DK138460B - Analogifremgangsmåde til fremstilling af 2beta, 16beta-diamino-3alfa, 17beta-diacyloxy-5alfa-androstanderivater eller syreadditionssalte eller di- eller monokvaternære derivater deraf. - Google Patents

Analogifremgangsmåde til fremstilling af 2beta, 16beta-diamino-3alfa, 17beta-diacyloxy-5alfa-androstanderivater eller syreadditionssalte eller di- eller monokvaternære derivater deraf.

Info

Publication number
DK138460B
DK138460B DK340976AA DK340976A DK138460B DK 138460 B DK138460 B DK 138460B DK 340976A A DK340976A A DK 340976AA DK 340976 A DK340976 A DK 340976A DK 138460 B DK138460 B DK 138460B
Authority
DK
Denmark
Prior art keywords
derivatives
16beta
monoquaternary
2beta
3alpha
Prior art date
Application number
DK340976AA
Other languages
English (en)
Other versions
DK340976A (da
DK138460C (da
Inventor
Zoltan Tuba
Maria Marsai
Katalin Biro
Laszlo Szporny
Egon Karpati
Szabolcs Szeberenyi
Original Assignee
Richter Gedeon Vegyeszet
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Richter Gedeon Vegyeszet filed Critical Richter Gedeon Vegyeszet
Publication of DK340976A publication Critical patent/DK340976A/da
Publication of DK138460B publication Critical patent/DK138460B/da
Application granted granted Critical
Publication of DK138460C publication Critical patent/DK138460C/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J41/00Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0005Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring the nitrogen atom being directly linked to the cyclopenta(a)hydro phenanthrene skeleton
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00Drugs for disorders of the muscular or neuromuscular system
    • A61P21/02Muscle relaxants, e.g. for tetanus or cramps
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J13/00Normal steroids containing carbon, hydrogen, halogen or oxygen having a carbon-to-carbon double bond from or to position 17
    • C07J13/005Normal steroids containing carbon, hydrogen, halogen or oxygen having a carbon-to-carbon double bond from or to position 17 with double bond in position 16 (17)
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J43/00Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C07J43/003Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton not condensed
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J71/00Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
    • C07J71/0005Oxygen-containing hetero ring
    • C07J71/001Oxiranes

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Pain & Pain Management (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DK340976AA 1975-08-01 1976-07-29 Analogifremgangsmåde til fremstilling af 2beta, 16beta-diamino-3alfa, 17beta-diacyloxy-5alfa-androstanderivater eller syreadditionssalte eller di- eller monokvaternære derivater deraf. DK138460B (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
HU75RI00000575A HU172522B (hu) 1975-08-01 1975-08-01 Sposob poluchenija novykh proizvodnykh 2beta, 16beta-diamino-androstana i ikh chetvertichnykh solej

Publications (3)

Publication Number Publication Date
DK340976A DK340976A (da) 1977-02-02
DK138460B true DK138460B (da) 1978-09-11
DK138460C DK138460C (da) 1979-02-12

Family

ID=11000984

Family Applications (1)

Application Number Title Priority Date Filing Date
DK340976AA DK138460B (da) 1975-08-01 1976-07-29 Analogifremgangsmåde til fremstilling af 2beta, 16beta-diamino-3alfa, 17beta-diacyloxy-5alfa-androstanderivater eller syreadditionssalte eller di- eller monokvaternære derivater deraf.

Country Status (19)

Country Link
US (1) US4101545A (da)
AT (1) AT359218B (da)
AU (1) AU499988B2 (da)
BE (1) BE844643A (da)
CA (1) CA1084044A (da)
CS (1) CS189782B2 (da)
DD (1) DD126820A5 (da)
DE (1) DE2634336C3 (da)
DK (1) DK138460B (da)
FR (1) FR2319370A1 (da)
GB (1) GB1540405A (da)
HU (1) HU172522B (da)
IL (1) IL50099A (da)
NL (1) NL185079C (da)
PL (1) PL101306B1 (da)
RO (1) RO75980A (da)
SE (1) SE409867B (da)
SU (1) SU1001859A3 (da)
YU (1) YU187776A (da)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ATE921T1 (de) * 1978-09-05 1982-05-15 Akzo N.V. Saeureadditionssalze von 2-beta, 16-beta-bis-piperidino-an drostan-16-beta-monoquaternaeren ammoniumderivaten und diese enthaltende pharmazeutische zusammensetzungen.
DE2944212C3 (de) * 1978-11-03 1994-10-20 Papst Motoren Gmbh & Co Kg Magnetplattenantrieb
IE50675B1 (en) * 1979-12-12 1986-06-11 Akzo Nv Bis-and mono-quaternary ammonium derivatives of 2beta,16beta-dipiperidino-5alpha-androstanes,processes for their preparation and pharmaceutical preparations
HU195972B (en) * 1985-07-01 1988-08-29 Richter Gedeon Vegyeszet Process for producing new diamino-androstane derivatives and pharmaceutical compositions containing them
US5380840A (en) * 1985-09-12 1995-01-10 The Upjohn Company Triazinylpiperazinyl steroids
US5099019A (en) * 1985-09-12 1992-03-24 Upjohn Company Amines useful in producing pharmaceutically active CNS compounds
USRE35053E (en) * 1985-09-12 1995-10-10 The Upjohn Company Amines useful in producing pharmaceutically active CNS compounds
IT1277700B1 (it) * 1995-12-22 1997-11-11 Poli Ind Chimica Spa Processo di preparazione di 2-beta, 16-beta-diamino 3-alfa, 17-beta- diacilossi 5-alfaandrostani, bloccanti neuromuscolari a struttura

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1138605A (en) * 1965-02-19 1969-01-01 Organon Labor Ltd Improvements in or relating to new 2-ß,16-ß-diamino-androstanes
HU168431B (da) * 1972-07-27 1976-04-28

Also Published As

Publication number Publication date
YU187776A (en) 1982-05-31
DK340976A (da) 1977-02-02
GB1540405A (en) 1979-02-14
HU172522B (hu) 1978-09-28
BE844643A (fr) 1976-11-16
NL7608538A (nl) 1977-02-03
US4101545A (en) 1978-07-18
DD126820A5 (da) 1977-08-17
RO75980A (ro) 1981-08-17
AT359218B (de) 1980-10-27
DK138460C (da) 1979-02-12
DE2634336B2 (de) 1978-03-23
NL185079B (nl) 1989-08-16
PL101306B1 (pl) 1978-12-30
IL50099A0 (en) 1976-09-30
AU1612576A (en) 1978-01-26
ATA564176A (de) 1980-03-15
SU1001859A3 (ru) 1983-02-28
FR2319370B1 (da) 1980-07-25
SE409867B (sv) 1979-09-10
IL50099A (en) 1980-02-29
DE2634336C3 (de) 1978-11-23
CS189782B2 (en) 1979-04-30
FR2319370A1 (fr) 1977-02-25
NL185079C (nl) 1990-01-16
AU499988B2 (en) 1979-05-10
DE2634336A1 (de) 1977-02-03
SE7608608L (sv) 1977-02-02
CA1084044A (en) 1980-08-19

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