DK328579A - Alkylderivater af c-076 forbindelser og fremgangsmaade til fremstilling deraf - Google Patents

Alkylderivater af c-076 forbindelser og fremgangsmaade til fremstilling deraf

Info

Publication number
DK328579A
DK328579A DK328579A DK328579A DK328579A DK 328579 A DK328579 A DK 328579A DK 328579 A DK328579 A DK 328579A DK 328579 A DK328579 A DK 328579A DK 328579 A DK328579 A DK 328579A
Authority
DK
Denmark
Prior art keywords
carbon atoms
hydrocarbon
substituted
alkyl
phenyl
Prior art date
Application number
DK328579A
Other languages
English (en)
Inventor
M H Fisher
A Lusi
R L Tolman
Original Assignee
Merck & Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck & Co Inc filed Critical Merck & Co Inc
Publication of DK328579A publication Critical patent/DK328579A/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/01—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing oxygen
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Molecular Biology (AREA)
  • Veterinary Medicine (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Biochemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Saccharide Compounds (AREA)
DK328579A 1978-08-04 1979-08-03 Alkylderivater af c-076 forbindelser og fremgangsmaade til fremstilling deraf DK328579A (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US05/930,845 US4200581A (en) 1978-08-04 1978-08-04 Alkyl derivatives of C-076 compounds

Publications (1)

Publication Number Publication Date
DK328579A true DK328579A (da) 1980-02-05

Family

ID=25459864

Family Applications (1)

Application Number Title Priority Date Filing Date
DK328579A DK328579A (da) 1978-08-04 1979-08-03 Alkylderivater af c-076 forbindelser og fremgangsmaade til fremstilling deraf

Country Status (10)

Country Link
US (1) US4200581A (da)
EP (1) EP0008184B1 (da)
JP (1) JPS5524165A (da)
AT (1) ATE7300T1 (da)
AU (1) AU526571B2 (da)
DE (1) DE2966954D1 (da)
DK (1) DK328579A (da)
IE (1) IE48913B1 (da)
NZ (1) NZ191088A (da)
ZA (1) ZA793993B (da)

Families Citing this family (50)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5296011A (en) * 1976-02-06 1977-08-12 Nippon Telegr & Teleph Corp <Ntt> Production of magnetic head
JPS52130316A (en) * 1976-04-26 1977-11-01 Nippon Telegr & Teleph Corp <Ntt> Production of magnetic heads
US4289760A (en) * 1980-05-02 1981-09-15 Merck & Co., Inc. 23-Keto derivatives of C-076 compounds
US4389397A (en) * 1980-08-04 1983-06-21 Merck & Co., Inc. Solubilization of ivermectin in water
US4285963A (en) * 1980-08-07 1981-08-25 Merck & Co., Inc. Novel derivatives of C-076 compounds
US4378353A (en) * 1981-02-17 1983-03-29 Merck & Co., Inc. Novel C-076 compounds
US4333925A (en) * 1981-05-11 1982-06-08 Merck & Co., Inc. Derivatives of C-076 compounds
US4399274A (en) * 1981-07-02 1983-08-16 Merck & Co., Inc. Isolation of non-ionic lipophilic materials on macroreticular polymeric absorbents
US4408059A (en) * 1981-12-04 1983-10-04 University Patents, Inc. Spiroketals useful as intermediates in the synthesis of milbemycin and avermectin macrolides
US4427663A (en) * 1982-03-16 1984-01-24 Merck & Co., Inc. 4"-Keto-and 4"-amino-4"-deoxy avermectin compounds and substituted amino derivatives thereof
US4469682A (en) * 1983-01-28 1984-09-04 Merck & Co., Inc. Avermectin and milbemycin phosphate esters, pharmaceutical compositions, and method of use
US5169956A (en) * 1984-06-05 1992-12-08 American Cyanamid Company Macrolide antibiotic compounds
US5106994A (en) * 1984-06-05 1992-04-21 American Cyanamid Company Agents and method of production thereof
US5317030A (en) * 1984-06-05 1994-05-31 American Cyanamid Company Method and compositions for helmintic, arthropod ectoparasitic and acaridal infections with novel agents
US5198464A (en) * 1984-06-05 1993-03-30 American Cyanamid Company Method and compositions for helmintic, arthropod ectoparasitic and acaridal infections with novel agents
US4547491A (en) * 1984-07-18 1985-10-15 Merck & Co., Inc. C-8A-Oxo-avermectin and milbemycin derivatives, pharmaceutical compositions and method of use
BE903232A (fr) * 1984-09-14 1986-03-13 Glaxo Group Ltd Composes antibiotiques et leur procede de preparation
HUT39739A (en) * 1984-12-04 1986-10-29 Ciba Geigy Ag Process for production of derivatives of 13,3-milbemycin and medical preparatives containing thereof
GB2168345B (en) * 1984-12-14 1988-05-25 Ciba Geigy Ag Pesticidal 13b-substituted milbemycin derivatives
US4587247A (en) * 1985-02-25 1986-05-06 Merck & Co., Inc. Substituted and unsubstituted 13-(alkoxy)methoxy derivatives of the avermectin aglycones, compositions and use
ES8800986A1 (es) * 1985-07-27 1987-12-01 Pfizer Un procedimiento para la produccion de un nuevo derivado de avermectina
JPH0678342B2 (ja) * 1986-01-07 1994-10-05 三共株式会社 新規マクロライド化合物
EP0239528A1 (de) * 1986-03-05 1987-09-30 Ciba-Geigy Ag 13Beta-Carbamoyloxy-milbemycinderivate zur Bekämpfung von tier- und pflanzenparasitären Schädlingen
EP0246739B1 (en) * 1986-03-25 1991-01-23 Sankyo Company Limited Macrolide compounds, their preparation and their use
EP0245209A1 (de) * 1986-05-07 1987-11-11 Ciba-Geigy Ag Milbemycin-Derivate, ihre Herstellung und ihre Verwendung zur Bekämpfung von Schädlingen
EP0252879B1 (de) * 1986-07-02 1992-05-06 Ciba-Geigy Ag Pestizide
US5840704A (en) * 1986-07-16 1998-11-24 Pfizer Inc. Antiparasitic agents and process for their preparation
US4897416A (en) * 1987-02-18 1990-01-30 Ciba-Geigy Corporation Insecticides and parasiticides
ATE87926T1 (de) * 1987-11-09 1993-04-15 Pfizer Ethylierte avermectine.
GB8726730D0 (en) * 1987-11-14 1987-12-16 Pfizer Ltd Antiparasitic agents
US4895837A (en) * 1988-01-29 1990-01-23 Merck & Co., Inc. Avermectin derivatives
GB8804440D0 (en) * 1988-02-25 1988-03-23 Pfizer Ltd Antiparasitic agents
US4918097A (en) * 1988-03-11 1990-04-17 Ciba-Geigy Corporation Insecticides and parasiticides
US5428034A (en) * 1988-09-02 1995-06-27 Sankyo Co., Ltd. Milbemycin derivatives, their preparation and their use
NZ232422A (en) * 1989-02-16 1992-11-25 Merck & Co Inc 13-ketal milbemycin derivatives and parasiticides
JP2622197B2 (ja) * 1990-03-01 1997-06-18 三共株式会社 １３−エーテル置換ミルベマイシン誘導体
US5188944A (en) * 1990-06-22 1993-02-23 Merck & Co., Inc. Process for the glycosylation of avermectin agylcones
US5171742A (en) * 1991-10-15 1992-12-15 Merck & Co., Inc. Avermectin compounds with a 6,5-spiroketal ring system ad a 23-acyl substituent
US5240915A (en) * 1991-10-15 1993-08-31 Merck & Co., Inc. Avermectin derivatives
GB9201505D0 (en) * 1992-01-24 1992-03-11 Pfizer Ltd Antiparasitic agents
US5162363A (en) * 1992-03-18 1992-11-10 Merck & Co., Inc. 23-nor-23-thia avermectin analogs are active anthelmintic agents
US5229415A (en) * 1992-03-24 1993-07-20 Merck & Co., Inc. Alkylthio alkyl avermectins are active antiparasitic agents
US6103504A (en) * 1992-03-25 2000-08-15 Pfizer Inc. Process for production of avermectins and cultures therefor
EP0670067B1 (en) * 1992-11-20 1997-05-07 Btg International Limited Image reconstruction
RU2226531C1 (ru) 2000-04-27 2004-04-10 Санкио Компани, Лимитед 13-замещенные производные милбемицина, их получение и их применение против насекомых и других вредителей
AU2001278694A1 (en) * 2000-08-09 2002-02-18 The Kitasato Institute Avermectin derivatives
AU2001277712A1 (en) * 2000-08-09 2002-02-18 The Kitasato Institute Avermectin derivatives
US20060205681A1 (en) * 2002-06-21 2006-09-14 Maryam Moaddeb Homogenous paste formulations
US7001889B2 (en) * 2002-06-21 2006-02-21 Merial Limited Anthelmintic oral homogeneous veterinary pastes
US20080027011A1 (en) * 2005-12-20 2008-01-31 Hassan Nached Homogeneous paste and gel formulations

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2173778A1 (en) * 1972-03-02 1973-10-12 Aries Robert 5-phenoxyalkyltetrazoles - hypocholesterolaemics and anorectics
US3950360A (en) * 1972-06-08 1976-04-13 Sankyo Company Limited Antibiotic substances
SE434277B (sv) * 1976-04-19 1984-07-16 Merck & Co Inc Sett att framstella nya antihelmintiskt verkande foreningar genom odling av streptomyces avermitilis
NZ186851A (en) * 1977-04-11 1984-12-14 Merck & Co Inc Glycosyloxy derivatives of milbemycin and parasiticidal compositions
US4093629A (en) * 1977-04-11 1978-06-06 Merck & Co., Inc. Derivatives of antibiotic substance milbemycin and processes therefor
NZ188459A (en) * 1977-10-03 1982-09-07 Merck & Co Inc Derivatives of c-076 compounds and pesticidal compositions
PH15982A (en) * 1977-10-03 1983-05-18 Merck & Co Inc Selective hydrogenation producta of c-076 compounds and derivatives thereof
JPS6254113A (ja) * 1985-09-03 1987-03-09 Fuji Electric Co Ltd 管内スケ−ル厚さの測定方法

Also Published As

Publication number Publication date
DE2966954D1 (en) 1984-06-07
ATE7300T1 (de) 1984-05-15
AU526571B2 (en) 1983-01-20
EP0008184B1 (en) 1984-05-02
EP0008184A1 (en) 1980-02-20
AU4923379A (en) 1980-02-07
IE48913B1 (en) 1985-06-12
IE791437L (en) 1980-02-04
US4200581A (en) 1980-04-29
JPH0238596B2 (da) 1990-08-31
ZA793993B (en) 1981-03-25
NZ191088A (en) 1984-09-28
JPS5524165A (en) 1980-02-21

Similar Documents

Publication Publication Date Title
DK328579A (da) Alkylderivater af c-076 forbindelser og fremgangsmaade til fremstilling deraf
DE2965370D1 (en) Sugar derivatives of c-076 compounds, their preparation and their use as antiparasitic agents
IE781964L (en) Derivatives of c-076 compounds
SE8106125L (sv) 4,5-polymetylen-4-isotiazolin-3-oner, sett for framstellning derav och anvendning derav som baktericida och fungicida medel
FI914187A0 (fi) Menetelmä valmistaa kaavan /I/ mukaista 1-metyylikarbapeneemijohdosta
KR910002800A (ko) 4-아실록시퀴놀린 유도체와 이를 함유하는 살충 또는 살비조성물
KR840004082A (ko) 피리다지는 유도체와 그의 제조방법, 그리고 상기의 유도체를 함유하는 농업 및 원예용 살균, 살충, 진드기구충 석충박멸 조성물
KR900016178A (ko) 2-치환 n,n&#39;-디트리메톡시벤조일 피페라진, 그의 제조 방법 및 그를 함유하는 치료 조성물
KR860007251A (ko) 트리아졸 유도체의 제조방법
DK462580A (da) R fremgangsmaade til fremstilling af 3-substituerede propenoate
ES8305730A1 (es) Un procedimiento para la preparacion de un derivado del imidazol.
DE3472104D1 (en) N-substituted ûbis(hydroxymethyl)-methyl¨-isoquinoline derivatives, process for preparing them and pharmaceutical compositions containing them
PT96003A (pt) Processo para a preparacao de composicoes farmaceuticas, contendo um derivado triazol
ES8502700A1 (es) Procedimiento para la fabricacion de derivados de tetrahidrobenzotiazol.
ES8403891A1 (es) Un procedimiento para la preparacion de un derivado del acido furiloxazolila-cetico
DK0391673T3 (da) Fremstilling af glutarsyrederivater
KR930007952A (ko) 살균제
JPS54157562A (en) Substituted nnalkylimidazole derivative*its manufacture and composition containing it
TH9884B (th) กรรมวิธีใหม่สำหรับผลิตอนุพันธ์ 13-อีเธอร์ของมิลบีไมซิน, และอินเทอร์มิเดียทชนิดใหม่ของสารดังกล่าว
EP0273357A3 (en) Fluorine-containing macrolide compounds, pharmaceutical compositions comprising the same and their use for the manufacture of medicaments
FI924639A (fi) Farmaceutiska kompositioner innehaollande triazolderivat foer rektal administration
KR830004222A (ko) 벤즈아닐리드(benzanilide) 또는 티오 벤즈아닐리드(thio benzanilide) 유도체의 제조방법 및 이것을 유효성분으로 함유하는 농원예용 살균조성물
KR970019857A (ko) 신규 티아졸에톡시퀴나졸린 유도체, 그의 제조방법 및 그를 유효성분으로 하는 식물 병원균 퇴치용 조성물
KR910015588A (ko) 치환에텐일기를 갖는 유기규소계 화합물 및 그의 제조방법

Legal Events

Date Code Title Description
ARF Application refused