DK3186257T3 - Hitherto UNKNOWN CHROMONOXIME DERIVATIVE AND ITS USE AS AN ALLOSTERIC MODULATOR OF METABOTROPIC GLUTAMATE RECEPTORS - Google Patents
Hitherto UNKNOWN CHROMONOXIME DERIVATIVE AND ITS USE AS AN ALLOSTERIC MODULATOR OF METABOTROPIC GLUTAMATE RECEPTORS Download PDFInfo
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- DK3186257T3 DK3186257T3 DK15770814.0T DK15770814T DK3186257T3 DK 3186257 T3 DK3186257 T3 DK 3186257T3 DK 15770814 T DK15770814 T DK 15770814T DK 3186257 T3 DK3186257 T3 DK 3186257T3
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Landscapes
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Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP14182468 | 2014-08-27 | ||
| PCT/EP2015/069601 WO2016030444A1 (en) | 2014-08-27 | 2015-08-27 | Novel chromone oxime derivative and its use as allosteric modulator of metabotropic glutamate receptors |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DK3186257T3 true DK3186257T3 (en) | 2019-04-01 |
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| DK15770814.0T DK3186257T3 (en) | 2014-08-27 | 2015-08-27 | Hitherto UNKNOWN CHROMONOXIME DERIVATIVE AND ITS USE AS AN ALLOSTERIC MODULATOR OF METABOTROPIC GLUTAMATE RECEPTORS |
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| EP (3) | EP3502115A1 (enExample) |
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| SMT201900152T1 (it) | 2014-08-27 | 2019-05-10 | Prexton Therapeutics Sa | Nuovo derivato di cromone ossima e suo uso come modulatore allosterico di recettori metabotropici del glutammato |
| AU2016313138A1 (en) * | 2015-08-27 | 2018-03-15 | Prexton Therapeutics Sa | Brain-penetrant chromone oxime derivative for the therapy of levodopa-induced dyskinesia |
| IL280213B2 (en) | 2018-07-26 | 2024-06-01 | Domain Therapeutics | Substituted quinazolinone derivatives and their use as positive allosteric modulators of mglur4 |
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| US4065467A (en) | 1973-12-27 | 1977-12-27 | Carlo Erba, S. P. A. | 5:6-Benzo δ-pyrone derivatives and process for their preparation |
| US4777252A (en) | 1987-08-13 | 1988-10-11 | E. R. Squibb & Sons, Inc. | 2-oxo-1-[[(substituted sulfonyl)amino]-carbonyl]azetidines |
| JP3993651B2 (ja) | 1994-10-21 | 2007-10-17 | アスビオファーマ株式会社 | シクロプロパクロメンカルボン酸誘導体 |
| EP1298129A3 (en) | 2001-09-28 | 2003-06-04 | Central Glass Company, Limited | Process for producing 4-sustituted benzopyran derivatives |
| MY141521A (en) | 2002-12-12 | 2010-05-14 | Hoffmann La Roche | 5-substituted-six-membered heteroaromatic glucokinase activators |
| JP2006522124A (ja) | 2003-04-03 | 2006-09-28 | バーテックス ファーマシューティカルズ インコーポレイテッド | プロテインキナーゼのインヒビターとして有用な組成物 |
| WO2007011701A1 (en) | 2005-07-15 | 2007-01-25 | Transform Pharmaceuticals, Inc. | Novel hydrochloride salts of levodopa |
| WO2009010455A2 (en) | 2007-07-13 | 2009-01-22 | Addex Pharma S.A. | Pyrazole derivatives as modulators of metabotropic glutamate receptors |
| GB0713686D0 (en) | 2007-07-13 | 2007-08-22 | Addex Pharmaceuticals Sa | New compounds 2 |
| JP5806672B2 (ja) * | 2009-10-30 | 2015-11-10 | ドメイン・セラピューティクス | 新規オキシム誘導体及び代謝型グルタミン酸受容体のアロステリック調節因子としての利用 |
| KR102074089B1 (ko) * | 2009-12-04 | 2020-02-05 | 선오비온 파마슈티컬스 인코포레이티드 | 다환형 화합물 및 이의 사용 방법 |
| US20140349994A1 (en) * | 2012-01-18 | 2014-11-27 | Addex Pharma S.A. | Novel 2-Amino-4,5,6,8-Tetrahydropyrazolo[3,4-b]Thiazolo [4,5-d]Azepine Derivatives and Their Use as Allosteric Modulators of Metabotropic Glutamate Receptors |
| SMT201900152T1 (it) * | 2014-08-27 | 2019-05-10 | Prexton Therapeutics Sa | Nuovo derivato di cromone ossima e suo uso come modulatore allosterico di recettori metabotropici del glutammato |
| AU2016313138A1 (en) | 2015-08-27 | 2018-03-15 | Prexton Therapeutics Sa | Brain-penetrant chromone oxime derivative for the therapy of levodopa-induced dyskinesia |
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- 2015-08-27 PT PT15770814T patent/PT3186257T/pt unknown
- 2015-08-27 HR HRP20190343TT patent/HRP20190343T1/hr unknown
- 2015-08-27 CN CN201910567865.9A patent/CN110343118A/zh active Pending
- 2015-08-27 MX MX2017002429A patent/MX369643B/es active IP Right Grant
- 2015-08-27 WO PCT/EP2015/069601 patent/WO2016030444A1/en not_active Ceased
- 2015-08-27 JP JP2017530425A patent/JP6430015B2/ja not_active Expired - Fee Related
- 2015-08-27 EP EP15770814.0A patent/EP3186257B1/en active Active
- 2015-08-27 ES ES15770814T patent/ES2714073T3/es active Active
- 2015-08-27 LT LTEP15770814.0T patent/LT3186257T/lt unknown
- 2015-08-27 DK DK15770814.0T patent/DK3186257T3/en active
- 2015-08-27 MA MA040530A patent/MA40530A/fr unknown
- 2015-08-27 US US15/506,941 patent/US10017521B2/en not_active Expired - Fee Related
- 2015-08-27 EP EP19217991.9A patent/EP3696183A1/en not_active Withdrawn
- 2015-08-27 RU RU2017109818A patent/RU2672569C2/ru active
- 2015-08-27 AU AU2015308438A patent/AU2015308438B2/en not_active Ceased
- 2015-08-27 HU HUE15770814A patent/HUE041941T2/hu unknown
- 2015-08-27 SI SI201530640T patent/SI3186257T1/sl unknown
- 2015-08-27 MA MA052702A patent/MA52702A/fr unknown
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2017
- 2017-01-25 IL IL250287A patent/IL250287B/en active IP Right Grant
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2018
- 2018-06-05 US US16/000,338 patent/US10442818B2/en active Active
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2019
- 2019-03-08 CY CY20191100277T patent/CY1121352T1/el unknown
- 2019-09-30 US US16/587,670 patent/US20200024285A1/en not_active Abandoned
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