DK139940B - Analogifremgangsmåde til fremstilling af benzimidazolforbindelser eller syreadditionssalte eller metaladditionsforbindelser deraf. - Google Patents

Analogifremgangsmåde til fremstilling af benzimidazolforbindelser eller syreadditionssalte eller metaladditionsforbindelser deraf.

Info

Publication number
DK139940B
DK139940B DK41168AA DK41168A DK139940B DK 139940 B DK139940 B DK 139940B DK 41168A A DK41168A A DK 41168AA DK 41168 A DK41168 A DK 41168A DK 139940 B DK139940 B DK 139940B
Authority
DK
Denmark
Prior art keywords
compounds
preparation
analogous process
acid addition
addition salts
Prior art date
Application number
DK41168AA
Other languages
Danish (da)
English (en)
Other versions
DK139940C (fr
Inventor
Dale Richard Hoff
Michael Herbert Fisher
Original Assignee
Merck & Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck & Co Inc filed Critical Merck & Co Inc
Publication of DK139940B publication Critical patent/DK139940B/da
Application granted granted Critical
Publication of DK139940C publication Critical patent/DK139940C/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4151,2-Diazoles
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/04Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/04Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • EFIXED CONSTRUCTIONS
    • E21EARTH OR ROCK DRILLING; MINING
    • E21DSHAFTS; TUNNELS; GALLERIES; LARGE UNDERGROUND CHAMBERS
    • E21D11/00Lining tunnels, galleries or other underground cavities, e.g. large underground chambers; Linings therefor; Making such linings in situ, e.g. by assembling
    • E21D11/14Lining predominantly with metal
    • E21D11/28Longitudinal struts, i.e. longitudinal connections between adjoining arches

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Health & Medical Sciences (AREA)
  • Mining & Mineral Resources (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Geology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Life Sciences & Earth Sciences (AREA)
  • Geochemistry & Mineralogy (AREA)
  • Civil Engineering (AREA)
  • Architecture (AREA)
  • Medicinal Chemistry (AREA)
  • Structural Engineering (AREA)
  • Epidemiology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
DK41168AA 1967-02-03 1968-02-02 Analogifremgangsmåde til fremstilling af benzimidazolforbindelser eller syreadditionssalte eller metaladditionsforbindelser deraf. DK139940B (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US61374667A 1967-02-03 1967-02-03
US69649668A 1968-01-09 1968-01-09

Publications (2)

Publication Number Publication Date
DK139940B true DK139940B (da) 1979-05-21
DK139940C DK139940C (fr) 1979-10-15

Family

ID=27087090

Family Applications (1)

Application Number Title Priority Date Filing Date
DK41168AA DK139940B (da) 1967-02-03 1968-02-02 Analogifremgangsmåde til fremstilling af benzimidazolforbindelser eller syreadditionssalte eller metaladditionsforbindelser deraf.

Country Status (19)

Country Link
AT (5) AT289833B (fr)
BE (2) BE710081A (fr)
CH (5) CH545294A (fr)
CS (1) CS162651B2 (fr)
CY (1) CY653A (fr)
DE (2) DE1695545C3 (fr)
DK (1) DK139940B (fr)
ES (4) ES350083A1 (fr)
FI (1) FI52859C (fr)
FR (1) FR1580153A (fr)
GB (2) GB1198941A (fr)
IE (1) IE31812B1 (fr)
IT (1) IT1044176B (fr)
NL (1) NL157015B (fr)
NO (1) NO126484B (fr)
OA (1) OA04036A (fr)
SE (1) SE346321B (fr)
SU (1) SU540569A3 (fr)
YU (1) YU33831B (fr)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3711608A (en) * 1971-04-13 1973-01-16 Merck & Co Inc The treatment of pain, fever and inflammation with benzimidazoles
US3985755A (en) * 1972-06-02 1976-10-12 E. R. Squibb & Sons, Inc. Pyridine containing isothiocyanobenzoxazoles
US3983130A (en) * 1972-06-02 1976-09-28 E. R. Squibb & Sons, Inc. Anthelmintic isothiocyanobenzoxazoles
US3853894A (en) * 1972-06-02 1974-12-10 Squibb & Sons Inc Isothiocyanobenzimidazoles
MA19290A1 (fr) * 1980-05-22 1982-04-01 Ciba Geigy Ag Derives du benzole,leur preparaton et leur utilisations therapeutiques .
SE8604566D0 (sv) * 1986-10-27 1986-10-27 Haessle Ab Novel compunds
US7622592B2 (en) 2002-11-01 2009-11-24 Merck & Co., Inc. Carbonylamino-benzimidazole derivatives as androgen receptor modulators
GB0324792D0 (en) 2003-10-23 2003-11-26 Sterix Ltd Compound
WO2005042513A1 (fr) * 2003-10-23 2005-05-12 Sterix Limited Derives de carboxamide de phenyle et de sulfonamide utilisables comme 11-beta-hydroxysteroide deshydrogenase

Also Published As

Publication number Publication date
DE1795711A1 (de) 1974-02-28
BE735281A (fr) 1969-12-29
DE1695545B2 (de) 1978-08-31
DE1795711B2 (de) 1978-09-21
CY653A (en) 1972-08-31
CH509318A (de) 1971-06-30
CH545295A (de) 1974-01-31
BE710081A (fr) 1968-07-30
IE31812B1 (en) 1973-01-10
SE346321B (fr) 1972-07-03
FI52859B (fr) 1977-08-31
NL157015B (nl) 1978-06-15
GB1198942A (en) 1970-07-15
CH545293A (de) 1974-01-31
AT289835B (de) 1971-05-10
AT293378B (de) 1971-10-11
AT301244B (de) 1972-08-25
ES363761A1 (es) 1970-12-16
IE31812L (en) 1968-08-03
DE1695545C3 (de) 1979-05-03
DK139940C (fr) 1979-10-15
OA04036A (fr) 1979-09-30
ES363760A1 (es) 1970-12-16
ES363762A1 (es) 1970-12-16
YU33831B (en) 1978-06-30
FI52859C (fi) 1977-12-12
AT289833B (de) 1971-05-10
NO126484B (fr) 1973-02-12
CH545294A (de) 1974-01-31
GB1198941A (en) 1970-07-15
NL6801482A (fr) 1968-08-05
YU21268A (en) 1977-12-31
DE1695545A1 (de) 1971-05-06
CH545796A (fr) 1974-02-15
AT289828B (de) 1971-05-10
SU540569A3 (ru) 1976-12-25
IT1044176B (it) 1980-03-20
CS162651B2 (fr) 1975-07-15
DE1795711C3 (de) 1979-05-17
FR1580153A (fr) 1969-09-05
ES350083A1 (es) 1969-11-16

Similar Documents

Publication Publication Date Title
DK124942B (da) Analogifremgangsmåde til fremstilling af alkanolaminderivater eller syreadditionssalte deraf.
DK119153B (da) Analogifremgangsmåde til fremstilling af 3-benzoyl-phenyleddikesyre-derivater eller salte deraf.
DK124884B (da) Analogifremgangsmåde til fremstilling af 2-brom-α-ergokryptin eller syreadditionssalte deraf.
DK120750B (da) Analogifremgangsmåde til fremstilling af azaspiroalkandion-forbindelser eller syreadditionssalte deraf.
DK115473B (da) Fremgangsmåde til fremstilling af 2,3,4,5-tetrahydro-1H-3-benzazepiner eller syreadditionssalte deraf.
DK123022B (da) Analogifremgangsmåde til fremstilling af amino-monohalogen-phenylethanolaminer eller syreadditionssalte deraf.
DK120400B (da) Analogifremgangsmåde til fremstilling af 1-(3,5-dihalogen-4-hydroxyphenyl)-2-(2-phenoxy- eller 2-phenylalkyl-isopropylamino)-propanoler eller syreadditionssalte deraf.
DK129238B (da) Fremgangsmåde til fremstilling af morphinanderivater eller syreadditionssalte deraf.
DK118607B (da) Analogifremgangsmåde til fremstilling af 2-phenylhydrazino-imidazolin-2-forbindelser eller syreadditionssalte deraf.
DK131935B (da) Analogifremgangsmåde til fremstilling af aminoalkynyllaktamforbindelser eller syreadditionssalte deraf.
DK118187B (da) Fremgangsmåde til fremstilling af indolderivater eller syreadditionssalte deraf.
DK139940B (da) Analogifremgangsmåde til fremstilling af benzimidazolforbindelser eller syreadditionssalte eller metaladditionsforbindelser deraf.
DK127644B (da) Analogifremgangsmåde til fremstilling af ergopeptiner eller syreadditionssalte deraf.
DK129448B (da) Analogifremgangsmåde til fremstilling af bis-(benzylidenamino)-guanidiner eller syreadditionssalte deraf.
DK117425B (da) Fremgangsmåde til fremstilling af heterocyclisk substituerede hydrazino-imidazoliner-(2) eller syreadditionssalte deraf.
DK120155B (da) Analogifremgangsmåde til fremstilling af aminopropiofenoner eller syreadditionssalte deraf.
DK127331B (da) Analogifremgangsmåde til fremstilling af aryloxyisoalkyl-Δ<2>-imidazoliner eller syreadditionssalte heraf.
DK130587B (da) Analogifremgangsmåde til fremstilling af difenylpyridazoner eller syreadditionssalt deraf.
DK137674B (da) Analogifremgangsmåde til fremstilling af monophenylsubstituerede oxazoler eller syreadditionssalte deraf.
DK126781B (da) Analogifremgangsmåde til fremstilling af pyrrolidinoguanidinforbindelser eller syreadditionssalte deraf.
DK125129B (da) Analogifremgangsmåde til fremstilling af oximderivater eller syreadditionssalte deraf.
DK124944B (da) Analogifremgangsmåde til fremstilling af substituerede 2-arylalkyloxybenzamider eller syreadditionssalte eller kvaternære ammoniumsalter deraf.
DK140591B (da) Analogifremgangsmåde til fremstilling af cyclopeptider eller syreadditionssalte deraf.
DK128813B (da) Analogifremgangsmåde til fremstilling af basisk substituerede thiophthalaner eller syreadditionssalte deraf.
DK123227B (da) Analogifremgangsmåde til fremstilling af substituerede 3-phenylindanforbindelser eller syreadditionssalte deraf.

Legal Events

Date Code Title Description
PBP Patent lapsed