DK1389207T3 - Polymorfe og andre krystallinske former af cis-FTC - Google Patents

Polymorfe og andre krystallinske former af cis-FTC

Info

Publication number
DK1389207T3
DK1389207T3 DK02748367T DK02748367T DK1389207T3 DK 1389207 T3 DK1389207 T3 DK 1389207T3 DK 02748367 T DK02748367 T DK 02748367T DK 02748367 T DK02748367 T DK 02748367T DK 1389207 T3 DK1389207 T3 DK 1389207T3
Authority
DK
Denmark
Prior art keywords
ftc
cis
forms
manufacture
polymorphic
Prior art date
Application number
DK02748367T
Other languages
Danish (da)
English (en)
Inventor
Kenneth R Phares
Devalina Law
Yuerong Hu
Original Assignee
Gilead Sciences Inc
Abbott Lab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Gilead Sciences Inc, Abbott Lab filed Critical Gilead Sciences Inc
Application granted granted Critical
Publication of DK1389207T3 publication Critical patent/DK1389207T3/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D411/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen and sulfur atoms as the only ring hetero atoms
    • C07D411/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen and sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D411/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen and sulfur atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/18—Antivirals for RNA viruses for HIV
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/20—Antivirals for DNA viruses
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/20—Antivirals for DNA viruses
    • A61P31/22—Antivirals for DNA viruses for herpes viruses

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Virology (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Molecular Biology (AREA)
  • Engineering & Computer Science (AREA)
  • Biotechnology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • AIDS & HIV (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
DK02748367T 2001-03-01 2002-03-01 Polymorfe og andre krystallinske former af cis-FTC DK1389207T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US27256001P 2001-03-01 2001-03-01
US30960501P 2001-08-02 2001-08-02

Publications (1)

Publication Number Publication Date
DK1389207T3 true DK1389207T3 (da) 2006-04-18

Family

ID=26955597

Family Applications (2)

Application Number Title Priority Date Filing Date
DK02748367T DK1389207T3 (da) 2001-03-01 2002-03-01 Polymorfe og andre krystallinske former af cis-FTC
DK05076347T DK1574512T3 (da) 2001-03-01 2002-03-01 Polymorfe og andre krystallinske former af cis-FTC

Family Applications After (1)

Application Number Title Priority Date Filing Date
DK05076347T DK1574512T3 (da) 2001-03-01 2002-03-01 Polymorfe og andre krystallinske former af cis-FTC

Country Status (14)

Country Link
US (3) US6723728B2 (enExample)
EP (3) EP1574512B1 (enExample)
JP (4) JP5105689B2 (enExample)
KR (4) KR101015510B1 (enExample)
CN (4) CN102911166B (enExample)
AT (2) ATE383355T1 (enExample)
AU (1) AU2002335489B2 (enExample)
CA (4) CA2788498C (enExample)
CY (2) CY1107983T1 (enExample)
DE (2) DE60224592T2 (enExample)
DK (2) DK1389207T3 (enExample)
ES (3) ES2253544T3 (enExample)
PT (2) PT1574512E (enExample)
WO (1) WO2002070518A1 (enExample)

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* Cited by examiner, † Cited by third party
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PT1583542E (pt) 2003-01-14 2008-09-17 Gilead Sciences Inc Composições e métodos para terapia de combinação antiviral
US6943249B2 (en) * 2003-03-17 2005-09-13 Ash Stevens, Inc. Methods for isolating crystalline Form I of 5-azacytidine
US6887855B2 (en) 2003-03-17 2005-05-03 Pharmion Corporation Forms of 5-azacytidine
US20060014949A1 (en) * 2004-07-13 2006-01-19 Supergen Inc. Compositions and formulations of decitabine polymorphs and methods of use thereof
TWI375560B (en) 2005-06-13 2012-11-01 Gilead Sciences Inc Composition comprising dry granulated emtricitabine and tenofovir df and method for making the same
TWI471145B (zh) 2005-06-13 2015-02-01 Bristol Myers Squibb & Gilead Sciences Llc 單一式藥學劑量型
WO2009005338A2 (en) * 2007-07-05 2009-01-08 Ultimorphix Technologies B.V. Solid forms ult-i, ult-2 and ult-3 of emtricitabine
US20110288298A1 (en) 2008-11-12 2011-11-24 Lupin Limited novel polymorph of emtricitabine and a process for preparing of the same
US8710218B2 (en) 2009-07-15 2014-04-29 Lupin Limited Process for preparation of Efavirenz

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Also Published As

Publication number Publication date
CA2867970A1 (en) 2002-09-12
CA2788498C (en) 2016-02-16
KR20080065317A (ko) 2008-07-11
JP2009197005A (ja) 2009-09-03
ATE383355T1 (de) 2008-01-15
US6723728B2 (en) 2004-04-20
US7544692B2 (en) 2009-06-09
AU2002335489B2 (en) 2008-06-05
CA2788498A1 (en) 2002-09-12
CN1503796B (zh) 2012-07-04
ES2253544T3 (es) 2006-06-01
WO2002070518A1 (en) 2002-09-12
CA2439831C (en) 2010-01-12
CA2690137A1 (en) 2002-09-12
DK1574512T3 (da) 2008-03-03
EP1903041A3 (en) 2008-04-23
US20030060645A1 (en) 2003-03-27
EP1389207A1 (en) 2004-02-18
CN102911165A (zh) 2013-02-06
CN102911165B (zh) 2016-08-17
CA2439831A1 (en) 2002-09-12
KR101150250B1 (ko) 2012-06-12
EP1903041A2 (en) 2008-03-26
EP1574512A1 (en) 2005-09-14
EP1903041B1 (en) 2015-02-18
CN102911166A (zh) 2013-02-06
KR20040002871A (ko) 2004-01-07
PT1903041E (pt) 2015-06-23
DE60207850D1 (de) 2006-01-12
DE60207850T2 (de) 2006-08-10
CN1503796A (zh) 2004-06-09
JP2004530660A (ja) 2004-10-07
JP5105689B2 (ja) 2012-12-26
ES2299950T3 (es) 2008-06-01
KR100927024B1 (ko) 2009-11-17
DE60224592D1 (de) 2008-02-21
CY1107983T1 (el) 2013-09-04
EP1574512B1 (en) 2008-01-09
DE60224592T2 (de) 2009-01-29
US20090306114A1 (en) 2009-12-10
US20050026934A1 (en) 2005-02-03
PT1574512E (pt) 2008-03-05
CN102911166B (zh) 2016-08-17
KR101015510B1 (ko) 2011-02-16
ATE312097T1 (de) 2005-12-15
CN102942563A (zh) 2013-02-27
EP1389207B1 (en) 2005-12-07
US8637535B2 (en) 2014-01-28
KR20080065316A (ko) 2008-07-11
CY1107913T1 (el) 2013-09-04
ES2537007T3 (es) 2015-06-01
CA2690137C (en) 2012-11-13
JP2015028045A (ja) 2015-02-12
KR20100091265A (ko) 2010-08-18
JP2013040192A (ja) 2013-02-28

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