DK307184A - Aryl- og heteroaryl(7-(aryl- og heteroaryl)pyrazolo(1,5-a)pyrimidin-3-yl)methanoner - Google Patents

Aryl- og heteroaryl(7-(aryl- og heteroaryl)pyrazolo(1,5-a)pyrimidin-3-yl)methanoner Download PDF

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Publication number
DK307184A
DK307184A DK307184A DK307184A DK307184A DK 307184 A DK307184 A DK 307184A DK 307184 A DK307184 A DK 307184A DK 307184 A DK307184 A DK 307184A DK 307184 A DK307184 A DK 307184A
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Prior art keywords
heteroaryl
aryl
methanones
pyrazolo
pyrimidin
Prior art date
Application number
DK307184A
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English (en)
Other versions
DK307184D0 (da
Inventor
John Paul Dusza
Andrew Stephen Tomcufcik
Jay Donald Albright
Original Assignee
American Cyanamid Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by American Cyanamid Co filed Critical American Cyanamid Co
Publication of DK307184D0 publication Critical patent/DK307184D0/da
Publication of DK307184A publication Critical patent/DK307184A/da

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00—Drugs for disorders of the muscular or neuromuscular system
    • A61P21/02—Muscle relaxants, e.g. for tetanus or cramps
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Neurology (AREA)
  • Public Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Pain & Pain Management (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Anesthesiology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DK307184A 1983-06-23 1984-06-22 Aryl- og heteroaryl(7-(aryl- og heteroaryl)pyrazolo(1,5-a)pyrimidin-3-yl)methanoner DK307184A (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US50696683A 1983-06-23 1983-06-23

Publications (2)

Publication Number Publication Date
DK307184D0 DK307184D0 (da) 1984-06-22
DK307184A true DK307184A (da) 1984-12-24

Family

ID=24016730

Family Applications (1)

Application Number Title Priority Date Filing Date
DK307184A DK307184A (da) 1983-06-23 1984-06-22 Aryl- og heteroaryl(7-(aryl- og heteroaryl)pyrazolo(1,5-a)pyrimidin-3-yl)methanoner

Country Status (17)

Country Link
EP (1) EP0129847B1 (da)
JP (1) JPS6019788A (da)
KR (1) KR900001886B1 (da)
AT (1) ATE53391T1 (da)
AU (1) AU568656B2 (da)
CA (1) CA1233174A (da)
DD (1) DD228257A5 (da)
DE (2) DE3422844A1 (da)
DK (1) DK307184A (da)
ES (1) ES8505958A1 (da)
HK (1) HK91592A (da)
HU (1) HUT37620A (da)
IE (1) IE58012B1 (da)
IL (1) IL72208A (da)
NZ (1) NZ208554A (da)
PH (1) PH21523A (da)
ZA (1) ZA844776B (da)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4626538A (en) * 1983-06-23 1986-12-02 American Cyanamid Company [7-(3-disubstituted amino)phenyl]pyrazolo[1,5-a]pyrimidines
DE19975048I2 (de) * 1985-05-13 2001-06-13 American Cyanamid Co 7-(3-Disubstituierte Amino)phenyl pyrazolo 1,5-a -pyrimidine
JPS61223072A (ja) * 1986-02-21 1986-10-03 Canon Inc インクジエツト記録方法
US4847256A (en) * 1986-10-16 1989-07-11 American Cyanamid Company 4,5-dihydro and 4,5,6,7-tetrahydropyrazolo(1,5-A)-pyrimidines
EP0264773A1 (en) * 1986-10-16 1988-04-27 American Cyanamid Company 4,5-dihydro and 4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidines
FI864570A0 (fi) * 1986-11-11 1986-11-11 Farmos Oy Terapeutiskt anvaendbar foerening.
US5714607A (en) * 1995-12-01 1998-02-03 American Cyanamid Company Process improvement in the synthesis of N- 3-(3-cyano-pyrazolo 1,5-a!pyrimidin-7-yl)phenyl!-N-ethylacetamide
WO2000059908A2 (en) 1999-04-06 2000-10-12 Du Pont Pharmaceuticals Company Pyrazolopyrimidines as crf antagonists
US6472528B1 (en) * 1999-08-10 2002-10-29 Neurocrine Biosciences, Inc. Synthesis of substituted pyrazolopyrimidines
BR0014459A (pt) * 1999-09-02 2002-07-16 Neurocrine Biosciences Inc Polìmeros de n-metil-n- (3-{3-[2-tienilcarbonil]-pirazol-[1,5-"alfa"]-pirimidin-7-il } fenil) acetamida e composições e métodos relacionados aos mesmos
WO2004110454A1 (ja) * 2003-06-13 2004-12-23 Ishihara Sangyo Kaisha, Ltd. アデノシンＡ2ａ受容体アゴニストの投与が必要な疾患を治療又は予防するための組成物
ES2222814B1 (es) * 2003-07-24 2005-12-01 Ferrer Internacional, S.A. 3-nitro-pirazolo(1,5-a)pirimidinas 7-sustituidas y composiciones y metodos relacionados.
ES2222813B1 (es) * 2003-07-24 2005-12-16 Ferrer Internacional, S.A. N-(3-(3-sustituidas-pirazolo(1,5-a)pirimidin-7-il)-fenil)-sulfonamidas y composiciones y metodos relacionados.

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE792533A (fr) * 1971-12-09 1973-06-08 Int Chem & Nuclear Corp Nouvelles pyrazolo (1,5a) pyrimidines et leur procede de preparation
US4093617A (en) * 1974-11-12 1978-06-06 Icn Pharmaceuticals, Inc. 3,5,7-Trisubstituted pyrazolo[1,5-a]pyrimidines
US4178449A (en) * 1978-04-17 1979-12-11 American Cyanamid Company Pyrazolo[1,5-a]pyrimidines and imidazo-[1,5-a]pyrimidines
US4236005A (en) * 1979-07-02 1980-11-25 American Cyanamid Company Imidazo[1,5-a]pyrimidines
US4281000A (en) * 1979-07-09 1981-07-28 American Cyanamid Company Substituted pyrazolo (1,5-a)pyrimidines and their use as anxiolytic agents
ZA803591B (en) * 1979-07-09 1981-06-24 American Cyanamid Co Substituted pyrazolo(1,5-a)pyrimidines

Also Published As

Publication number Publication date
IE58012B1 (en) 1993-06-16
HK91592A (en) 1992-11-27
AU568656B2 (en) 1988-01-07
CA1233174A (en) 1988-02-23
JPH0531551B2 (da) 1993-05-12
NZ208554A (en) 1987-06-30
DE3422844A1 (de) 1985-01-17
IL72208A (en) 1987-11-30
ES533654A0 (es) 1985-07-01
EP0129847A2 (en) 1985-01-02
HUT37620A (en) 1986-01-23
PH21523A (en) 1987-11-16
ATE53391T1 (de) 1990-06-15
DE3482419D1 (de) 1990-07-12
ES8505958A1 (es) 1985-07-01
DK307184D0 (da) 1984-06-22
KR900001886B1 (ko) 1990-03-26
EP0129847B1 (en) 1990-06-06
JPS6019788A (ja) 1985-01-31
EP0129847A3 (en) 1987-05-20
KR850000443A (ko) 1985-02-27
IL72208A0 (en) 1984-10-31
ZA844776B (en) 1985-02-27
AU2977084A (en) 1985-01-03
IE841580L (en) 1984-12-23
DD228257A5 (de) 1985-10-09

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AHS Application shelved for other reasons than non-payment