DK340987A - Tricykliske forbindelser, som er agonister af cholinerge receptorer, fremgangsmaade til fremstilling deraf, samt laegemidler indeholdende disse - Google Patents

Tricykliske forbindelser, som er agonister af cholinerge receptorer, fremgangsmaade til fremstilling deraf, samt laegemidler indeholdende disse

Info

Publication number
DK340987A
DK340987A DK340987A DK340987A DK340987A DK 340987 A DK340987 A DK 340987A DK 340987 A DK340987 A DK 340987A DK 340987 A DK340987 A DK 340987A DK 340987 A DK340987 A DK 340987A
Authority
DK
Denmark
Prior art keywords
cholinerge
tricyclic
agonists
relations
receptors
Prior art date
Application number
DK340987A
Other languages
English (en)
Other versions
DK162220C (da
DK340987D0 (da
DK162220B (da
Inventor
Kathleen Biziere
Camille Georges Wermuth
Paul Worms
Jean-Jacques Bourguignon
Original Assignee
Sanofi Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Sa filed Critical Sanofi Sa
Publication of DK340987D0 publication Critical patent/DK340987D0/da
Publication of DK340987A publication Critical patent/DK340987A/da
Publication of DK162220B publication Critical patent/DK162220B/da
Application granted granted Critical
Publication of DK162220C publication Critical patent/DK162220C/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D237/00Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings
    • C07D237/26Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings condensed with carbocyclic rings or ring systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D237/00Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings
    • C07D237/26Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings condensed with carbocyclic rings or ring systems
    • C07D237/36Benzo-cinnolines
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Neurosurgery (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Hospice & Palliative Care (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Psychiatry (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
DK340987A 1986-07-03 1987-07-02 Tricykliske pyridazinderivater, som er agonister af cholinerge receptorer, fremgangsmaade til fremstilling af derivaterne, og laegemidler, hvori de er til stede DK162220C (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR8609681 1986-07-03
FR8609681A FR2601011B1 (fr) 1986-07-03 1986-07-03 Nouveaux derives tricycliques agonistes des recepteurs cholinergiques et medicaments en contenant

Publications (4)

Publication Number Publication Date
DK340987D0 DK340987D0 (da) 1987-07-02
DK340987A true DK340987A (da) 1988-01-04
DK162220B DK162220B (da) 1991-09-30
DK162220C DK162220C (da) 1992-03-02

Family

ID=9337042

Family Applications (1)

Application Number Title Priority Date Filing Date
DK340987A DK162220C (da) 1986-07-03 1987-07-02 Tricykliske pyridazinderivater, som er agonister af cholinerge receptorer, fremgangsmaade til fremstilling af derivaterne, og laegemidler, hvori de er til stede

Country Status (16)

Country Link
US (1) US4977152A (da)
EP (1) EP0251937B1 (da)
JP (1) JPH029866A (da)
KR (1) KR880001614A (da)
AR (1) AR245123A1 (da)
AT (1) ATE60589T1 (da)
AU (1) AU602339B2 (da)
CA (1) CA1312864C (da)
DE (1) DE3767794D1 (da)
DK (1) DK162220C (da)
ES (1) ES2039256T3 (da)
FR (1) FR2601011B1 (da)
GR (1) GR3001646T3 (da)
NZ (1) NZ220926A (da)
PT (1) PT85234B (da)
ZA (1) ZA874846B (da)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2625201B1 (fr) * 1987-12-24 1990-06-15 Sanofi Sa Nouveaux derives tricycliques agonistes des recepteurs cholinergiques et medicaments en contenant
US4985560A (en) * 1990-01-12 1991-01-15 American Home Products Corporation Pyridazino(4,5-b)indolizines
US20100210590A1 (en) * 1995-09-27 2010-08-19 Northwestern University Compositions and treatments for seizure-related disorders
US20030176437A1 (en) * 2001-08-31 2003-09-18 D.M. Watterson Anti-inflammatory and protein kinase inhibitor compositions and related methods for downregulation of detrimental cellular responses and inhibition of cell death
KR100422589B1 (ko) * 2001-11-20 2004-03-16 (주)경인양행 셀룰로오스 섬유 또는 셀룰로오스 혼방섬유의 염색 방법
ES2441718T3 (es) 2004-11-02 2014-02-06 Northwestern University Compuestos de piridazina, composiciones y métodos
WO2006050359A2 (en) * 2004-11-02 2006-05-11 Northwestern University Pyridazine compounds and methods
CN101754762A (zh) 2006-04-28 2010-06-23 西北大学 用于治疗神经炎症性疾病的包含哒嗪化合物的制剂
US20100168120A1 (en) * 2006-04-28 2010-07-01 Neuromedix Inc. Salts of pyridazine compounds
EP2015750A2 (en) * 2006-04-28 2009-01-21 Northwestern University Compositions and treatments using pyridazine compounds and cholinesterase inhibitors
JP2011509261A (ja) * 2008-01-07 2011-03-24 シンタ ファーマシューティカルズ コーポレーション 炎症および免疫関連用途向けの化合物

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2510997A1 (fr) * 1981-08-10 1983-02-11 Sanofi Sa Nouveaux derives de la methyl-4 phenyl-6 pyridazine, procede pour leur preparation et medicaments actifs sur le systeme nerveux central en contenant
FR2619818B1 (fr) * 1987-09-01 1990-01-12 Sanofi Sa Imidazo (1,2-b) pyridazines, procede pour leur preparation et compositions pharmaceutiques les contenant

Also Published As

Publication number Publication date
AU7504987A (en) 1988-01-07
NZ220926A (en) 1989-11-28
AU602339B2 (en) 1990-10-11
AR245123A1 (es) 1993-12-30
KR880001614A (ko) 1988-04-25
DK162220C (da) 1992-03-02
ES2039256T3 (es) 1993-09-16
DK340987D0 (da) 1987-07-02
FR2601011B1 (fr) 1988-10-28
DK162220B (da) 1991-09-30
US4977152A (en) 1990-12-11
EP0251937A1 (fr) 1988-01-07
PT85234B (pt) 1990-04-30
GR3001646T3 (en) 1992-11-23
ZA874846B (en) 1988-03-30
JPH029866A (ja) 1990-01-12
DE3767794D1 (de) 1991-03-07
FR2601011A1 (fr) 1988-01-08
CA1312864C (en) 1993-01-19
EP0251937B1 (fr) 1991-01-30
ATE60589T1 (de) 1991-02-15
PT85234A (fr) 1987-08-01

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