl101在制备治疗急性、慢性排斥反应药物中的应用
WO2023122000A1 (en) * 2021-12-20 2023-06-29 Newave Pharmaceutical Inc. Bcl-2 inhibitors
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US11964990B2 (en) 2022-01-21 2024-04-23 Abbvie Inc. 1,3,4,7-tetrahydro-2H-pyrrolo[3′,2′:5,6]pyrido[2,3-b][1,4]oxazepine bcl-2 inhibitors
CN116236583A (zh) * 2023-03-30 2023-06-09 广州麓鹏制药有限公司 一种含Bcl-2/Bcl-xl抑制剂的组合物及其制备方法与应用
CN116270660A (zh) * 2023-03-30 2023-06-23 广州麓鹏制药有限公司 一种含Bcl-2/Bcl-xl抑制剂的组合物及其制备方法与应用

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WO2020041405A1 (en) 2018-08-22 2020-02-27 Newave Pharmaceutical Inc. Bcl-2 inhibitors
US20220372042A1 (en) 2019-10-03 2022-11-24 Newave Pharmaceutical Inc. Condensed heterocycles as bcl-2 inhibitors
US12552784B2 (en) 2019-12-27 2026-02-17 Newave Pharmaceutical Inc. 1H-pyrrolo[2,3-b]pyridine derivatives as BCL-2 inhibitors for the treatment of neoplastic and autoimmune diseases

Also Published As

Publication number Publication date
JP2020531506A (ja) 2020-11-05
US20250179090A1 (en) 2025-06-05
EP4227311A1 (en) 2023-08-16
JP7467331B2 (ja) 2024-04-15
KR102705861B1 (ko) 2024-09-10
MX2020002033A (es) 2020-08-20
IL272762B1 (en) 2023-11-01
CA3073446A1 (en) 2019-02-28
US11993610B2 (en) 2024-05-28
US20240425520A1 (en) 2024-12-26
ZA202001301B (en) 2025-04-30
CN116425771A (zh) 2023-07-14
ES2948287T3 (es) 2023-09-07
US11680072B2 (en) 2023-06-20
US20200190109A1 (en) 2020-06-18
KR20200090738A (ko) 2020-07-29
US20200197406A1 (en) 2020-06-25
CN111511748A (zh) 2020-08-07
JP2020531501A (ja) 2020-11-05
US20220402941A1 (en) 2022-12-22
MX2020002032A (es) 2020-09-17
EP3672976A1 (en) 2020-07-01
ES2971457T3 (es) 2024-06-05
US20220220126A1 (en) 2022-07-14
AU2018322059A1 (en) 2020-04-02
AU2018321496A1 (en) 2020-04-02
IL272762A (en) 2020-04-30
AU2018321496B2 (en) 2023-11-02
CN111448198B (zh) 2023-02-03
CA3073445A1 (en) 2019-02-28
SG11202001553UA (en) 2020-03-30
US12410190B2 (en) 2025-09-09
JP7467332B2 (ja) 2024-04-15
WO2019040550A1 (en) 2019-02-28
AU2018322059C1 (en) 2024-09-12
KR20200092308A (ko) 2020-08-03
US20230271979A1 (en) 2023-08-31
EP3672975B1 (en) 2023-04-12
WO2019040573A1 (en) 2019-02-28
DK3672975T3 (da) 2023-07-24
IL272762B2 (en) 2024-03-01
US11365206B2 (en) 2022-06-21
CN111448198A (zh) 2020-07-24
KR102680163B1 (ko) 2024-06-28
US11279711B2 (en) 2022-03-22
EP3672976B1 (en) 2023-12-13
FI3672976T3 (fi) 2024-02-21
CN116621860A (zh) 2023-08-22
FI3672975T3 (fi) 2023-06-28
CN111511748B (zh) 2023-05-02
AU2018322059B2 (en) 2023-11-02
EP3672975A1 (en) 2020-07-01

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