DK1419174T3 - Fremgangsmåde til fremstilling af glycopeptidderivater - Google Patents

Fremgangsmåde til fremstilling af glycopeptidderivater

Info

Publication number
DK1419174T3
DK1419174T3 DK02759433T DK02759433T DK1419174T3 DK 1419174 T3 DK1419174 T3 DK 1419174T3 DK 02759433 T DK02759433 T DK 02759433T DK 02759433 T DK02759433 T DK 02759433T DK 1419174 T3 DK1419174 T3 DK 1419174T3
Authority
DK
Denmark
Prior art keywords
preparation
glycopeptide derivatives
derivatives
glycopeptide
isolation
Prior art date
Application number
DK02759433T
Other languages
English (en)
Inventor
Junning Lee
Jyanwei Liu
Original Assignee
Theravance Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Theravance Inc filed Critical Theravance Inc
Application granted granted Critical
Publication of DK1419174T3 publication Critical patent/DK1419174T3/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/50—Cyclic peptides containing at least one abnormal peptide link
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K9/00—Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof
    • C07K9/006—Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof the peptide sequence being part of a ring structure
    • C07K9/008—Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof the peptide sequence being part of a ring structure directly attached to a hetero atom of the saccharide radical, e.g. actaplanin, avoparcin, ristomycin, vancomycin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
DK02759433T 2001-08-24 2002-08-23 Fremgangsmåde til fremstilling af glycopeptidderivater DK1419174T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US31471101P 2001-08-24 2001-08-24
PCT/US2002/026831 WO2003018607A2 (en) 2001-08-24 2002-08-23 Process for preparing glycopeptide derivatives

Publications (1)

Publication Number Publication Date
DK1419174T3 true DK1419174T3 (da) 2007-07-02

Family

ID=23221113

Family Applications (1)

Application Number Title Priority Date Filing Date
DK02759433T DK1419174T3 (da) 2001-08-24 2002-08-23 Fremgangsmåde til fremstilling af glycopeptidderivater

Country Status (14)

Country Link
US (2) US7015305B2 (da)
EP (1) EP1419174B1 (da)
JP (1) JP4116546B2 (da)
KR (1) KR100909435B1 (da)
CN (1) CN1281619C (da)
AT (1) ATE360029T1 (da)
AU (1) AU2002324768A1 (da)
CA (1) CA2457215C (da)
DE (1) DE60219638T2 (da)
DK (1) DK1419174T3 (da)
ES (1) ES2284907T3 (da)
NO (1) NO335304B1 (da)
TW (1) TWI312785B (da)
WO (1) WO2003018607A2 (da)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2003106399A2 (en) 2002-06-17 2003-12-24 Theravance, Inc. PROCESS FOR PREPARING N-PROTECTED β-AMINO ALDEHYDE COMPOUNDS
TWI342312B (en) * 2003-10-22 2011-05-21 Theravance Inc Hydrochloride salts of a glycopeptide phosphonate derivative
BRPI0514381A (pt) * 2004-07-30 2008-06-10 Palumed Sa compostos hìbridos de aminoquinolina-antibiótico, composições farmacêuticas, método de preparação e uso destes
WO2013034676A1 (en) 2011-09-09 2013-03-14 Sandoz Ag Process for the synthesis of telavancin, its pharmaceutically acceptable salts as well as an n-protected imine-derivative of telavancin
WO2013034675A1 (en) 2011-09-09 2013-03-14 Sandoz Ag Process for the synthesis of telavancin and its pharmaceutically acceptable salts as well as n-protected derivatives thereof
BR112017017883A2 (pt) 2015-02-23 2018-07-17 Theravance Biopharma Antibiotics Ip Llc doses e métodos para administrar telavancina
CN106467570B (zh) * 2015-08-14 2020-04-07 正大天晴药业集团股份有限公司 糖肽类抗生素的还原烷基化方法
CN106631902A (zh) * 2016-09-23 2017-05-10 上海步越化工科技有限公司 一种特拉万星侧链癸基(2‑氧代乙基)氨基甲酸9h‑芴‑9‑甲基酯的制备方法
US20200368312A1 (en) 2017-05-22 2020-11-26 Insmed Incorporated Glycopeptide derivative compounds and uses thereof
CN111233713A (zh) * 2020-01-20 2020-06-05 福建康鸿生物科技有限公司 一种特拉万星中间体合成方法
WO2022198009A1 (en) * 2021-03-18 2022-09-22 Insmed Incorporated Dry powder compositions of glycopeptide derivative compounds and methods of use thereof

Family Cites Families (24)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3160632A (en) * 1961-01-30 1964-12-08 Stauffer Chemical Co Aminomethylenephosphinic acids, salts thereof, and process for their production
US4698327A (en) * 1985-04-25 1987-10-06 Eli Lilly And Company Novel glycopeptide derivatives
IL78597A0 (en) 1985-04-25 1986-08-31 Lilly Co Eli Novel glycopeptide derivatives
US4643987A (en) * 1985-08-14 1987-02-17 Eli Lilly And Company Modified glycopeptides
EP0273727A3 (en) 1986-12-30 1990-01-17 Smithkline Beecham Corporation Glycosylated glycopeptides
ES2083374T3 (es) * 1988-12-27 1996-04-16 Lepetit Spa Derivados amidicos en posicion c63 de 34-des(acetilglucosaminil)-34-desoxi-teicoplaninas.
IL96603A (en) * 1989-12-13 1998-02-08 Lilly Co Eli Antibacterial glycopeptide derivativesProcess for their preparation and pharmaceutical preparations containing the same
US5750509A (en) * 1991-07-29 1998-05-12 Gruppo Lepetit S.P.A. Amide derivatives of antibiotic A 40926
UA41283C2 (uk) * 1991-07-29 2001-09-17 Біосерч Італіа С.П.А. Похідні антибіотику а 40926 та способи їх одержання
US5840684A (en) * 1994-01-28 1998-11-24 Eli Lilly And Company Glycopeptide antibiotic derivatives
MY128335A (en) 1994-01-28 2007-01-31 Lilly Co Eli Glycopeptide antibiotic derivatives
US5918873A (en) * 1995-03-30 1999-07-06 Canon Kabushiki Kaisha Sheet supplying apparatus which regulates tip end of sheet by first and second abutment means
US5919756A (en) 1996-06-28 1999-07-06 Eli Lilly And Company Amides
US5939382A (en) 1996-11-21 1999-08-17 Eli Lilly And Company Reducing agent for reductive alkylation of glycopeptide antibiotics
US5952466A (en) * 1997-11-12 1999-09-14 Eli Lilly And Company Reductive alkylation of glycopeptide antibiotics
US5916873A (en) 1997-04-17 1999-06-29 Eli Lilly And Company Teicoplanin derivatives
US6518242B1 (en) * 1998-02-20 2003-02-11 Theravance, Inc. Derivatives of glycopeptide antibacterial agents
IT1307018B1 (it) 1998-02-20 2001-10-23 Advanced Medicine Inc Agenti antibatterici.
CN1249081C (zh) 1998-12-23 2006-04-05 施万制药 糖肽衍生物或含有它们的药物组合物
EP1173193A4 (en) 1999-04-02 2003-01-29 Univ Princeton DES-LEUCYL GLYCOPEPTIDE ANTIBIOTICS AND METHOD OF PREPARATION
WO2001057071A2 (en) 2000-02-04 2001-08-09 Advanced Medicine, Inc. Glycopeptide derivatives having antibiotic activity
CA2726789A1 (en) * 2000-02-05 2001-11-08 Theravance, Inc. Cyclodextrin containing glycopeptide antibiotic compositions
CA2407994C (en) * 2000-05-02 2010-02-02 Advanced Medecine Inc. Reductive alkylation process
UA75083C2 (uk) 2000-06-22 2006-03-15 Тераванс, Інк. Похідні глікопептидфосфонатів

Also Published As

Publication number Publication date
AU2002324768A1 (en) 2003-03-10
CN1281619C (zh) 2006-10-25
KR20040028997A (ko) 2004-04-03
US7015305B2 (en) 2006-03-21
ATE360029T1 (de) 2007-05-15
DE60219638D1 (de) 2007-05-31
EP1419174A4 (en) 2005-10-12
EP1419174B1 (en) 2007-04-18
TWI312785B (en) 2009-08-01
KR100909435B1 (ko) 2009-07-28
CA2457215C (en) 2011-12-13
US7160984B2 (en) 2007-01-09
CA2457215A1 (en) 2003-03-06
ES2284907T3 (es) 2007-11-16
WO2003018607A3 (en) 2003-11-27
CN1610692A (zh) 2005-04-27
US20030045457A1 (en) 2003-03-06
DE60219638T2 (de) 2007-12-20
WO2003018607A2 (en) 2003-03-06
JP4116546B2 (ja) 2008-07-09
US20060058503A1 (en) 2006-03-16
NO335304B1 (no) 2014-11-10
JP2005525997A (ja) 2005-09-02
EP1419174A2 (en) 2004-05-19
NO20040779L (no) 2004-02-23

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