DK170024B1 - Imidazo(2,1-b)thiazolderivater, deres fremstilling, mellemprodukter til anvendelse i forbindelse hermed, deres anvendelse som lægemidler samt farmaceutiske præparater med indhold heraf - Google Patents

Imidazo(2,1-b)thiazolderivater, deres fremstilling, mellemprodukter til anvendelse i forbindelse hermed, deres anvendelse som lægemidler samt farmaceutiske præparater med indhold heraf Download PDF

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Publication number
DK170024B1
DK170024B1 DK579688A DK579688A DK170024B1 DK 170024 B1 DK170024 B1 DK 170024B1 DK 579688 A DK579688 A DK 579688A DK 579688 A DK579688 A DK 579688A DK 170024 B1 DK170024 B1 DK 170024B1
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DK
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Prior art keywords
formula
compound
imidazo
group
hydrogen atom
Prior art date
Application number
DK579688A
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Danish (da)
English (en)
Other versions
DK579688A (da
DK579688D0 (da
Inventor
Charles John Robert Hedgecock
David Paul Kay
Original Assignee
Roussel Uclaf
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Roussel Uclaf filed Critical Roussel Uclaf
Publication of DK579688D0 publication Critical patent/DK579688D0/da
Publication of DK579688A publication Critical patent/DK579688A/da
Application granted granted Critical
Publication of DK170024B1 publication Critical patent/DK170024B1/da

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Neurology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Biomedical Technology (AREA)
  • Public Health (AREA)
  • Diabetes (AREA)
  • Child & Adolescent Psychology (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Anesthesiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pyrane Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Adhesives Or Adhesive Processes (AREA)
  • Photoreceptors In Electrophotography (AREA)
DK579688A 1987-10-20 1988-10-18 Imidazo(2,1-b)thiazolderivater, deres fremstilling, mellemprodukter til anvendelse i forbindelse hermed, deres anvendelse som lægemidler samt farmaceutiske præparater med indhold heraf DK170024B1 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB878724566A GB8724566D0 (en) 1987-10-20 1987-10-20 Chemical compounds
GB8724566 1987-10-20

Publications (3)

Publication Number Publication Date
DK579688D0 DK579688D0 (da) 1988-10-18
DK579688A DK579688A (da) 1989-04-21
DK170024B1 true DK170024B1 (da) 1995-05-01

Family

ID=10625613

Family Applications (1)

Application Number Title Priority Date Filing Date
DK579688A DK170024B1 (da) 1987-10-20 1988-10-18 Imidazo(2,1-b)thiazolderivater, deres fremstilling, mellemprodukter til anvendelse i forbindelse hermed, deres anvendelse som lægemidler samt farmaceutiske præparater med indhold heraf

Country Status (16)

Country Link
US (1) US4895863A (el)
EP (1) EP0313458B1 (el)
JP (1) JPH01193274A (el)
AT (1) ATE92928T1 (el)
AU (1) AU613413B2 (el)
CA (1) CA1331991C (el)
DE (1) DE3883140T2 (el)
DK (1) DK170024B1 (el)
ES (1) ES2059552T3 (el)
GB (2) GB8724566D0 (el)
GR (1) GR3009703T3 (el)
HU (1) HU201769B (el)
MX (1) MX173422B (el)
PT (1) PT88795B (el)
RU (1) RU2014334C1 (el)
ZA (1) ZA887433B (el)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8908846D0 (en) * 1989-04-19 1989-06-07 Roussel Lab Ltd Chemical compounds
GB8908845D0 (en) * 1989-04-19 1989-06-07 Roussel Lab Ltd Chemical compounds
FR2679232B1 (fr) * 1991-07-19 1994-01-14 Synthelabo Derives d'alpha-hydroxyimidazo [2,1-b] benzothiazole-3-acetamide, leur preparation et leur application en therapeutique.
EP0524055A1 (fr) * 1991-07-19 1993-01-20 Synthelabo Dérivés d'imidazo[2,1-b]benzothiazole-3-acétamide, leur préparation et leur application en thérapeutique
FR2679233B1 (fr) * 1991-07-19 1993-10-15 Synthelabo Derives d'imidazo [2,1-b] benzothiazole-3-acetamide, leur preparation et leur application en therapeutique.
FR2679136A1 (fr) * 1991-07-19 1993-01-22 Synthelabo Medicaments et compositions pharmaceutiques a base de derives d'imidazo[2,1-b]benzothiazole-3-acetamide.
FR2679231B1 (fr) * 1991-07-19 1994-01-14 Synthelabo Derives d'imidazo [2,1-b] benzothiazole-3-acetamide, leur preparation et leur application, en therapeutique.
FR2699920B1 (fr) * 1992-12-24 1995-02-10 Synthelabo Dérivés d'imidazo [2,1-b] benzothiazole-3-acétamide, leur préparation et leur application en thérapeutique.
FR2699921B1 (fr) * 1992-12-30 1995-02-10 Synthelabo Dérivés d'acide 2-(thien-2-yl)imidazo[2,1-b]benzothiazole-3-acétique, leur préparation et leur application en thérapeutique.
EP0799830B1 (de) * 1996-04-04 2002-05-29 Rolic AG Imidazothiazol-Derivate als komponente flüssigkristalline Mischungen
DE10004572A1 (de) * 2000-02-02 2001-08-09 Boehringer Ingelheim Pharma Neue positive allosterische AMPA-Rezeptor Modulatoren (PAARM), Verfahren zu deren Herstellung und deren Verwendung als Arzneimittel
AR039475A1 (es) 2002-05-01 2005-02-23 Wyeth Corp 6-alquiliden-penems triciclicos como inhibidores de beta-lactamasa
AR039774A1 (es) 2002-05-01 2005-03-02 Wyeth Corp 6-alquiliden-penems biciclicos como inhibidores de beta-lactamasas
GT200600380A (es) * 2005-08-24 2007-03-29 Proceso para la preparacion de inhibidores de beta-lactamasa
TWI648282B (zh) 2014-03-27 2019-01-21 印度商托仁特生技有限公司 新熔合咪唑苯并噻唑化合物

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH621126A5 (el) * 1974-02-07 1981-01-15 Plantex Ltd
US4464384A (en) * 1981-12-23 1984-08-07 Yamanouchi Pharmaceutical Co., Ltd. 2-Phenylimidazo[2,1-b]benzothiazole compounds, salts thereof, process of producing them, and pharmaceutical compositions containing them
US4721721A (en) * 1984-12-18 1988-01-26 Rorer Pharmaceutical Corporation 6-(4-thiazole) compounds, cardiotonic compositions including the same, and their uses
IL78834A (en) * 1985-05-23 1992-07-15 Smithkline Beckman Corp 2,3-dihydro-5-(1,4-dihydropyridin-4-yl)-6-phenylimidazo(2,1-b)thiazoles and 6,7-dihydro-3-(1,4-dihydropyridin-4-yl)-2-phenyl-5h-imidazo(2,1-b)(1,3)thiazines and their use as intermediates in a process for preparing the corresponding pyridyl-substituted imidazo(2,1-b)thiazoles and 5h-imidazo(2,1-b)(1,3)thiazines
ZW24186A1 (en) * 1985-12-12 1987-07-08 Smithkline Beckman Corp Inhibition of the 5-lipoxygenase pathway

Also Published As

Publication number Publication date
MX13455A (es) 1993-10-01
JPH01193274A (ja) 1989-08-03
AU613413B2 (en) 1991-08-01
CA1331991C (en) 1994-09-13
ZA887433B (en) 1990-01-31
HU201769B (en) 1990-12-28
DK579688A (da) 1989-04-21
EP0313458B1 (fr) 1993-08-11
GB8824492D0 (en) 1988-11-23
DE3883140T2 (de) 1994-01-13
EP0313458A2 (fr) 1989-04-26
GB2211186B (en) 1991-07-31
EP0313458A3 (en) 1990-10-31
GR3009703T3 (el) 1994-02-28
GB8724566D0 (en) 1987-11-25
MX173422B (es) 1994-03-03
PT88795B (pt) 1993-01-29
RU2014334C1 (ru) 1994-06-15
HUT50836A (en) 1990-03-28
GB2211186A (en) 1989-06-28
AU2397888A (en) 1989-04-20
ATE92928T1 (de) 1993-08-15
ES2059552T3 (es) 1994-11-16
DK579688D0 (da) 1988-10-18
DE3883140D1 (de) 1993-09-16
US4895863A (en) 1990-01-23

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Legal Events

Date Code Title Description
B1 Patent granted (law 1993)
PBP Patent lapsed