DK2081937T3 - Triazolopyridazin-proteinkinasemodulatorer - Google Patents

Triazolopyridazin-proteinkinasemodulatorer

Info

Publication number
DK2081937T3
DK2081937T3 DK07854193.5T DK07854193T DK2081937T3 DK 2081937 T3 DK2081937 T3 DK 2081937T3 DK 07854193 T DK07854193 T DK 07854193T DK 2081937 T3 DK2081937 T3 DK 2081937T3
Authority
DK
Denmark
Prior art keywords
proteinkinasemodulatorer
triazolopyridazine
Prior art date
Application number
DK07854193.5T
Other languages
Danish (da)
English (en)
Inventor
Christopher Ronald Smith
Pierre-Yves Bounaud
Elizabeth Anne Jefferson
Patrick S Lee
Eduardo Torres
Original Assignee
Sgx Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sgx Pharmaceuticals Inc filed Critical Sgx Pharmaceuticals Inc
Application granted granted Critical
Publication of DK2081937T3 publication Critical patent/DK2081937T3/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
DK07854193.5T 2006-10-23 2007-10-18 Triazolopyridazin-proteinkinasemodulatorer DK2081937T3 (da)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US86255206P 2006-10-23 2006-10-23
US87138406P 2006-12-21 2006-12-21
US91375207P 2007-04-24 2007-04-24
US95283307P 2007-07-30 2007-07-30
PCT/US2007/081832 WO2008051805A2 (en) 2006-10-23 2007-10-18 Triazolo-pyridazine protein kinase modulators

Publications (1)

Publication Number Publication Date
DK2081937T3 true DK2081937T3 (da) 2012-10-01

Family

ID=39031065

Family Applications (1)

Application Number Title Priority Date Filing Date
DK07854193.5T DK2081937T3 (da) 2006-10-23 2007-10-18 Triazolopyridazin-proteinkinasemodulatorer

Country Status (16)

Country Link
US (1) US8071581B2 (OSRAM)
EP (1) EP2081937B1 (OSRAM)
JP (1) JP2010507577A (OSRAM)
KR (1) KR101083177B1 (OSRAM)
AU (1) AU2007309237B2 (OSRAM)
BR (1) BRPI0717317A2 (OSRAM)
CA (1) CA2667453A1 (OSRAM)
DK (1) DK2081937T3 (OSRAM)
EA (1) EA016527B1 (OSRAM)
ES (1) ES2393132T3 (OSRAM)
MX (1) MX2009004060A (OSRAM)
PE (1) PE20081256A1 (OSRAM)
PL (1) PL2081937T3 (OSRAM)
PT (1) PT2081937E (OSRAM)
TW (1) TW200833692A (OSRAM)
WO (1) WO2008051805A2 (OSRAM)

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KR20140144726A (ko) 2012-03-30 2014-12-19 리젠 파마슈티컬스 소시에떼 아노님 C-met 단백질 키나제의 조절제로서의 신규한 3,5-디치환-3h-이미다조[4,5-b]피리딘 및 3,5- 디치환 -3h-[1,2,3]트리아졸로[4,5-b] 피리딘 화합물
AU2013290444B2 (en) 2012-07-16 2018-04-26 Vertex Pharmaceuticals Incorporated Pharmaceutical compositions of (R)-1-(2,2-diflurorbenzo[d][1,3]dioxol-5-yl)-N-(1-(2,3-dihydroxypropyl)-6-fluoro-2-(1-hydroxy-2-methylpropan-2-yl)-1H-indol-5-yl) cyclopropanecarboxamide and administration thereof
CN103122000B (zh) * 2012-09-03 2013-12-25 中美冠科生物技术（太仓）有限公司 用作抗肿瘤药物的高选择性的c-Met激酶抑制剂
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Also Published As

Publication number Publication date
KR101083177B1 (ko) 2011-11-11
EA016527B1 (ru) 2012-05-30
EP2081937A2 (en) 2009-07-29
AU2007309237A1 (en) 2008-05-02
TW200833692A (en) 2008-08-16
WO2008051805A3 (en) 2008-07-10
US8071581B2 (en) 2011-12-06
KR20090069303A (ko) 2009-06-30
ES2393132T3 (es) 2012-12-18
BRPI0717317A2 (pt) 2013-10-22
WO2008051805A2 (en) 2008-05-02
EP2081937B1 (en) 2012-09-12
US20100120739A1 (en) 2010-05-13
EA200970402A1 (ru) 2009-10-30
JP2010507577A (ja) 2010-03-11
CA2667453A1 (en) 2008-05-02
MX2009004060A (es) 2009-06-19
AU2007309237B2 (en) 2012-03-22
PE20081256A1 (es) 2008-10-13
PL2081937T3 (pl) 2013-01-31
PT2081937E (pt) 2012-10-15

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