DK163510C - Fremgangsmaade til fremstilling af (3s)-3-oeoe(2-amino-4-thioazolyl)-oe(1-carboxy-1-methylethoxy)iminoaaacetylaaaminoaa-2-oxo-1-azetidinsulfonsyre og 4-alkylsubstituerede derivater deraf samt mellemprodukt til brug ved fremgangsmaaden - Google Patents
Fremgangsmaade til fremstilling af (3s)-3-oeoe(2-amino-4-thioazolyl)-oe(1-carboxy-1-methylethoxy)iminoaaacetylaaaminoaa-2-oxo-1-azetidinsulfonsyre og 4-alkylsubstituerede derivater deraf samt mellemprodukt til brug ved fremgangsmaadenInfo
- Publication number
- DK163510C DK163510C DK280783A DK280783A DK163510C DK 163510 C DK163510 C DK 163510C DK 280783 A DK280783 A DK 280783A DK 280783 A DK280783 A DK 280783A DK 163510 C DK163510 C DK 163510C
- Authority
- DK
- Denmark
- Prior art keywords
- amino
- methyl
- procedure
- preparation
- thiazoyl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/38—Nitrogen atoms
- C07D277/44—Acylated amino or imino radicals
- C07D277/46—Acylated amino or imino radicals by carboxylic acids, or sulfur or nitrogen analogues thereof
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Oncology (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Communicable Diseases (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Saccharide Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Cephalosporin Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US39072882 | 1982-06-21 | ||
| US06/390,728 US4704457A (en) | 1982-06-21 | 1982-06-21 | Process for the preparation of (3S)-3-[[[2-(protected amino)-4-thiazolyl]-oxoacetyl]amino]-2-oxo-1-azetidinesulfonic acid and 4-substituted derivatives thereof |
Publications (4)
| Publication Number | Publication Date |
|---|---|
| DK280783D0 DK280783D0 (da) | 1983-06-17 |
| DK280783A DK280783A (da) | 1983-12-22 |
| DK163510B DK163510B (da) | 1992-03-09 |
| DK163510C true DK163510C (da) | 1992-07-27 |
Family
ID=23543684
Family Applications (3)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK280783A DK163510C (da) | 1982-06-21 | 1983-06-17 | Fremgangsmaade til fremstilling af (3s)-3-oeoe(2-amino-4-thioazolyl)-oe(1-carboxy-1-methylethoxy)iminoaaacetylaaaminoaa-2-oxo-1-azetidinsulfonsyre og 4-alkylsubstituerede derivater deraf samt mellemprodukt til brug ved fremgangsmaaden |
| DK146591A DK166322C (da) | 1982-06-21 | 1991-08-14 | Fremgangsmaade til fremstilling af azetidinsulfonsyrederivater |
| DK106592A DK166209C (da) | 1982-06-21 | 1992-08-27 | Mellemprodukt til fremstilling af azetidinsulfonsyrederivater |
Family Applications After (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK146591A DK166322C (da) | 1982-06-21 | 1991-08-14 | Fremgangsmaade til fremstilling af azetidinsulfonsyrederivater |
| DK106592A DK166209C (da) | 1982-06-21 | 1992-08-27 | Mellemprodukt til fremstilling af azetidinsulfonsyrederivater |
Country Status (18)
| Country | Link |
|---|---|
| US (1) | US4704457A (da) |
| EP (1) | EP0097352B1 (da) |
| JP (1) | JPS597190A (da) |
| KR (1) | KR880001048B1 (da) |
| AT (1) | ATE30155T1 (da) |
| AU (1) | AU563938B2 (da) |
| CA (1) | CA1205076A (da) |
| DE (1) | DE3374008D1 (da) |
| DK (3) | DK163510C (da) |
| ES (2) | ES8503682A1 (da) |
| GR (1) | GR78278B (da) |
| HU (3) | HU194560B (da) |
| IE (1) | IE55234B1 (da) |
| NO (1) | NO832229L (da) |
| NZ (1) | NZ204214A (da) |
| PH (2) | PH18423A (da) |
| PT (1) | PT76896B (da) |
| ZA (1) | ZA833623B (da) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5484928A (en) * | 1984-04-10 | 1996-01-16 | Biochemie Gesellschaft M.B.H. | 2-(2-aminothiazol-4-yl)-2-oxoacetic acid derivatives |
| US4647660A (en) * | 1985-05-02 | 1987-03-03 | E. R. Squibb & Sons, Inc. | 3-acylamino-2-oxo-1-azetidinesulfonic acids |
| US4675398A (en) * | 1985-08-16 | 1987-06-23 | E. R. Squibb & Sons, Inc. | Copper-mediated oximation reaction |
| US4684722A (en) * | 1986-01-06 | 1987-08-04 | E. R. Squibb & Sons, Inc. | Monosulfactams |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB1575803A (en) * | 1976-03-09 | 1980-10-01 | Fujisawa Pharmaceutical Co | 3,7 disubstituted 3 cephem 4 carboxylic acid compounds andprocesses for the preparation thereof |
| US4166115A (en) * | 1976-04-12 | 1979-08-28 | Fujisawa Pharmaceutical Co., Ltd. | Syn 7-oxoimino substituted derivatives of cephalosporanic acid |
| US4237128A (en) * | 1979-04-12 | 1980-12-02 | E. R. Squibb & Sons, Inc. | 7-[2-(2-Amino-4-thiazolyl)-2-[(1-carboxy-1,1-dialkyl)alkoxyimino]acetamido]cephem sulfoxides |
| NZ196202A (en) * | 1980-02-07 | 1984-07-31 | Squibb & Sons Inc | Beta-lactam antibiotics (of azetidine-sulphonic acid type) |
| EP0048953B1 (en) * | 1980-09-29 | 1988-03-09 | E.R. Squibb & Sons, Inc. | Beta-lactam antibiotics |
| US4443374A (en) * | 1982-02-01 | 1984-04-17 | E. R. Squibb & Sons, Inc. | Process for preparing (3S)-3-[[(2-amino-4-thiazolyl)[(1-carboxy-1-methylethoxy)imino]-acetyl]amino]-2-oxo-1-azetidinesulfonic acid, and 4-substituted derivatives |
-
1982
- 1982-06-21 US US06/390,728 patent/US4704457A/en not_active Expired - Lifetime
-
1983
- 1983-05-10 CA CA000427829A patent/CA1205076A/en not_active Expired
- 1983-05-12 NZ NZ204214A patent/NZ204214A/en unknown
- 1983-05-12 AU AU14499/83A patent/AU563938B2/en not_active Expired
- 1983-05-19 ZA ZA833623A patent/ZA833623B/xx unknown
- 1983-05-20 PH PH28939A patent/PH18423A/en unknown
- 1983-06-03 JP JP58100110A patent/JPS597190A/ja active Granted
- 1983-06-03 GR GR71555A patent/GR78278B/el unknown
- 1983-06-13 IE IE1382/83A patent/IE55234B1/en not_active IP Right Cessation
- 1983-06-17 DK DK280783A patent/DK163510C/da not_active IP Right Cessation
- 1983-06-20 HU HU831047A patent/HU194560B/hu unknown
- 1983-06-20 ES ES523420A patent/ES8503682A1/es not_active Expired
- 1983-06-20 PT PT76896A patent/PT76896B/pt unknown
- 1983-06-20 HU HU831046A patent/HU194558B/hu unknown
- 1983-06-20 NO NO832229A patent/NO832229L/no unknown
- 1983-06-20 KR KR1019830002746A patent/KR880001048B1/ko not_active IP Right Cessation
- 1983-06-20 DE DE8383106005T patent/DE3374008D1/de not_active Expired
- 1983-06-20 EP EP83106005A patent/EP0097352B1/en not_active Expired
- 1983-06-20 HU HU832191A patent/HU190903B/hu unknown
- 1983-06-20 AT AT83106005T patent/ATE30155T1/de not_active IP Right Cessation
-
1984
- 1984-11-26 ES ES537960A patent/ES537960A0/es active Granted
- 1984-12-10 PH PH31557A patent/PH22121A/en unknown
-
1991
- 1991-08-14 DK DK146591A patent/DK166322C/da not_active IP Right Cessation
-
1992
- 1992-08-27 DK DK106592A patent/DK166209C/da not_active IP Right Cessation
Also Published As
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| DK160939C (da) | Analogifremgangsmaade til fremstilling af benzisothiazol- og benzisoxazolpiperazinderivater, samt mellemprodukter til anvendelse ved fremgangsmaaden | |
| DK503288A (da) | Oxazol- eller thiazolforbindelse, farmaceutisk anvendelse deraf og fremgangsmaade til fremstillig af en saadan forbindelse | |
| DK590787D0 (da) | Cephalosporinsulfonforbindelse, fremgangsmaade og mellemprodukt til fremstilling deraf samt farmaceutisk praeparat indeholdende en saadan forbindelse | |
| DK63388A (da) | Isocyanomethylforbindelse samt fremgangsmaade til fremstilling af et oxadiazolimidazobenzodiazepinderivat | |
| DK163510C (da) | Fremgangsmaade til fremstilling af (3s)-3-oeoe(2-amino-4-thioazolyl)-oe(1-carboxy-1-methylethoxy)iminoaaacetylaaaminoaa-2-oxo-1-azetidinsulfonsyre og 4-alkylsubstituerede derivater deraf samt mellemprodukt til brug ved fremgangsmaaden | |
| AU6845990A (en) | Karl-fishcher reagent and a process for the determination of water with the aid of this reagent | |
| DK0460446T3 (da) | Koblingsreagens til peptidsyntesen | |
| DK355081A (da) | 7-beta-(alfa-syn-methoxyimino-alfa(2-aminothiazol-4-yl) acetamido)-3-( (1,2,3-triadiazol-5-ylthio) methyl)-3-cephem-4-carboxylsyre samt c1-c6-alkylderivater heraf fremgangsmaade til fremstilling heraf samt deres anvendelse som antibakterielle midler | |
| DK0466963T3 (da) | Fremgangsmåde til fremstilling af alfa-L-aspartyl-L-phenyl-alaninmethylester, hydroclorid ved anvend else af isoleret N-formyl-asparaginsyreanhydrid | |
| DK451888A (da) | C12-modificerede erythromycin-a-derivater og fremgangsmaade til fremstilling deraf samt forbindelser til anvendelse som udgangsmateriale ved fremgangsmaaden | |
| NO177348C (no) | Fremgangsmåte til fremstilling av et cefalosporin-antibiotikum, samt 3-(fluorsulfonyl)oksy-substituerte cefemer og karbacefemer | |
| DK439082A (da) | 4-acylamino-1-aza-adamantan-forbindelser samt fremgangsmaade til fremstilling deraf | |
| ZA907976B (en) | Novel 2-spirocyclopropyl cephalosporin sulfone derivatives and processes for the preparation thereof | |
| DK155604C (da) | Fremgangsmaade til fremstilling af 6-aminopenicillansyre-1,1-dioxid og dets ikke-toxiske, farmaceutisk acceptable salte | |
| DK0778827T3 (da) | Fremgangsmåde til fremstilling af en beta-aminoalkohol | |
| DK193580A (da) | Fremgangsmaade til fremstilling af 5-(2-( (2,3-dihydro-1,4-benzodioxan-2-yl-methyl)amino)-1-hydroxyethyl)-2-hydroxybenzoesyre-derivater | |
| DK165007C (da) | Fremgangsmaade til fremstilling af et phosphinoxidderivat ved chlorering og hydrolyse af det tilsvarende phosphinsulfidderivat | |
| DK555288D0 (da) | Cephalosporinderivater og fremgangsmaade til fremstilling deraf, farmaceutiske midler indeholdende derivaterne og mellemprodukter til anvendelse ved fremgangsmaaden | |
| DK513888D0 (da) | Fremgangsmaade til fremstilling af 2-(1-halogenalkyl)thiazol-forbindelser samt hidtil ukendte forbindelser, som kan fremstilles ved fremgangsmaaden | |
| NO168339C (no) | Fremgangsmaate for aa synkronisere et flertall av navigasjonslanterner ved daggry og moerkning, samt et navigasjonslanternesystem for utfoerelse av fremgangsmaaten | |
| DK165263C (da) | Fremgangsmaade ved og anlaeg til hoejvaerdig udnyttelse af biobraendsler | |
| IT221288Z2 (it) | Congegno a strappo per l'apertura dei films termoretraenti di imbal= laggio. | |
| FI910956A0 (fi) | Menetelmä terapeuttisesti käyttökelpoisen 2-(1-(pentyyli-3-guanidino)-2-metyyli-4-imidatsolyyli)tiatsolihemifosfaattihemihydraattisuolan valmistamiseksi |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PUP | Patent expired |