PT1574512E - Formas polimórficas e outras formas cristalinas de cis-ftc - Google Patents

Formas polimórficas e outras formas cristalinas de cis-ftc Download PDF

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Publication number
PT1574512E
PT1574512E PT05076347T PT05076347T PT1574512E PT 1574512 E PT1574512 E PT 1574512E PT 05076347 T PT05076347 T PT 05076347T PT 05076347 T PT05076347 T PT 05076347T PT 1574512 E PT1574512 E PT 1574512E
Authority
PT
Portugal
Prior art keywords
ftc
cis
forms
manufacture
polymorphic
Prior art date
Application number
PT05076347T
Other languages
English (en)
Portuguese (pt)
Inventor
Devalina Law
Kenneth R Phares
Yuerong Hu
Original Assignee
Abbott Lab
Gilead Sciences Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Abbott Lab, Gilead Sciences Inc filed Critical Abbott Lab
Publication of PT1574512E publication Critical patent/PT1574512E/pt

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D411/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen and sulfur atoms as the only ring hetero atoms
    • C07D411/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen and sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D411/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen and sulfur atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/18—Antivirals for RNA viruses for HIV
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/20—Antivirals for DNA viruses
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/20—Antivirals for DNA viruses
    • A61P31/22—Antivirals for DNA viruses for herpes viruses

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Virology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Engineering & Computer Science (AREA)
  • Molecular Biology (AREA)
  • Biotechnology (AREA)
  • AIDS & HIV (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
PT05076347T 2001-03-01 2002-03-01 Formas polimórficas e outras formas cristalinas de cis-ftc PT1574512E (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US27256001P 2001-03-01 2001-03-01
US30960501P 2001-08-02 2001-08-02

Publications (1)

Publication Number Publication Date
PT1574512E true PT1574512E (pt) 2008-03-05

Family

ID=26955597

Family Applications (2)

Application Number Title Priority Date Filing Date
PT05076347T PT1574512E (pt) 2001-03-01 2002-03-01 Formas polimórficas e outras formas cristalinas de cis-ftc
PT80002645T PT1903041E (pt) 2001-03-01 2002-03-01 Formas polimórficas e outras formas cristalinas de cis-ftc

Family Applications After (1)

Application Number Title Priority Date Filing Date
PT80002645T PT1903041E (pt) 2001-03-01 2002-03-01 Formas polimórficas e outras formas cristalinas de cis-ftc

Country Status (14)

Country Link
US (3) US6723728B2 (enExample)
EP (3) EP1574512B1 (enExample)
JP (4) JP5105689B2 (enExample)
KR (4) KR101015510B1 (enExample)
CN (4) CN102942563A (enExample)
AT (2) ATE383355T1 (enExample)
AU (1) AU2002335489B2 (enExample)
CA (4) CA2788498C (enExample)
CY (2) CY1107983T1 (enExample)
DE (2) DE60224592T2 (enExample)
DK (2) DK1574512T3 (enExample)
ES (3) ES2537007T3 (enExample)
PT (2) PT1574512E (enExample)
WO (1) WO2002070518A1 (enExample)

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* Cited by examiner, † Cited by third party
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DE60224592T2 (de) * 2001-03-01 2009-01-29 Abbott Laboratories, Abbott Park Polymorphe und andere kristalline Formen von cis-FTC
TWI244393B (en) * 2002-08-06 2005-12-01 Idenix Pharmaceuticals Inc Crystalline and amorphous forms of beta-L-2'-deoxythymidine
NZ540728A (en) 2003-01-14 2008-08-29 Gilead Sciences Inc Compositions and methods for combination antiviral therapy
US6887855B2 (en) 2003-03-17 2005-05-03 Pharmion Corporation Forms of 5-azacytidine
US6943249B2 (en) * 2003-03-17 2005-09-13 Ash Stevens, Inc. Methods for isolating crystalline Form I of 5-azacytidine
US20060014949A1 (en) * 2004-07-13 2006-01-19 Supergen Inc. Compositions and formulations of decitabine polymorphs and methods of use thereof
TWI375560B (en) 2005-06-13 2012-11-01 Gilead Sciences Inc Composition comprising dry granulated emtricitabine and tenofovir df and method for making the same
TWI471145B (zh) 2005-06-13 2015-02-01 Bristol Myers Squibb & Gilead Sciences Llc 單一式藥學劑量型
WO2009005338A2 (en) * 2007-07-05 2009-01-08 Ultimorphix Technologies B.V. Solid forms ult-i, ult-2 and ult-3 of emtricitabine
EP2350065A1 (en) 2008-11-12 2011-08-03 Lupin Ltd. A novel polymorph of emtricitabine and a process for preparing of the same
EP2454244B1 (en) 2009-07-15 2013-06-26 Lupin Limited An improved process for preparation of efavirenz

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Also Published As

Publication number Publication date
DE60224592D1 (de) 2008-02-21
JP2013040192A (ja) 2013-02-28
ATE383355T1 (de) 2008-01-15
CA2690137C (en) 2012-11-13
EP1574512A1 (en) 2005-09-14
CN1503796A (zh) 2004-06-09
JP2009197005A (ja) 2009-09-03
EP1903041B1 (en) 2015-02-18
KR101015510B1 (ko) 2011-02-16
US20090306114A1 (en) 2009-12-10
CA2690137A1 (en) 2002-09-12
DK1574512T3 (da) 2008-03-03
CA2788498A1 (en) 2002-09-12
CN102911165A (zh) 2013-02-06
CA2788498C (en) 2016-02-16
PT1903041E (pt) 2015-06-23
JP5105689B2 (ja) 2012-12-26
DE60207850T2 (de) 2006-08-10
DE60224592T2 (de) 2009-01-29
US7544692B2 (en) 2009-06-09
DK1389207T3 (da) 2006-04-18
ES2253544T3 (es) 2006-06-01
DE60207850D1 (de) 2006-01-12
EP1389207B1 (en) 2005-12-07
EP1574512B1 (en) 2008-01-09
KR101150250B1 (ko) 2012-06-12
US8637535B2 (en) 2014-01-28
KR20080065316A (ko) 2008-07-11
ES2299950T3 (es) 2008-06-01
WO2002070518A1 (en) 2002-09-12
CA2439831C (en) 2010-01-12
AU2002335489B2 (en) 2008-06-05
US6723728B2 (en) 2004-04-20
CY1107983T1 (el) 2013-09-04
EP1903041A2 (en) 2008-03-26
ES2537007T3 (es) 2015-06-01
US20030060645A1 (en) 2003-03-27
CA2439831A1 (en) 2002-09-12
KR100927024B1 (ko) 2009-11-17
CN102911165B (zh) 2016-08-17
ATE312097T1 (de) 2005-12-15
KR20040002871A (ko) 2004-01-07
JP2004530660A (ja) 2004-10-07
US20050026934A1 (en) 2005-02-03
CN102911166A (zh) 2013-02-06
KR20080065317A (ko) 2008-07-11
CY1107913T1 (el) 2013-09-04
CA2867970A1 (en) 2002-09-12
JP2015028045A (ja) 2015-02-12
EP1903041A3 (en) 2008-04-23
CN102942563A (zh) 2013-02-27
EP1389207A1 (en) 2004-02-18
CN102911166B (zh) 2016-08-17
KR20100091265A (ko) 2010-08-18
CN1503796B (zh) 2012-07-04

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