DK167393B1 - 1-sulfonyl-2-oxo-pyrrolidinderivater, deres fremstilling og farmaceutiske praeparater med indhold deraf - Google Patents

1-sulfonyl-2-oxo-pyrrolidinderivater, deres fremstilling og farmaceutiske praeparater med indhold deraf Download PDF

Info

Publication number
DK167393B1
DK167393B1 DK621486A DK621486A DK167393B1 DK 167393 B1 DK167393 B1 DK 167393B1 DK 621486 A DK621486 A DK 621486A DK 621486 A DK621486 A DK 621486A DK 167393 B1 DK167393 B1 DK 167393B1
Authority
DK
Denmark
Prior art keywords
formula
compounds
compound
oxo
pyrrolidine
Prior art date
Application number
DK621486A
Other languages
Danish (da)
English (en)
Other versions
DK621486A (da
DK621486D0 (da
Inventor
Emilio Toja
Carlo Gorini
Carlo Zirotti
Fernando Barzaghi
Giulio Galliani
Original Assignee
Roussel Uclaf
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from IT23406/85A external-priority patent/IT1201513B/it
Priority claimed from IT21105/86A external-priority patent/IT1196483B/it
Application filed by Roussel Uclaf filed Critical Roussel Uclaf
Publication of DK621486D0 publication Critical patent/DK621486D0/da
Publication of DK621486A publication Critical patent/DK621486A/da
Application granted granted Critical
Publication of DK167393B1 publication Critical patent/DK167393B1/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D207/00Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/46Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with hetero atoms directly attached to the ring nitrogen atom
    • C07D207/48Sulfur atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • General Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Psychiatry (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Hospice & Palliative Care (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyrrole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
DK621486A 1985-12-30 1986-12-22 1-sulfonyl-2-oxo-pyrrolidinderivater, deres fremstilling og farmaceutiske praeparater med indhold deraf DK167393B1 (da)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
IT23406/85A IT1201513B (it) 1985-12-30 1985-12-30 Derivati della 1-benzensolfonil 2-osso 5-alcossi pirrolidina,loro procedimento di preparazione e loro impiego come sostanze medicinali
IT2340685 1985-12-30
IT21105/86A IT1196483B (it) 1986-07-11 1986-07-11 Derivati della 1-benzene solfonil 2-osso 5-alcossi pirrolidina,loro procedimento di preparazione e loro applicazione come farmaci
IT2110586 1986-07-11

Publications (3)

Publication Number Publication Date
DK621486D0 DK621486D0 (da) 1986-12-22
DK621486A DK621486A (da) 1987-07-01
DK167393B1 true DK167393B1 (da) 1993-10-25

Family

ID=26327781

Family Applications (1)

Application Number Title Priority Date Filing Date
DK621486A DK167393B1 (da) 1985-12-30 1986-12-22 1-sulfonyl-2-oxo-pyrrolidinderivater, deres fremstilling og farmaceutiske praeparater med indhold deraf

Country Status (15)

Country Link
US (1) US4829079A (ru)
EP (1) EP0229566B1 (ru)
JP (1) JPH064585B2 (ru)
AU (1) AU592605B2 (ru)
CA (1) CA1265804A (ru)
DE (1) DE3685210D1 (ru)
DK (1) DK167393B1 (ru)
ES (1) ES2032752T3 (ru)
FI (1) FI82447C (ru)
GR (1) GR3004847T3 (ru)
HU (1) HU198013B (ru)
IE (1) IE59604B1 (ru)
MX (1) MX173418B (ru)
PT (1) PT84023B (ru)
SU (1) SU1480765A3 (ru)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1204494B (it) * 1986-03-28 1989-03-01 Roussel Maestretti Spa Derivati della 1-stirene solfonil 2-osso 5-alcossi pirrolidina,loro procedimento di preparazione e loro applicazione come farmaci
IT1215590B (it) * 1987-06-29 1990-02-14 Roussel Maestretti Spa Derivati della 1-benzene solfonil 2-oco 5-alchiltio pirrolidina, un loro procedimentodi preparazione e il loro impiegocome stostanze medicinali.
US5280032A (en) * 1989-02-14 1994-01-18 Toyama Chemical Co., Ltd. 1,2-ethanediol derivative and salt thereof, process for producing the same, and cerebral function-improving agent comprising the same
IT1228462B (it) * 1989-02-23 1991-06-19 Roussel Maestretti S P A Milan Derivati del 1 arilsolfonil pirrolidin 2 tione oppure del 1 arilsolfonil piperidin 2 tione, loro procedimento di preparazione e loro impiego come medicinali.
FR2647785B1 (fr) * 1989-05-31 1991-09-06 Adir Nouveaux derives de la pyrrolidone, leur procede de preparation et les compositions pharmaceutiques les renfermant
IT1244881B (it) * 1990-12-13 1994-09-12 Roussel Pharma Spa Derivati dell'1-arilsolfonil 2-pirrolidone, loro procedimento di preparazione e i nuovi intermedi cosi' ottenuti ,il loro impiego come farmaci e le composizioni farmaceutiche che li contengono
FR2686878B1 (fr) 1992-01-30 1995-06-30 Sanofi Elf Derives du n-sulfonyl oxo-2 indole, leur preparation, les compositions pharmaceutiques en contenant.
JP2873898B2 (ja) * 1992-04-13 1999-03-24 富山化学工業株式会社 ベンゾ[b]チオフェン−5−イル誘導体もしくはその光学活性体またはそれらの塩並びにそれらの製造法
WO1995025101A1 (en) * 1994-03-14 1995-09-21 Merck & Co., Inc. Pyridil ethylation of lactams
US5707985A (en) * 1995-06-07 1998-01-13 Tanabe Seiyaku Co. Ltd. Naphthyl-, quinolyl- and isoquinolyl- sulfonamide derivatives as cell adhesion modulators
KR100442031B1 (ko) * 2001-10-30 2004-07-30 신국현 신규한 알칼로이드 화합물 및 그의 제조방법
JP6746605B2 (ja) 2014-12-19 2020-08-26 ガイストリッヒ・ファルマ・アーゲーGeistlich Pharma Ag オキサチアジン様化合物を作製する方法
US11591302B2 (en) 2014-12-19 2023-02-28 Geistlich Pharm A Ag Processes for preparing oxathiazin-like compounds

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3117975A (en) * 1960-04-22 1964-01-14 Rohm & Haas Substituted pyrrolidinones and piperidinones
US3453289A (en) * 1966-01-21 1969-07-01 American Home Prod P-substituted-phenylsulfonyl pyrrolidine derivatives
JPS5822111B2 (ja) * 1977-10-29 1983-05-06 協和醗酵工業株式会社 柑橘類果実の改質剤
FR2553409B1 (fr) * 1983-10-18 1986-04-18 Choay Sa Nouveaux benzenesulfonyl-lactames, leur procede de preparation et leur application comme substance active de compositions pharmaceutiques

Also Published As

Publication number Publication date
MX173418B (es) 1994-03-03
CA1265804A (fr) 1990-02-13
EP0229566A2 (fr) 1987-07-22
IE863384L (en) 1987-06-30
DK621486A (da) 1987-07-01
GR3004847T3 (ru) 1993-04-28
FI82447C (fi) 1991-03-11
AU592605B2 (en) 1990-01-18
PT84023B (pt) 1989-07-31
JPH064585B2 (ja) 1994-01-19
EP0229566B1 (fr) 1992-05-06
FI82447B (fi) 1990-11-30
DK621486D0 (da) 1986-12-22
US4829079A (en) 1989-05-09
IE59604B1 (en) 1994-03-09
MX9260A (es) 1993-11-01
PT84023A (fr) 1987-01-01
DE3685210D1 (de) 1992-06-11
EP0229566A3 (en) 1988-07-27
JPS62195362A (ja) 1987-08-28
ES2032752T3 (es) 1993-03-01
HUT43562A (en) 1987-11-30
FI865315A (fi) 1987-07-01
AU6697786A (en) 1987-07-02
FI865315A0 (fi) 1986-12-29
SU1480765A3 (ru) 1989-05-15
HU198013B (en) 1989-07-28

Similar Documents

Publication Publication Date Title
DK167393B1 (da) 1-sulfonyl-2-oxo-pyrrolidinderivater, deres fremstilling og farmaceutiske praeparater med indhold deraf
DK171614B1 (da) Tiazolidindionderivater og deres fremstilling og anvendelse
DK163501B (da) (s)-alfa-ethyl-2-oxo-1-pyrrolidinacetamid, fremgangsmaader til dets fremstilling samt farmaceutisk praeparat indeholdende denne forbindelse
KR910007882B1 (ko) 1-벤질-아미노알킬-피롤리디논의 제조방법
IE68346B1 (en) Condensed heterocyclic compounds their production and use
NO122814B (ru)
DK155278B (da) Analogifremgangsmaade til fremstilling af 1-(p-methoxybenzoyl)-2-pyrrolidinon samt 4-(p-methoxybenzoylamino)smoersyre til anvendelse som udgangsmateriale ved denne fremgangsmaade
NO156385B (no) Anordning for laasing av dreibare maskinelementer.
JPH03133960A (ja) キノロンカルボン酸誘導体、それらを調製する方法および抗ウイルス剤としてのそれらの使用
WO2011142825A2 (en) Novel sulfur containing compounds
NO863790L (no) Kinolinderivater.
NL8700119A (nl) Pyroglutamidederivaten, nootropisch geneesmiddel dat specifieke pyroglutamidederivaten bevat, specifieke pyroglutamidederivaten alsmede werkwijze voor de bereiding van deze laatsten.
NO157141B (no) Analogifremgangsmaate for fremstilling av terapeutisk aktive 4-metyl-6-fenylpyridazinderivater.
NO311761B1 (no) 2-(3H)-Oksazolonderivater og deres anvendelse
CA1068707A (en) 4-piperidinylalkyl-3,3-diphenyl-2-pyrrolidinones
US4324791A (en) Heterocyclic antidiarrheal compositions & methods of use
HU198676B (en) Process for production of derivatives of hydrocinnamic acid and medical compositions containing them as active substance
NO832894L (no) Fremgangsmaate for fremstilling av n-substituerte nikotinamid-1-oksyd-derivater
DK158944B (da) Analogifremgangsmaade til fremstilling af substituerede methylimidazolforbindelser
NO752174L (ru)
DK145781B (da) Analogifremgangsmaade til fremstilling af ditiino(1,4)(2,3-c)pyrrolderivater
DD223616A5 (de) Verfahren zur herstellung trisubstituierter oxazolidinone
DK149750B (da) Analogifremgangsmaade til fremstilling af n-alkenylmoranolin-derivater eller farmaceutiske acceptable syreadditionssalte deraf
US4897414A (en) Derivatives of 1-benzensulphonyl-2-oxo-5-alkylthio pyrrolidine, and compositions containing them
NO160139B (no) Analogifremgangsmaate for fremstilling av terapeutisk aktive akridanonderivater.

Legal Events

Date Code Title Description
B1 Patent granted (law 1993)
PBP Patent lapsed