DK283487D0 - Thiazolyl-2-yl-imidazo(1,2-a)pyrimidiner, deres fremstilling og brug - Google Patents

Thiazolyl-2-yl-imidazo(1,2-a)pyrimidiner, deres fremstilling og brug

Info

Publication number
DK283487D0
DK283487D0 DK283487A DK283487A DK283487D0 DK 283487 D0 DK283487 D0 DK 283487D0 DK 283487 A DK283487 A DK 283487A DK 283487 A DK283487 A DK 283487A DK 283487 D0 DK283487 D0 DK 283487D0
Authority
DK
Denmark
Prior art keywords
carbon atoms
alkyl
optionally substituted
pyrimidines
imidazo
Prior art date
Application number
DK283487A
Other languages
English (en)
Other versions
DK283487A (da
Inventor
Robert Michael John Deacon
Colin Robert Gardner
Roger John Gillespie
Wilfred Roger Tully
Original Assignee
Roussel Uclaf
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Roussel Uclaf filed Critical Roussel Uclaf
Publication of DK283487D0 publication Critical patent/DK283487D0/da
Publication of DK283487A publication Critical patent/DK283487A/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/26—Psychostimulants, e.g. nicotine, cocaine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Diabetes (AREA)
  • Psychiatry (AREA)
  • Anesthesiology (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Physical Water Treatments (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
DK283487A 1986-06-04 1987-06-03 Thiazolyl-2-yl-imidazo(1,2-a)pyrimidiner, deres fremstilling og brug DK283487A (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB868613591A GB8613591D0 (en) 1986-06-04 1986-06-04 Chemical compounds

Publications (2)

Publication Number Publication Date
DK283487D0 true DK283487D0 (da) 1987-06-03
DK283487A DK283487A (da) 1987-12-05

Family

ID=10598934

Family Applications (1)

Application Number Title Priority Date Filing Date
DK283487A DK283487A (da) 1986-06-04 1987-06-03 Thiazolyl-2-yl-imidazo(1,2-a)pyrimidiner, deres fremstilling og brug

Country Status (14)

Country Link
US (1) US4925846A (da)
EP (1) EP0248735B1 (da)
JP (1) JPS6366183A (da)
KR (1) KR880000436A (da)
AT (1) ATE53032T1 (da)
AU (1) AU594776B2 (da)
DE (1) DE3762860D1 (da)
DK (1) DK283487A (da)
ES (1) ES2014482B3 (da)
GB (2) GB8613591D0 (da)
GR (1) GR3000565T3 (da)
HU (1) HU197576B (da)
PT (1) PT85008B (da)
ZA (1) ZA873884B (da)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZA919797B (en) * 1990-12-13 1992-10-28 Smithkline Beecham Corp Bicyclo-5,6-dihydro-7h-pyrrolo-1,20-imidazol-7-ols and 7-ones
CA2502511A1 (en) * 2002-10-18 2004-05-29 Pfizer Products Inc. Cannabinoid receptor ligands and uses thereof
US7129239B2 (en) * 2002-10-28 2006-10-31 Pfizer Inc. Purine compounds and uses thereof
US7247628B2 (en) * 2002-12-12 2007-07-24 Pfizer, Inc. Cannabinoid receptor ligands and uses thereof
US7329658B2 (en) * 2003-02-06 2008-02-12 Pfizer Inc Cannabinoid receptor ligands and uses thereof
US7176210B2 (en) * 2003-02-10 2007-02-13 Pfizer Inc. Cannabinoid receptor ligands and uses thereof
US7268133B2 (en) * 2003-04-23 2007-09-11 Pfizer, Inc. Patent Department Cannabinoid receptor ligands and uses thereof
US7145012B2 (en) 2003-04-23 2006-12-05 Pfizer Inc. Cannabinoid receptor ligands and uses thereof
US7141669B2 (en) * 2003-04-23 2006-11-28 Pfizer Inc. Cannabiniod receptor ligands and uses thereof
US20040214856A1 (en) * 2003-04-23 2004-10-28 Pfizer Inc Cannabinoid receptor ligands and uses thereof
EP1622876A1 (en) * 2003-05-07 2006-02-08 Pfizer Products Inc. Cannabinoid receptor ligands and uses thereof
US7232823B2 (en) 2003-06-09 2007-06-19 Pfizer, Inc. Cannabinoid receptor ligands and uses thereof
US20040259887A1 (en) * 2003-06-18 2004-12-23 Pfizer Inc Cannabinoid receptor ligands and uses thereof
BR112019025049A2 (pt) 2017-05-31 2020-06-16 Chemocentryx, Inc. Anéis 6- 5 fundidos como inibidores de c5a
MX2020010390A (es) 2018-04-02 2021-01-15 Chemocentryx Inc Profarmacos de antagonistas de c5ar biciclicos fusionados.

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL69417A (en) * 1982-08-27 1987-12-20 Roussel Uclaf 2-acyl imidazo(1,2-a)pyrimidines,their preparation and pharmaceutical compositions containing them
US4649146A (en) * 1983-01-31 1987-03-10 Fujisawa Pharmaceutical Co., Ltd. Thiazole derivatives and pharmaceutical composition comprising the same
US4521422A (en) * 1983-06-23 1985-06-04 American Cyanamid Company Aryl and heteroaryl[7-(aryl and heteroaryl)pyrazolo[1,5-a]pyrimidin-3-yl]methanones
GB8432073D0 (en) * 1984-12-19 1985-01-30 Roussel Lab Ltd Chemical compounds

Also Published As

Publication number Publication date
DK283487A (da) 1987-12-05
AU7379187A (en) 1987-12-10
HU197576B (en) 1989-04-28
ZA873884B (en) 1988-07-27
GB8613591D0 (en) 1986-07-09
ATE53032T1 (de) 1990-06-15
AU594776B2 (en) 1990-03-15
KR880000436A (ko) 1988-03-25
GR3000565T3 (en) 1991-07-31
EP0248735B1 (fr) 1990-05-23
EP0248735A1 (fr) 1987-12-09
DE3762860D1 (de) 1990-06-28
US4925846A (en) 1990-05-15
ES2014482B3 (es) 1990-07-16
GB2191196B (en) 1990-03-28
HUT46917A (en) 1988-12-28
JPS6366183A (ja) 1988-03-24
GB2191196A (en) 1987-12-09
PT85008A (en) 1987-07-01
GB8713010D0 (en) 1987-07-08
PT85008B (pt) 1990-03-08

Similar Documents

Publication Publication Date Title
DK283487D0 (da) Thiazolyl-2-yl-imidazo(1,2-a)pyrimidiner, deres fremstilling og brug
NO149888C (no) Analogifremgangsmaate for fremstilling av terapeutisk aktive 2-substituerte-2`-hydroksyl-6,7-benzomorfaner og syreaddisjonssalter derav
NO883994D0 (no) Fremgangsmaate for fremstilling av terapeutisk aktive pyrimidinylaminer.
ES8306142A1 (es) "procedimiento para la preparacion de nuevas n-(4-indolil-piperidino-alcohil)-bencimidazolonas sustituidas".
SE8800638L (sv) Antihypercholesterolemic tetrazole compounds
DK0484223T3 (da) 3-cyclopropanamider, deres tautomere former og deres salte samt en fremgangsmåde til deres fremstilling, deres anvendelse som lægemidler og præparater med indhold deraf
AU554959B2 (en) Triazolo(4,3-a) quinazolin-5-ones
FI871637A (fi) Foerfarande foer framstaellning av 1,5-benzotiazepinderivat.
DE3474145D1 (en) Benzothiazolone derivatives, processes for preparation thereof and pharmaceutical compositions comprising the same
DE3666223D1 (en) Anticonvulsant agents
NO150436C (no) Analogifremgangsmaate for fremstilling av terapeutisk aktive 2-fenylamino-imidazolin-derivater
NO164352C (no) Analogifremgangsmaate for fremstilling av farmasoeytisk aktive, antivirale, substituerte isoksazolderivater.
ES500108A0 (es) Procedimiento para preparar nuevas benzotiopirano (2,3-c)pi-ridinas

Legal Events

Date Code Title Description
AHB Application shelved due to non-payment