DK134489B - Fremgangsmåde til fremstilling af alkyl-7-desoxy-7(S)-substituerede-alfa-thiolincosaminider. - Google Patents

Fremgangsmåde til fremstilling af alkyl-7-desoxy-7(S)-substituerede-alfa-thiolincosaminider.

Info

Publication number
DK134489B
DK134489B DK155471AA DK155471A DK134489B DK 134489 B DK134489 B DK 134489B DK 155471A A DK155471A A DK 155471AA DK 155471 A DK155471 A DK 155471A DK 134489 B DK134489 B DK 134489B
Authority
DK
Denmark
Prior art keywords
thiolincosaminides
deoxy
alpha
substituted
alkyl
Prior art date
Application number
DK155471AA
Other languages
Danish (da)
English (en)
Other versions
DK134489C (de
Inventor
Brian Bannister
Original Assignee
Upjohn Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Upjohn Co filed Critical Upjohn Co
Priority to DK229072A priority Critical patent/DK135536B/da
Publication of DK134489B publication Critical patent/DK134489B/da
Application granted granted Critical
Publication of DK134489C publication Critical patent/DK134489C/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C08—ORGANIC MACROMOLECULAR COMPOUNDS; THEIR PREPARATION OR CHEMICAL WORKING-UP; COMPOSITIONS BASED THEREON
    • C08G—MACROMOLECULAR COMPOUNDS OBTAINED OTHERWISE THAN BY REACTIONS ONLY INVOLVING UNSATURATED CARBON-TO-CARBON BONDS
    • C08G18/00—Polymeric products of isocyanates or isothiocyanates
    • C08G18/06—Polymeric products of isocyanates or isothiocyanates with compounds having active hydrogen
    • C08G18/28—Polymeric products of isocyanates or isothiocyanates with compounds having active hydrogen characterised by the compounds used containing active hydrogen
    • C08G18/30—Low-molecular-weight compounds
    • C08G18/38—Low-molecular-weight compounds having heteroatoms other than oxygen
    • C08G18/3855—Low-molecular-weight compounds having heteroatoms other than oxygen having sulfur
    • C08G18/3863—Low-molecular-weight compounds having heteroatoms other than oxygen having sulfur containing groups having sulfur atoms between two carbon atoms, the sulfur atoms being directly linked to carbon atoms or other sulfur atoms
    • C08G18/3865—Low-molecular-weight compounds having heteroatoms other than oxygen having sulfur containing groups having sulfur atoms between two carbon atoms, the sulfur atoms being directly linked to carbon atoms or other sulfur atoms containing groups having one sulfur atom between two carbon atoms
    • C08G18/3868—Low-molecular-weight compounds having heteroatoms other than oxygen having sulfur containing groups having sulfur atoms between two carbon atoms, the sulfur atoms being directly linked to carbon atoms or other sulfur atoms containing groups having one sulfur atom between two carbon atoms the sulfur atom belonging to a sulfide group
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/02—Acyclic radicals, not substituted by cyclic structures
    • C07H15/14—Acyclic radicals, not substituted by cyclic structures attached to a sulfur, selenium or tellurium atom of a saccharide radical
    • C07H15/16—Lincomycin; Derivatives thereof

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biotechnology (AREA)
  • Medicinal Chemistry (AREA)
  • Crystallography & Structural Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biochemistry (AREA)
  • Polymers & Plastics (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Cephalosporin Compounds (AREA)
DK155471AA 1970-04-06 1971-03-31 Fremgangsmåde til fremstilling af alkyl-7-desoxy-7(S)-substituerede-alfa-thiolincosaminider. DK134489B (da)

Priority Applications (1)

Application Number Priority Date Filing Date Title
DK229072A DK135536B (da) 1970-04-06 1972-05-08 Fremgangsmåde til fremstilling af N-acyl-6,7-aziridino-6-desamino-7-desoxy-alfa-thiolincosaminider.

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US2611970A 1970-04-06 1970-04-06

Publications (2)

Publication Number Publication Date
DK134489B true DK134489B (da) 1976-11-15
DK134489C DK134489C (de) 1977-04-25

Family

ID=21830031

Family Applications (1)

Application Number Title Priority Date Filing Date
DK155471AA DK134489B (da) 1970-04-06 1971-03-31 Fremgangsmåde til fremstilling af alkyl-7-desoxy-7(S)-substituerede-alfa-thiolincosaminider.

Country Status (14)

Country Link
US (1) US3702322A (de)
JP (1) JPS5527071B1 (de)
BE (1) BE765370A (de)
CA (1) CA945149A (de)
CH (2) CH554858A (de)
DE (4) DE2167182C3 (de)
DK (1) DK134489B (de)
ES (1) ES389524A1 (de)
FR (1) FR2092009B1 (de)
GB (1) GB1311438A (de)
IL (1) IL36435A (de)
NL (1) NL170960C (de)
SE (2) SE385011B (de)
ZA (1) ZA711709B (de)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3853843A (en) * 1972-12-13 1974-12-10 Upjohn Co Derivatives of thiolincosaminide compounds
US3870699A (en) * 1973-03-06 1975-03-11 Upjohn Co Lincomycin analogs
CA2458644A1 (en) * 2001-08-28 2003-03-13 Pharmacia Corporation Crystaline clindamycin free base
US7199105B2 (en) * 2002-08-15 2007-04-03 Vicuron Pharmaceuticals, Inc. Lincomycin derivatives possessing antibacterial activity
EP1529052A2 (de) * 2002-08-15 2005-05-11 Vicuron Pharmaceuticals, Inc. Lincomycinderivate mit antibakterieller aktivität
US7199106B2 (en) 2003-06-17 2007-04-03 Vicuron Pharmaceuticals, Inc. Lincomycin derivatives possessing antimicrobial activity
US7256177B2 (en) 2003-06-17 2007-08-14 Vicuron Pharmaceuticals, Inc. Lincomycin derivatives possessing antibacterial activity
US7361743B2 (en) * 2004-02-11 2008-04-22 Pfizer Inc Lincomycin derivatives possessing antibacterial activity

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR1467501A (fr) * 1965-10-20 1967-01-27 Upjohn Co 7-halogéno-7-deoxylincomycine et 7-halogéno-7-dexoyepilincomycine, leurs analogues et isomères et leurs procédés de fabrication

Also Published As

Publication number Publication date
US3702322A (en) 1972-11-07
DE2167180C3 (de) 1981-07-30
DE2116066C3 (de) 1980-11-13
DE2167181B1 (de) 1980-11-27
NL170960C (nl) 1983-01-17
DE2116066B2 (de) 1980-01-17
ZA711709B (en) 1972-01-26
DK134489C (de) 1977-04-25
SE385011B (sv) 1976-05-31
SE409209B (sv) 1979-08-06
BE765370A (fr) 1971-10-06
DE2116066A1 (de) 1971-11-04
NL170960B (nl) 1982-08-16
JPS5527071B1 (de) 1980-07-17
DE2167181C3 (de) 1981-07-02
GB1311438A (en) 1973-03-28
CA945149A (en) 1974-04-09
DE2167182C3 (de) 1981-09-17
DE2167182B1 (de) 1981-01-08
CH556325A (de) 1974-11-29
CH554858A (de) 1974-10-15
IL36435A0 (en) 1971-05-26
IL36435A (en) 1975-04-25
FR2092009B1 (de) 1974-09-27
DE2167180B1 (de) 1980-12-18
NL7104221A (de) 1971-10-08
FR2092009A1 (de) 1972-01-21
ES389524A1 (es) 1974-03-16

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