DK146591A - Fremgangsmaade og mellemprodukt til fremstilling af azetidinsulfonsyrederivater - Google Patents

Fremgangsmaade og mellemprodukt til fremstilling af azetidinsulfonsyrederivater Download PDF

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Publication number
DK146591A
DK146591A DK146591A DK146591A DK146591A DK 146591 A DK146591 A DK 146591A DK 146591 A DK146591 A DK 146591A DK 146591 A DK146591 A DK 146591A DK 146591 A DK146591 A DK 146591A
Authority
DK
Denmark
Prior art keywords
preparation
acid derivatives
sulphonic acid
azetidine
azetidine sulphonic
Prior art date
Application number
DK146591A
Other languages
English (en)
Other versions
DK166322C (da
DK146591D0 (da
DK166322B (da
Inventor
Jerome Leon Moniot
Christopher Michael Cimarusti
Rita Therese Fox
Original Assignee
Squibb & Sons Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Squibb & Sons Inc filed Critical Squibb & Sons Inc
Publication of DK146591A publication Critical patent/DK146591A/da
Publication of DK146591D0 publication Critical patent/DK146591D0/da
Publication of DK166322B publication Critical patent/DK166322B/da
Application granted granted Critical
Publication of DK166322C publication Critical patent/DK166322C/da

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/38—Nitrogen atoms
    • C07D277/44—Acylated amino or imino radicals
    • C07D277/46—Acylated amino or imino radicals by carboxylic acids, or sulfur or nitrogen analogues thereof
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Saccharide Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Cephalosporin Compounds (AREA)
DK146591A 1982-06-21 1991-08-14 Fremgangsmaade til fremstilling af azetidinsulfonsyrederivater DK166322C (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US39072882 1982-06-21
US06/390,728 US4704457A (en) 1982-06-21 1982-06-21 Process for the preparation of (3S)-3-[[[2-(protected amino)-4-thiazolyl]-oxoacetyl]amino]-2-oxo-1-azetidinesulfonic acid and 4-substituted derivatives thereof

Publications (4)

Publication Number Publication Date
DK146591A true DK146591A (da) 1991-08-14
DK146591D0 DK146591D0 (da) 1991-08-14
DK166322B DK166322B (da) 1993-04-05
DK166322C DK166322C (da) 1993-08-23

Family

ID=23543684

Family Applications (3)

Application Number Title Priority Date Filing Date
DK280783A DK163510C (da) 1982-06-21 1983-06-17 Fremgangsmaade til fremstilling af (3s)-3-oeoe(2-amino-4-thioazolyl)-oe(1-carboxy-1-methylethoxy)iminoaaacetylaaaminoaa-2-oxo-1-azetidinsulfonsyre og 4-alkylsubstituerede derivater deraf samt mellemprodukt til brug ved fremgangsmaaden
DK146591A DK166322C (da) 1982-06-21 1991-08-14 Fremgangsmaade til fremstilling af azetidinsulfonsyrederivater
DK106592A DK166209C (da) 1982-06-21 1992-08-27 Mellemprodukt til fremstilling af azetidinsulfonsyrederivater

Family Applications Before (1)

Application Number Title Priority Date Filing Date
DK280783A DK163510C (da) 1982-06-21 1983-06-17 Fremgangsmaade til fremstilling af (3s)-3-oeoe(2-amino-4-thioazolyl)-oe(1-carboxy-1-methylethoxy)iminoaaacetylaaaminoaa-2-oxo-1-azetidinsulfonsyre og 4-alkylsubstituerede derivater deraf samt mellemprodukt til brug ved fremgangsmaaden

Family Applications After (1)

Application Number Title Priority Date Filing Date
DK106592A DK166209C (da) 1982-06-21 1992-08-27 Mellemprodukt til fremstilling af azetidinsulfonsyrederivater

Country Status (18)

Country Link
US (1) US4704457A (da)
EP (1) EP0097352B1 (da)
JP (1) JPS597190A (da)
KR (1) KR880001048B1 (da)
AT (1) ATE30155T1 (da)
AU (1) AU563938B2 (da)
CA (1) CA1205076A (da)
DE (1) DE3374008D1 (da)
DK (3) DK163510C (da)
ES (2) ES523420A0 (da)
GR (1) GR78278B (da)
HU (3) HU194558B (da)
IE (1) IE55234B1 (da)
NO (1) NO832229L (da)
NZ (1) NZ204214A (da)
PH (2) PH18423A (da)
PT (1) PT76896B (da)
ZA (1) ZA833623B (da)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5484928A (en) * 1984-04-10 1996-01-16 Biochemie Gesellschaft M.B.H. 2-(2-aminothiazol-4-yl)-2-oxoacetic acid derivatives
US4647660A (en) * 1985-05-02 1987-03-03 E. R. Squibb & Sons, Inc. 3-acylamino-2-oxo-1-azetidinesulfonic acids
US4675398A (en) * 1985-08-16 1987-06-23 E. R. Squibb & Sons, Inc. Copper-mediated oximation reaction
US4684722A (en) * 1986-01-06 1987-08-04 E. R. Squibb & Sons, Inc. Monosulfactams

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1575803A (en) * 1976-03-09 1980-10-01 Fujisawa Pharmaceutical Co 3,7 disubstituted 3 cephem 4 carboxylic acid compounds andprocesses for the preparation thereof
US4166115A (en) * 1976-04-12 1979-08-28 Fujisawa Pharmaceutical Co., Ltd. Syn 7-oxoimino substituted derivatives of cephalosporanic acid
US4237128A (en) * 1979-04-12 1980-12-02 E. R. Squibb & Sons, Inc. 7-[2-(2-Amino-4-thiazolyl)-2-[(1-carboxy-1,1-dialkyl)alkoxyimino]acetamido]cephem sulfoxides
NZ196202A (en) * 1980-02-07 1984-07-31 Squibb & Sons Inc Beta-lactam antibiotics (of azetidine-sulphonic acid type)
EP0048953B1 (en) * 1980-09-29 1988-03-09 E.R. Squibb & Sons, Inc. Beta-lactam antibiotics
US4443374A (en) * 1982-02-01 1984-04-17 E. R. Squibb & Sons, Inc. Process for preparing (3S)-3-[[(2-amino-4-thiazolyl)[(1-carboxy-1-methylethoxy)imino]-acetyl]amino]-2-oxo-1-azetidinesulfonic acid, and 4-substituted derivatives

Also Published As

Publication number Publication date
ATE30155T1 (de) 1987-10-15
PT76896B (en) 1986-01-24
PH22121A (en) 1988-06-01
CA1205076A (en) 1986-05-27
AU1449983A (en) 1984-01-05
JPS597190A (ja) 1984-01-14
ES8503682A1 (es) 1985-03-16
DK163510C (da) 1992-07-27
DK280783A (da) 1983-12-22
NO832229L (no) 1983-12-22
PH18423A (en) 1985-06-26
GR78278B (da) 1984-09-26
DK166209B (da) 1993-03-22
AU563938B2 (en) 1987-07-30
NZ204214A (en) 1986-01-24
DK106592A (da) 1992-08-27
DK166322C (da) 1993-08-23
EP0097352A3 (en) 1984-09-12
DK166209C (da) 1993-08-16
PT76896A (en) 1983-07-01
ES8601984A1 (es) 1985-11-01
KR840005114A (ko) 1984-11-03
HU194558B (en) 1988-02-29
HU190903B (en) 1986-12-28
IE55234B1 (en) 1990-07-04
ES523420A0 (es) 1985-03-16
DK106592D0 (da) 1992-08-27
KR880001048B1 (ko) 1988-06-18
DK163510B (da) 1992-03-09
ZA833623B (en) 1984-02-29
HU194560B (en) 1988-02-29
EP0097352A2 (en) 1984-01-04
EP0097352B1 (en) 1987-10-07
JPH0348910B2 (da) 1991-07-25
DK280783D0 (da) 1983-06-17
DK146591D0 (da) 1991-08-14
DK166322B (da) 1993-04-05
IE831382L (en) 1983-12-21
ES537960A0 (es) 1985-11-01
US4704457A (en) 1987-11-03
DE3374008D1 (en) 1987-11-12

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