DK135374B - Analogifremgangsmåde til fremstilling af 2,4-diamino-5-benzylpyrimidiner eller syreadditionssalte deraf. - Google Patents
Analogifremgangsmåde til fremstilling af 2,4-diamino-5-benzylpyrimidiner eller syreadditionssalte deraf.Info
- Publication number
- DK135374B DK135374B DK374174AA DK374174A DK135374B DK 135374 B DK135374 B DK 135374B DK 374174A A DK374174A A DK 374174AA DK 374174 A DK374174 A DK 374174A DK 135374 B DK135374 B DK 135374B
- Authority
- DK
- Denmark
- Prior art keywords
- benzylpyrimidines
- diamino
- preparation
- acid addition
- addition salts
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
- C07D239/48—Two nitrogen atoms
- C07D239/49—Two nitrogen atoms with an aralkyl radical, or substituted aralkyl radical, attached in position 5, e.g. trimethoprim
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C229/00—Compounds containing amino and carboxyl groups bound to the same carbon skeleton
- C07C229/38—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino groups bound to acyclic carbon atoms and carboxyl groups bound to carbon atoms of six-membered aromatic rings of the same carbon skeleton
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C255/00—Carboxylic acid nitriles
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
- C07C45/51—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by pyrolysis, rearrangement or decomposition
- C07C45/511—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by pyrolysis, rearrangement or decomposition involving transformation of singly bound oxygen functional groups to >C = O groups
- C07C45/515—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by pyrolysis, rearrangement or decomposition involving transformation of singly bound oxygen functional groups to >C = O groups the singly bound functional group being an acetalised, ketalised hemi-acetalised, or hemi-ketalised hydroxyl group
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
- C07C45/61—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
- C07C45/67—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton
- C07C45/673—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by change of size of the carbon skeleton
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D265/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
- C07D265/28—1,4-Oxazines; Hydrogenated 1,4-oxazines
- C07D265/30—1,4-Oxazines; Hydrogenated 1,4-oxazines not condensed with other rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
- C07D295/14—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D295/145—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals with the ring nitrogen atoms and the carbon atoms with three bonds to hetero atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Priority Applications (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DK374175A DK134549B (da) | 1973-07-27 | 1975-08-19 | Analogifremgangsmåde til fremstilling af 2,4-diamino-5-benzylpyrimidiner eller syreadditionssalte deraf. |
| DK188376A DK188376A (da) | 1973-07-27 | 1976-04-27 | 2,4-diamino-5-benzylpyrimidiner samt preparat indeholdende disse forbindelser |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CH1099573A CH598231A5 (da) | 1973-07-27 | 1973-07-27 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| DK374174A DK374174A (da) | 1975-04-01 |
| DK135374B true DK135374B (da) | 1977-04-18 |
| DK135374C DK135374C (da) | 1977-10-03 |
Family
ID=4368954
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK374174AA DK135374B (da) | 1973-07-27 | 1974-07-11 | Analogifremgangsmåde til fremstilling af 2,4-diamino-5-benzylpyrimidiner eller syreadditionssalte deraf. |
Country Status (11)
| Country | Link |
|---|---|
| JP (1) | JPS5041876A (da) |
| BE (1) | BE818131A (da) |
| CA (1) | CA1026759A (da) |
| CH (1) | CH598231A5 (da) |
| DE (1) | DE2435934A1 (da) |
| DK (1) | DK135374B (da) |
| FR (1) | FR2238496B1 (da) |
| GB (5) | GB1455738A (da) |
| NL (1) | NL7410100A (da) |
| SE (1) | SE415975B (da) |
| ZA (1) | ZA744512B (da) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA1084498A (en) | 1977-05-05 | 1980-08-26 | Alexander E. Wick | Benzylpyrimidines and process for the preparation thereof |
| HU188588B (en) * | 1982-08-13 | 1986-04-28 | Egyt Gyogyszervegyeszeti Gyar | Process for the production of 2,4-diamino-5-benzyl-pyrimidine-derivatives |
| MX2007014928A (es) | 2005-06-02 | 2008-02-15 | Hoffmann La Roche | Derivados de piperidin-4-il-amida y su uso como antagonistas de subtipo 5 del receptor de somatostatina. |
| US7855194B2 (en) | 2006-03-27 | 2010-12-21 | Hoffmann-La Roche Inc. | Pyrimidine, quinazoline, pteridine and triazine derivatives |
-
1973
- 1973-07-27 CH CH1099573A patent/CH598231A5/xx not_active IP Right Cessation
-
1974
- 1974-07-11 DK DK374174AA patent/DK135374B/da not_active IP Right Cessation
- 1974-07-15 ZA ZA00744512A patent/ZA744512B/xx unknown
- 1974-07-19 FR FR7425210A patent/FR2238496B1/fr not_active Expired
- 1974-07-25 DE DE2435934A patent/DE2435934A1/de not_active Ceased
- 1974-07-26 CA CA205,706A patent/CA1026759A/en not_active Expired
- 1974-07-26 SE SE7409733A patent/SE415975B/xx unknown
- 1974-07-26 GB GB456076A patent/GB1455738A/en not_active Expired
- 1974-07-26 GB GB456176A patent/GB1455739A/en not_active Expired
- 1974-07-26 JP JP49085239A patent/JPS5041876A/ja active Pending
- 1974-07-26 GB GB455976A patent/GB1455737A/en not_active Expired
- 1974-07-26 BE BE146980A patent/BE818131A/xx not_active IP Right Cessation
- 1974-07-26 GB GB456276A patent/GB1455740A/en not_active Expired
- 1974-07-26 GB GB3316974A patent/GB1455736A/en not_active Expired
- 1974-07-26 NL NL7410100A patent/NL7410100A/xx not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| SE415975B (sv) | 1980-11-17 |
| GB1455740A (en) | 1976-11-17 |
| DE2435934A1 (de) | 1975-02-13 |
| FR2238496B1 (da) | 1977-09-09 |
| NL7410100A (nl) | 1975-01-29 |
| DK374174A (da) | 1975-04-01 |
| AU7148874A (en) | 1976-01-22 |
| GB1455736A (en) | 1976-11-17 |
| JPS5041876A (da) | 1975-04-16 |
| FR2238496A1 (da) | 1975-02-21 |
| DK135374C (da) | 1977-10-03 |
| GB1455739A (en) | 1976-11-17 |
| BE818131A (fr) | 1975-01-27 |
| CA1026759A (en) | 1978-02-21 |
| ZA744512B (en) | 1975-09-24 |
| SE7409733L (da) | 1975-01-28 |
| CH598231A5 (da) | 1978-04-28 |
| GB1455737A (en) | 1976-11-17 |
| GB1455738A (en) | 1976-11-17 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PBP | Patent lapsed |